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Levocetirizine only — Competitive Intelligence Brief
marketed
H1-receptor antagonist (second-generation antihistamine)
H1 receptor
Allergy/Immunology
Small molecule
Live · refreshed every 30 min
Target snapshot
Levocetirizine only (Levocetirizine only) — University Hospital, Grenoble. Levocetirizine is a selective H1-receptor antagonist that blocks histamine signaling to reduce allergic symptoms.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Levocetirizine only TARGET | Levocetirizine only | University Hospital, Grenoble | marketed | H1-receptor antagonist (second-generation antihistamine) | H1 receptor | |
| Lastacaft | ALCAFTADINE | AbbVie | marketed | Histamine-1 Receptor Antagonist [EPC] | Histamine H1 receptor | 2010-01-01 |
| Xyzal | LEVOCETIRIZINE | Sanofi | marketed | Histamine-1 Receptor Antagonist | Histamine H1 receptor | 2007-01-01 |
| Elestat | EPINASTINE | AbbVie | marketed | Adrenergic Receptor Agonist | Histamine H1 receptor | 2003-01-01 |
| Rupax | RUPATADINE | Teikoku Seiyaku | marketed | rupatadine | Histamine H1 receptor | 2001-01-01 |
| Zaditor | KETOTIFEN | marketed | Histamine-1 Receptor Inhibitor | Histamine H1 receptor | 1999-01-01 | |
| Mizollen | MIZOLASTINE | Sanofi | marketed | mizolastine | Histamine H1 receptor | 1998-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (H1-receptor antagonist (second-generation antihistamine) class)
- UCB Pharma · 5 drugs in this class
- Organon and Co · 3 drugs in this class
- Brian J Lipworth · 1 drug in this class
- GlaxoSmithKline · 1 drug in this class
- Goldman, Butterwick, Fitzpatrick and Groff · 1 drug in this class
- HK inno.N Corporation · 1 drug in this class
- AAADRS Clinical Research Center · 1 drug in this class
- University Hospital, Grenoble · 1 drug in this class
- Azienda Ospedaliera OO.RR. S. Giovanni di Dio e Ruggi D'Aragona · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Levocetirizine only — Competitive Intelligence Brief. https://druglandscape.com/ci/levocetirizine-only. Accessed 2026-05-15.
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