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DICYCLOMINE — Competitive Intelligence Brief
marketed
Antispasmodic and anticholinergic (antimuscarinic) agent
Muscarinic receptors
Gastroenterology
Small molecule
Live · refreshed every 30 min
Target snapshot
DICYCLOMINE (DICYCLOMINE). Dicyclomine relieves smooth muscle spasm of the gastrointestinal tract via a dual mechanism: anticholinergic effects at acetylcholine receptors and direct smooth muscle relaxation.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| DICYCLOMINE TARGET | DICYCLOMINE | marketed | Antispasmodic and anticholinergic (antimuscarinic) agent | Muscarinic receptors | 1950-01-01 | |
| SOLIFENACIN SUCCINATE | SOLIFENACIN SUCCINATE | marketed | Muscarinic receptors | 2004-01-01 | ||
| Tolterodine 6 | Tolterodine 6 | KYU-SUNG LEE | marketed | Muscarinic receptor antagonist | M2 and M3 muscarinic receptors | |
| Tolterodine Tartrate ER | Tolterodine Tartrate ER | University of California, San Francisco | marketed | Muscarinic receptor antagonist | M2 and M3 muscarinic receptors | |
| Aceclidin | ACECLIDINE | marketed | aceclidine | muscarinic receptors | ||
| Xanomeline and Trospium Chloride | Xanomeline and Trospium Chloride | Collaborative Neuroscience Research, LLC | marketed | Muscarinic M1/M4 receptor agonist with peripheral anticholinergic antagonist | Muscarinic acetylcholine receptors M1 and M4 (xanomeline); muscarinic receptors peripherally (trospium chloride antagonism) | |
| Tropicamide Ophthalmic | Tropicamide Ophthalmic | Semnan University of Medical Sciences | phase 3 | Anticholinergic | Muscarinic receptors |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Antispasmodic and anticholinergic (antimuscarinic) agent class)
- · 1 drug in this class
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Cite this brief
Drug Landscape (2026). DICYCLOMINE — Competitive Intelligence Brief. https://druglandscape.com/ci/dicyclomine. Accessed 2026-05-14.
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