Last reviewed · How we verify
Detantol — Competitive Intelligence Brief
phase 3
bunazosin
Alpha-1A adrenergic receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Detantol (BUNAZOSIN). Detanidol works by blocking the alpha-1A adrenergic receptor, which helps to relax blood vessels and lower blood pressure.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Detantol TARGET | BUNAZOSIN | phase 3 | bunazosin | Alpha-1A adrenergic receptor | ||
| Dexmedetomidine Hydrochloride | dexmedetomidine-hydrochloride | Pfizer | marketed | dexmedetomidine | Alpha-1A adrenergic receptor | 1999-01-01 |
| Levadil | DILEVALOL | marketed | dilevalol | Alpha-1A adrenergic receptor, Alpha-1B adrenergic receptor, Beta-1 adrenergic receptor | 1990-01-01 | |
| Wellbutrin | bupropion | GSK (GlaxoSmithKline) | marketed | NDRI (Norepinephrine-dopamine reuptake inhibitor) | Cytochrome P450 2C19, Neuronal acetylcholine receptor subunit alpha-7, Alpha-1A adrenergic receptor | 1985-12-30 |
| Hylorel | GUANADREL | Pfizer | marketed | guanadrel | Alpha-1A adrenergic receptor | 1982-01-01 |
| Methoxamin | METHOXAMINE | GSK | marketed | methoxamine | Alpha-1A adrenergic receptor | 1982-01-01 |
| MAPROTILINE | MAPROTILINE | marketed | maprotiline | Alpha-1A adrenergic receptor | 1980-01-01 |
Recent regulatory actions (last 90 days)
- — Dexmedetomidine Hydrochloride · FDA · approved · US · Pfizer
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
- — Dexmedetomidine Hydrochloride · 8242158 · US
- — Dexmedetomidine Hydrochloride · 9616049 · US
- — Dexmedetomidine Hydrochloride · 8648106 · US
- — Dexmedetomidine Hydrochloride · 9320712 · US
- — Dexmedetomidine Hydrochloride · 8455527 · US
- — Dexmedetomidine Hydrochloride · 10016396 · US
- — Dexmedetomidine Hydrochloride · 8338470 · US
- — Dexmedetomidine Hydrochloride · 8242158*PED · US
- — Dexmedetomidine Hydrochloride · 8648106*PED · US
- — Dexmedetomidine Hydrochloride · 8455527*PED · US
- — Dexmedetomidine Hydrochloride · 8338470*PED · US
- — Dexmedetomidine Hydrochloride · 9320712*PED · US
- — Dexmedetomidine Hydrochloride · 9616049*PED · US
- — Dexmedetomidine Hydrochloride · 9717796 · US
- — Dexmedetomidine Hydrochloride · 9649296 · US
- — Dexmedetomidine Hydrochloride · 11517524 · US
- — Dexmedetomidine Hydrochloride · 11497711 · US
- — Dexmedetomidine Hydrochloride · 10792246 · US
- — Dexmedetomidine Hydrochloride · 11478422 · US
Sponsor landscape (bunazosin class)
- · 1 drug in this class
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- Detantol CI watch — RSS
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- Whole bunazosin class — RSS
Cite this brief
Drug Landscape (2026). Detantol — Competitive Intelligence Brief. https://druglandscape.com/ci/bunazosin. Accessed 2026-06-10.
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