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Indacaterol/glycopyrronium — Competitive Intelligence Brief
marketed
Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination)
Beta-2 adrenergic receptor; M3 muscarinic acetylcholine receptor
Respiratory / Pulmonology
Small molecule
Live · refreshed every 30 min
Target snapshot
Indacaterol/glycopyrronium (Indacaterol/glycopyrronium) — Orion Corporation, Orion Pharma. Indacaterol is a long-acting beta-2 agonist that stimulates airway smooth muscle relaxation, while glycopyrronium is an anticholinergic that blocks muscarinic receptors to further dilate airways.
Comparator set (5 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Indacaterol/glycopyrronium TARGET | Indacaterol/glycopyrronium | Orion Corporation, Orion Pharma | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic acetylcholine receptor | |
| Albuterol, ipratropium bromide | Albuterol, ipratropium bromide | Children's Hospital of Philadelphia | marketed | Combination bronchodilator (beta-2 agonist + anticholinergic) | Beta-2 adrenergic receptor; M3 muscarinic acetylcholine receptor | |
| Anoro® Ellipta® | Anoro® Ellipta® | AstraZeneca | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor and M3 muscarinic acetylcholine receptor | |
| Olodaterol-Tiotropium | Olodaterol-Tiotropium | Fraunhofer-Institute of Toxicology and Experimental Medicine | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic receptor | |
| indacaterol/glycopyrronium 110/50 Breezhaler® | indacaterol/glycopyrronium 110/50 Breezhaler® | Wouter H. van Geffen | marketed | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; Muscarinic M3 acetylcholine receptor | |
| FF/GW642444 Inhalation Powder | FF/GW642444 Inhalation Powder | GlaxoSmithKline | phase 3 | Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) | Beta-2 adrenergic receptor; M3 muscarinic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Long-acting beta-2 agonist / Long-acting muscarinic antagonist (LABA/LAMA combination) class)
- AstraZeneca · 1 drug in this class
- Fraunhofer-Institute of Toxicology and Experimental Medicine · 1 drug in this class
- GlaxoSmithKline · 1 drug in this class
- Orion Corporation, Orion Pharma · 1 drug in this class
- Wouter H. van Geffen · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Indacaterol/glycopyrronium — Competitive Intelligence Brief. https://druglandscape.com/ci/indacaterol-glycopyrronium. Accessed 2026-05-16.
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