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Decitabine/Cedazuridine — Competitive Intelligence Brief
phase 3
DNA methyltransferase inhibitor; hypomethylating agent
DNA methyltransferase (DNMT)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Decitabine/Cedazuridine (Decitabine/Cedazuridine) — Astex Pharmaceuticals, Inc.. Decitabine is a DNA methyltransferase inhibitor that causes hypomethylation of DNA, leading to reactivation of silenced tumor suppressor genes and differentiation of myelodysplastic cells.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Decitabine/Cedazuridine TARGET | Decitabine/Cedazuridine | Astex Pharmaceuticals, Inc. | phase 3 | DNA methyltransferase inhibitor; hypomethylating agent | DNA methyltransferase (DNMT) | |
| Azacitidine Injection | Azacitidine Injection | Ascentage Pharma Group Inc. | marketed | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) | |
| Azacitidine (AZA) | Azacitidine (AZA) | Memorial Sloan Kettering Cancer Center | marketed | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) | |
| decitabine injection | decitabine injection | Janssen Korea, Ltd., Korea | marketed | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) | |
| Azacytidine, HAG Regimen | Azacytidine, HAG Regimen | Shenzhen Second People's Hospital | marketed | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) | |
| 5-Azacytidin | 5-Azacytidin | Technische Universität Dresden | phase 3 | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) | |
| Dacogen (decitabine) only | Dacogen (decitabine) only | Eisai Inc. | phase 3 | DNA methyltransferase inhibitor | DNA methyltransferase (DNMT) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (DNA methyltransferase inhibitor; hypomethylating agent class)
- Astex Pharmaceuticals, Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Decitabine/Cedazuridine — Competitive Intelligence Brief. https://druglandscape.com/ci/decitabine-cedazuridine. Accessed 2026-06-10.
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