Last reviewed · How we verify
ASP5541 — Competitive Intelligence Brief
phase 2
Complement C5a receptor antagonist
C5a receptor (C5aR)
Immunology
Small molecule
Live · refreshed every 30 min
Target snapshot
ASP5541 (ASP5541) — Astellas Pharma Global Development, Inc.. ASP5541 is a selective antagonist of the complement C5a receptor that inhibits complement-mediated inflammation.
Comparator set (3 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| ASP5541 TARGET | ASP5541 | Astellas Pharma Global Development, Inc. | phase 2 | Complement C5a receptor antagonist | C5a receptor (C5aR) | |
| MP-513 | MP-513 | Tanabe Pharma Corporation | phase 3 | Complement C5a receptor antagonist | C5a receptor (C5aR) | |
| LJPC-501 | LJPC-501 | La Jolla Pharmaceutical Company | phase 3 | Complement C5a receptor antagonist | C5a receptor (C5aR) | |
| KK8398 | KK8398 | Kyowa Kirin Co., Ltd. | phase 3 | Complement C5a receptor antagonist | C5aR1 (C5a receptor 1) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Complement C5a receptor antagonist class)
- Astellas Pharma Global Development, Inc. · 1 drug in this class
- Kyowa Kirin Co., Ltd. · 1 drug in this class
- La Jolla Pharmaceutical Company · 1 drug in this class
- Tanabe Pharma Corporation · 1 drug in this class
Subscribe to ongoing alerts
Push every new event for this competitive set into your RSS reader, IFTTT/Zapier workflow, or email digest:
- ASP5541 CI watch — RSS
- ASP5541 CI watch — Atom
- ASP5541 CI watch — JSON
- ASP5541 alone — RSS
- Whole Complement C5a receptor antagonist class — RSS
Cite this brief
Drug Landscape (2026). ASP5541 — Competitive Intelligence Brief. https://druglandscape.com/ci/asp5541. Accessed 2026-05-13.
Build your own brief
Pick any drug + add comparators:
https://druglandscape.com/ci/{slug}— auto-detected competitorshttps://druglandscape.com/ci/{slug}?vs=drug1,drug2,drug3— explicit comparators- Brand names auto-resolve:
/ci/keytruda→ 301 →/ci/pembrolizumab