Last reviewed · How we verify
Cinarizine — Competitive Intelligence Brief
phase 2
cinnarizine
Histamine H1 receptor
Neuroscience
Small molecule
Live · refreshed every 30 min
Target snapshot
Cinarizine (CINNARIZINE). Cinarizine works by blocking histamine receptors in the brain, which helps to reduce symptoms of motion sickness and vertigo.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Cinarizine TARGET | CINNARIZINE | phase 2 | cinnarizine | Histamine H1 receptor | ||
| Lastacaft | ALCAFTADINE | AbbVie | marketed | Histamine-1 Receptor Antagonist [EPC] | Histamine H1 receptor | 2010-01-01 |
| Xyzal | LEVOCETIRIZINE | Sanofi | marketed | Histamine-1 Receptor Antagonist | Histamine H1 receptor | 2007-01-01 |
| Elestat | EPINASTINE | AbbVie | marketed | Adrenergic Receptor Agonist | Histamine H1 receptor | 2003-01-01 |
| Rupax | RUPATADINE | Teikoku Seiyaku | marketed | rupatadine | Histamine H1 receptor | 2001-01-01 |
| Zaditor | KETOTIFEN | marketed | Histamine-1 Receptor Inhibitor | Histamine H1 receptor | 1999-01-01 | |
| Mizollen | MIZOLASTINE | Sanofi | marketed | mizolastine | Histamine H1 receptor | 1998-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (cinnarizine class)
- · 1 drug in this class
Subscribe to ongoing alerts
Push every new event for this competitive set into your RSS reader, IFTTT/Zapier workflow, or email digest:
- Cinarizine CI watch — RSS
- Cinarizine CI watch — Atom
- Cinarizine CI watch — JSON
- Cinarizine alone — RSS
- Whole cinnarizine class — RSS
Cite this brief
Drug Landscape (2026). Cinarizine — Competitive Intelligence Brief. https://druglandscape.com/ci/cinnarizine. Accessed 2026-06-10.
Build your own brief
Pick any drug + add comparators:
https://druglandscape.com/ci/{slug}— auto-detected competitorshttps://druglandscape.com/ci/{slug}?vs=drug1,drug2,drug3— explicit comparators- Brand names auto-resolve:
/ci/keytruda→ 301 →/ci/pembrolizumab
Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing