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Gilteritinib + Azacitidine + Venetoclax — Competitive Intelligence Brief

Gilteritinib + Azacitidine + Venetoclax (Gilteritinib + Azacitidine + Venetoclax) competitive landscape: 0 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination. Area: Oncology.

phase 3 FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination FLT3, DNA methyltransferase, BCL-2 Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Gilteritinib + Azacitidine + Venetoclax (Gilteritinib + Azacitidine + Venetoclax) — Institute of Hematology & Blood Diseases Hospital, China. This triple combination targets acute myeloid leukemia by inhibiting FLT3 signaling (gilteritinib), promoting DNA methylation-dependent differentiation (azacitidine), and blocking anti-apoptotic BCL-2 proteins (venetoclax).

Comparator set

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Gilteritinib + Azacitidine + Venetoclax TARGET Gilteritinib + Azacitidine + Venetoclax Institute of Hematology & Blood Diseases Hospital, China phase 3 FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination FLT3, DNA methyltransferase, BCL-2

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination class)

  1. Institute of Hematology & Blood Diseases Hospital, China · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Gilteritinib + Azacitidine + Venetoclax — Competitive Intelligence Brief. https://druglandscape.com/ci/gilteritinib-azacitidine-venetoclax. Accessed 2026-05-17.

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