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Bladder muscle dysfunction - overactive — Treatment Landscape & Competitive Intelligence
10 marketed
0 Phase 3
0 Phase 2
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Marketed treatment landscape
| Drug | Generic | Sponsor | Class | Target | Line of therapy | First approval |
|---|---|---|---|---|---|---|
| Myrbetriq | MIRABEGRON | Apgdi | beta3-Adrenergic Agonist [EPC] | Beta-3 adrenergic receptor | 2012-01-01 | |
| Toviaz | Fesoterodine Fumarate | Pfizer | fesoterodine | Muscarinic acetylcholine receptor M2 | 2008-01-01 | |
| Toviaz | FESOTERODINE | Pfizer | fesoterodine | Muscarinic acetylcholine receptor M2 | 2008-01-01 | |
| Vesicare | SOLIFENACIN | Astellas Pharma | Cholinergic Muscarinic Antagonist | Muscarinic acetylcholine receptor M1 | 2004-01-01 | |
| Sanctura | TROSPIUM | AbbVie | Cholinergic Muscarinic Antagonist | Muscarinic acetylcholine receptor M3 | 2004-01-01 | |
| Enablex | DARIFENACIN | AbbVie | Cholinergic Muscarinic Antagonist | Muscarinic acetylcholine receptor M3 | 2004-01-01 | |
| Detrol | TOLTERODINE | Upjohn | Cholinergic Muscarinic Antagonist | Muscarinic acetylcholine receptor M1 | 1998-01-01 | |
| Ditropan Xl | OXYBUTYNIN | Hisamitsu Pharmaceutical Co., Inc. | Cholinergic Muscarinic Antagonist | Muscarinic acetylcholine receptor M3 | 1975-01-01 | |
| Oxytrol | Oxytrol | Jewish General Hospital | Cytochrome P450 2C19, 5-hydroxytryptamine receptor 2B, D(3) dopamine receptor | |||
| Vesicare | Vesicare | University of California, Irvine | Muscarinic acetylcholine receptor M1, Muscarinic acetylcholine receptor M2, Muscarinic acetylcholine receptor M3 |
Phase 3 pipeline
Phase 2 pipeline
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Sponsor landscape
- Pfizer · 2 drugs in Bladder muscle dysfunction - overactive
- AbbVie · 2 drugs in Bladder muscle dysfunction - overactive
- · 2 drugs in Bladder muscle dysfunction - overactive
- Hisamitsu Pharmaceutical Co., Inc. · 1 drug in Bladder muscle dysfunction - overactive
- Jewish General Hospital · 1 drug in Bladder muscle dysfunction - overactive
- University of California, Irvine · 1 drug in Bladder muscle dysfunction - overactive
- Upjohn · 1 drug in Bladder muscle dysfunction - overactive
- Apgdi · 1 drug in Bladder muscle dysfunction - overactive
- Astellas Pharma · 1 drug in Bladder muscle dysfunction - overactive
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Cite this brief
Drug Landscape (2026). Bladder muscle dysfunction - overactive — Treatment Landscape & Competitive Intelligence Brief. https://druglandscape.com/ci/disease/bladder-muscle-dysfunction-overactive. Accessed 2026-06-10.
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