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Gilteritinib + Azacitidine + Venetoclax — Competitive Intelligence Brief
phase 3
FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination
FLT3, DNA methyltransferase, BCL-2
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Gilteritinib + Azacitidine + Venetoclax (Gilteritinib + Azacitidine + Venetoclax) — Institute of Hematology & Blood Diseases Hospital, China. This triple combination targets acute myeloid leukemia by inhibiting FLT3 signaling (gilteritinib), promoting DNA methylation-dependent differentiation (azacitidine), and blocking anti-apoptotic BCL-2 proteins (venetoclax).
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Gilteritinib + Azacitidine + Venetoclax TARGET | Gilteritinib + Azacitidine + Venetoclax | Institute of Hematology & Blood Diseases Hospital, China | phase 3 | FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination | FLT3, DNA methyltransferase, BCL-2 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (FLT3 inhibitor + hypomethylating agent + BCL-2 inhibitor combination class)
- Institute of Hematology & Blood Diseases Hospital, China · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Gilteritinib + Azacitidine + Venetoclax — Competitive Intelligence Brief. https://druglandscape.com/ci/gilteritinib-azacitidine-venetoclax. Accessed 2026-05-17.
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