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Arotinolol Hydrochloride — Competitive Intelligence Brief
marketed
Alpha-beta blocker
Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Arotinolol Hydrochloride (Arotinolol Hydrochloride) — Sumitomo Pharma (Suzhou) Co., Ltd.. Arotinolol hydrochloride is a non-selective beta-adrenergic receptor antagonist with alpha-1 blocking activity that reduces heart rate and blood pressure.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Arotinolol Hydrochloride TARGET | Arotinolol Hydrochloride | Sumitomo Pharma (Suzhou) Co., Ltd. | marketed | Alpha-beta blocker | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Carvedilol CR | Carvedilol CR | University of Florida | marketed | Non-selective beta-blocker with alpha-1 blocking activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Carvedilol alone | Carvedilol alone | Taipei Veterans General Hospital, Taiwan | marketed | Beta-blocker with alpha-1 antagonist activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Comparator: carvedilol | Comparator: carvedilol | Organon and Co | marketed | Beta-blocker with alpha-1 antagonist activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Beta Blockers Carvedilol Phosphate | Beta Blockers Carvedilol Phosphate | Seoul National University Hospital | marketed | Beta blocker (non-selective, with alpha-1 blocking activity) | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| CarVeDilol-SR (Slow Release) | CarVeDilol-SR (Slow Release) | Seoul National University Bundang Hospital | marketed | Beta-blocker with alpha-1 blocking activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor | |
| Carvedilol IR 25mg, QD | Carvedilol IR 25mg, QD | Chong Kun Dang Pharmaceutical | phase 3 | Beta-blocker with alpha-1 antagonist activity | Beta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Alpha-beta blocker class)
- Sumitomo Pharma (Suzhou) Co., Ltd. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Arotinolol Hydrochloride — Competitive Intelligence Brief. https://druglandscape.com/ci/arotinolol-hydrochloride. Accessed 2026-05-14.
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