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CarVeDilol-SR (Slow Release)

Seoul National University Bundang Hospital · FDA-approved active Small molecule

Carvedilol is a non-selective beta-adrenergic receptor antagonist with alpha-1 blocking activity that reduces heart rate, blood pressure, and cardiac workload.

Carvedilol is a non-selective beta-adrenergic receptor antagonist with alpha-1 blocking activity that reduces heart rate, blood pressure, and cardiac workload. Used for Hypertension, Heart failure with reduced ejection fraction, Left ventricular dysfunction following myocardial infarction.

At a glance

Generic nameCarVeDilol-SR (Slow Release)
SponsorSeoul National University Bundang Hospital
Drug classBeta-blocker with alpha-1 blocking activity
TargetBeta-1 adrenergic receptor, Beta-2 adrenergic receptor, Alpha-1 adrenergic receptor
ModalitySmall molecule
Therapeutic areaCardiovascular
PhaseFDA-approved

Mechanism of action

Carvedilol blocks beta-1 and beta-2 adrenergic receptors as well as alpha-1 adrenergic receptors, reducing sympathetic nervous system activity on the heart and vasculature. The slow-release formulation provides sustained drug delivery over an extended period, allowing for once-daily dosing. This combination of effects reduces cardiac oxygen demand, lowers blood pressure, and improves cardiac efficiency in heart failure and hypertension.

Approved indications

Common side effects

Key clinical trials

Primary sources

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SourceUsed for
ClinicalTrials.govTrial enrolment, design, endpoints, results

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