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Besifovir dipivoxil — Competitive Intelligence Brief

Besifovir dipivoxil (Besifovir dipivoxil) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Nucleotide reverse transcriptase inhibitor. Area: Virology / Hepatology.

marketed Nucleotide reverse transcriptase inhibitor Hepatitis B virus reverse transcriptase Virology / Hepatology Small molecule Live · refreshed every 30 min

Target snapshot

Besifovir dipivoxil (Besifovir dipivoxil) — IlDong Pharmaceutical Co Ltd. Besifovir dipivoxil is a nucleotide reverse transcriptase inhibitor that blocks hepatitis B virus replication by inhibiting the viral reverse transcriptase enzyme.

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Besifovir dipivoxil TARGET Besifovir dipivoxil IlDong Pharmaceutical Co Ltd marketed Nucleotide reverse transcriptase inhibitor Hepatitis B virus reverse transcriptase
NAs+IFN-α NAs+IFN-α Beijing 302 Hospital marketed Antiviral combination therapy Hepatitis B virus reverse transcriptase; interferon-alpha receptor signaling
Telbivudine treatment Telbivudine treatment Southeast University, China marketed Nucleoside reverse transcriptase inhibitor (NRTI) Hepatitis B virus reverse transcriptase
Tacrolimus &entecavir Tacrolimus &entecavir Guangdong Provincial People's Hospital marketed Combination immunosuppressant and antiviral Calcineurin (tacrolimus); Hepatitis B virus reverse transcriptase (entecavir)
Telbivudine (Standard of Care) Telbivudine (Standard of Care) Nanfang Hospital, Southern Medical University marketed Nucleoside reverse transcriptase inhibitor (NRTI) Hepatitis B virus reverse transcriptase
Telbivudine, Lamivudine, Adefovir ,Enecavir Telbivudine, Lamivudine, Adefovir ,Enecavir Shao-quan Zhang marketed Nucleoside/nucleotide reverse transcriptase inhibitor (NRTI/NtRTI) Hepatitis B virus reverse transcriptase
Blank maleate entecavir tablets Blank maleate entecavir tablets Chia Tai Tianqing Pharmaceutical Group Co., Ltd. marketed Nucleoside reverse transcriptase inhibitor Hepatitis B virus reverse transcriptase

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Nucleotide reverse transcriptase inhibitor class)

  1. GlaxoSmithKline · 2 drugs in this class
  2. IlDong Pharmaceutical Co Ltd · 1 drug in this class
  3. Bristol-Myers Squibb · 1 drug in this class
  4. Merck Sharp & Dohme LLC · 1 drug in this class
  5. National Institute of Allergy and Infectious Diseases (NIAID) · 1 drug in this class
  6. Sun Yat-sen University · 1 drug in this class
  7. Jiangxi Kvvit Pharmaceutical Co., Ltd. · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Besifovir dipivoxil — Competitive Intelligence Brief. https://druglandscape.com/ci/besifovir-dipivoxil. Accessed 2026-05-18.

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