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Pulmonary Arterial Hypertension (PAH) — Treatment Landscape & Competitive Intelligence
Cardiovascular
10 marketed
0 Phase 3
0 Phase 2
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Marketed treatment landscape
| Drug | Generic | Sponsor | Class | Target | Line of therapy | First approval |
|---|---|---|---|---|---|---|
| Uptravi | SELEXIPAG | AstraZeneca | Prostacyclin Receptor Agonist [EPC] | Prostacyclin receptor | 2015-01-01 | |
| Opsumit | MACITENTAN | AstraZeneca | Endothelin Receptor Antagonist [EPC] | Endothelin-1 receptor | 2013-01-01 | |
| Adempas | RIOCIGUAT | Bayer | Soluble Guanylate Cyclase Stimulator [EPC] | Guanylate cyclase soluble subunit beta-1 | 2013-01-01 | |
| Letairis | AMBRISENTAN | Gilead Sciences | Endothelin Receptor Antagonist [EPC] | Endothelin-1 receptor | 2007-01-01 | |
| Remodulin | TREPROSTINIL | United Therap | Prostacycline Vasodilator [EPC] | Prostacyclin receptor | 2002-01-01 | |
| Tracleer | BOSENTAN | AstraZeneca | Endothelin Receptor Antagonist | Endothelin-1 receptor | 2001-01-01 | |
| Viagra | sildenafil | Pfizer Inc. | PDE5 inhibitor | Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A, High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A, Multidrug resistance-associated protein 5 | 1998-03-27 | |
| Flolan | EPOPROSTENOL | AstraZeneca | Prostacycline Vasodilator [EPC] | Prostacyclin receptor | 1995-01-01 | |
| prostacyclin | prostacyclin | United Therapeutics | P2Y purinoceptor 12, Prostacyclin receptor, Prostaglandin E2 receptor EP1 subtype | |||
| Revatio | Sildenafil Citrate | Pfizer Inc. | PDE5 inhibitor | Phosphodiesterase type 5 (PDE5) |
Phase 3 pipeline
Phase 2 pipeline
Recent regulatory actions (last 90 days)
- — Tracleer · FDA · approved · US
Upcoming PDUFA dates (next 180 days)
Sponsor landscape
- AstraZeneca · 4 drugs in Pulmonary Arterial Hypertension (PAH)
- Pfizer Inc. · 2 drugs in Pulmonary Arterial Hypertension (PAH)
- Gilead Sciences · 1 drug in Pulmonary Arterial Hypertension (PAH)
- Meshalkin Research Institute of Pathology of Circulation · 1 drug in Pulmonary Arterial Hypertension (PAH)
- Pfizer · 1 drug in Pulmonary Arterial Hypertension (PAH)
- Prim PD Dr Afshin Assadian · 1 drug in Pulmonary Arterial Hypertension (PAH)
- United Therap · 1 drug in Pulmonary Arterial Hypertension (PAH)
- United Therapeutics · 1 drug in Pulmonary Arterial Hypertension (PAH)
- · 1 drug in Pulmonary Arterial Hypertension (PAH)
- University of Colorado, Denver · 1 drug in Pulmonary Arterial Hypertension (PAH)
- Bayer · 1 drug in Pulmonary Arterial Hypertension (PAH)
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Cite this brief
Drug Landscape (2026). Pulmonary Arterial Hypertension (PAH) — Treatment Landscape & Competitive Intelligence Brief. https://druglandscape.com/ci/disease/pulmonary-arterial-hypertension. Accessed 2026-05-16.
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