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INR101 — Competitive Intelligence Brief
phase 3
Vitamin K antagonist
VKORC1
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
INR101 (INR101) — Yunhe Pharmaceutical (Tianjin) Co., Ltd. INR101 is an anticoagulant that works by inhibiting the synthesis of vitamin K-dependent clotting factors.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| INR101 TARGET | INR101 | Yunhe Pharmaceutical (Tianjin) Co., Ltd | phase 3 | Vitamin K antagonist | VKORC1 | |
| PHYTONADIONE | PHYTONADIONE | marketed | Vitamin K [EPC] | Vitamin K epoxide reductase complex subunit 1 (VKORC1) | 1982-01-01 | |
| Warfarin or coumadin | Warfarin or coumadin | Ottawa Heart Institute Research Corporation | marketed | Vitamin K antagonist (oral anticoagulant) | Vitamin K epoxide reductase complex 1 (VKORC1) | |
| Warfarin duration | Warfarin duration | British Thoracic Society | marketed | Vitamin K antagonist (anticoagulant) | Vitamin K epoxide reductase complex 1 (VKORC1) | |
| Warfarin (Coumadin) | Warfarin (Coumadin) | University of Michigan | marketed | Vitamin K antagonist (oral anticoagulant) | Vitamin K epoxide reductase (VKORC1) | |
| Sodium warfarin | Sodium warfarin | University of Padova | marketed | Vitamin K antagonist (coumarin anticoagulant) | Vitamin K epoxide reductase complex 1 (VKORC1) | |
| Standard dose oral anticoagulant | Standard dose oral anticoagulant | Korea University Guro Hospital | marketed | Vitamin K antagonist (warfarin-type oral anticoagulant) | Vitamin K epoxide reductase complex 1 (VKORC1) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Vitamin K antagonist class)
- Joon Bum Kim · 1 drug in this class
- Population Health Research Institute · 1 drug in this class
- US Department of Veterans Affairs · 1 drug in this class
- University Hospital, Bonn · 1 drug in this class
- University Hospital, Limoges · 1 drug in this class
- Yunhe Pharmaceutical (Tianjin) Co., Ltd · 1 drug in this class
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- Whole Vitamin K antagonist class — RSS
Cite this brief
Drug Landscape (2026). INR101 — Competitive Intelligence Brief. https://druglandscape.com/ci/inr101. Accessed 2026-05-13.
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