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Low dose Oliceridine — Competitive Intelligence Brief
marketed
Mu-opioid receptor agonist
Mu-opioid receptor (OPRM1)
Pain Management
Small molecule
Live · refreshed every 30 min
Target snapshot
Low dose Oliceridine (Low dose Oliceridine) — Nanjing First Hospital, Nanjing Medical University. Low-dose oliceridine is a selective mu-opioid receptor agonist that provides analgesia with potentially reduced adverse effects compared to standard-dose opioids.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Low dose Oliceridine TARGET | Low dose Oliceridine | Nanjing First Hospital, Nanjing Medical University | marketed | Mu-opioid receptor agonist | Mu-opioid receptor (OPRM1) | |
| Viberzi | ELUXADOLINE | AbbVie | marketed | mu-Opioid Receptor Agonist [EPC] | Mu-type opioid receptor | 2015-01-01 |
| Tapentadol Prolonged Release | Tapentadol Prolonged Release | Grünenthal GmbH | marketed | Mu-opioid receptor agonist and noradrenaline reuptake inhibitor | Mu-opioid receptor; noradrenaline transporter (NET) | |
| Use of buprenorphine with FAO > 30 OME | Use of buprenorphine with FAO > 30 OME | Fox Chase Cancer Center | marketed | Partial mu-opioid receptor agonist | Mu-opioid receptor (μ-OR) | |
| opana then placebo then darvocet | opana then placebo then darvocet | University of Rochester | marketed | Opioid analgesic (mu-opioid receptor agonist) | Mu-opioid receptor | |
| High dose Oliceridine | High dose Oliceridine | Nanjing First Hospital, Nanjing Medical University | marketed | Mu-opioid receptor agonist (biased agonist) | Mu-opioid receptor (OPRM1) | |
| TM buprenorphine | TM buprenorphine | Indivior Inc. | marketed | Partial mu-opioid receptor agonist | Mu-opioid receptor (OPRM1) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Mu-opioid receptor agonist class)
- Nanjing First Hospital, Nanjing Medical University · 1 drug in this class
- Xiangya Hospital of Central South University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Low dose Oliceridine — Competitive Intelligence Brief. https://druglandscape.com/ci/low-dose-oliceridine. Accessed 2026-06-10.
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