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Drug: dorzolamide/timolol — Competitive Intelligence Brief
marketed
Carbonic anhydrase inhibitor / Beta-blocker combination
Carbonic anhydrase II / Beta-adrenergic receptors (β1 and β2)
Ophthalmology
Small molecule
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Target snapshot
Drug: dorzolamide/timolol (Drug: dorzolamide/timolol) — Aristotle University Of Thessaloniki. Dorzolamide inhibits carbonic anhydrase to reduce aqueous humor production, while timolol blocks beta-adrenergic receptors to further decrease intraocular pressure.
Comparator set (2 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Drug: dorzolamide/timolol TARGET | Drug: dorzolamide/timolol | Aristotle University Of Thessaloniki | marketed | Carbonic anhydrase inhibitor / Beta-blocker combination | Carbonic anhydrase II / Beta-adrenergic receptors (β1 and β2) | |
| tafluprost and dorzolamide/timolol | tafluprost and dorzolamide/timolol | Aristotle University Of Thessaloniki | marketed | Prostaglandin analogue / carbonic anhydrase inhibitor / beta-blocker combination | Prostaglandin F receptor (FP receptor), carbonic anhydrase II, beta-1 and beta-2 adrenergic receptors | |
| treatment with dorzolamide/timolol | treatment with dorzolamide/timolol | Aristotle University Of Thessaloniki | marketed | Carbonic anhydrase inhibitor / Beta-blocker combination | Carbonic anhydrase II; Beta-adrenergic receptors (β1 and β2) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Carbonic anhydrase inhibitor / Beta-blocker combination class)
- Aristotle University Of Thessaloniki · 2 drugs in this class
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Cite this brief
Drug Landscape (2026). Drug: dorzolamide/timolol — Competitive Intelligence Brief. https://druglandscape.com/ci/drug-dorzolamide-timolol. Accessed 2026-05-17.
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