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INR101 — Competitive Intelligence Brief

INR101 (INR101) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Vitamin K antagonist. Area: Cardiovascular.

phase 3 Vitamin K antagonist VKORC1 Cardiovascular Small molecule Live · refreshed every 30 min

Target snapshot

INR101 (INR101) — Yunhe Pharmaceutical (Tianjin) Co., Ltd. INR101 is an anticoagulant that works by inhibiting the synthesis of vitamin K-dependent clotting factors.

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
INR101 TARGET INR101 Yunhe Pharmaceutical (Tianjin) Co., Ltd phase 3 Vitamin K antagonist VKORC1
PHYTONADIONE PHYTONADIONE marketed Vitamin K [EPC] Vitamin K epoxide reductase complex subunit 1 (VKORC1) 1982-01-01
Warfarin or coumadin Warfarin or coumadin Ottawa Heart Institute Research Corporation marketed Vitamin K antagonist (oral anticoagulant) Vitamin K epoxide reductase complex 1 (VKORC1)
Warfarin duration Warfarin duration British Thoracic Society marketed Vitamin K antagonist (anticoagulant) Vitamin K epoxide reductase complex 1 (VKORC1)
Warfarin (Coumadin) Warfarin (Coumadin) University of Michigan marketed Vitamin K antagonist (oral anticoagulant) Vitamin K epoxide reductase (VKORC1)
Sodium warfarin Sodium warfarin University of Padova marketed Vitamin K antagonist (coumarin anticoagulant) Vitamin K epoxide reductase complex 1 (VKORC1)
Standard dose oral anticoagulant Standard dose oral anticoagulant Korea University Guro Hospital marketed Vitamin K antagonist (warfarin-type oral anticoagulant) Vitamin K epoxide reductase complex 1 (VKORC1)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Vitamin K antagonist class)

  1. Joon Bum Kim · 1 drug in this class
  2. Population Health Research Institute · 1 drug in this class
  3. US Department of Veterans Affairs · 1 drug in this class
  4. University Hospital, Bonn · 1 drug in this class
  5. University Hospital, Limoges · 1 drug in this class
  6. Yunhe Pharmaceutical (Tianjin) Co., Ltd · 1 drug in this class

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Cite this brief

Drug Landscape (2026). INR101 — Competitive Intelligence Brief. https://druglandscape.com/ci/inr101. Accessed 2026-05-13.

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