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ApatinibMesylateTablets — Competitive Intelligence Brief
phase 2
Tyrosine kinase inhibitor
VEGFR2
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
ApatinibMesylateTablets (ApatinibMesylateTablets) — Chang-Ming Huang, Prof.. Tyrosine kinase inhibitor
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| ApatinibMesylateTablets TARGET | ApatinibMesylateTablets | Chang-Ming Huang, Prof. | phase 2 | Tyrosine kinase inhibitor | VEGFR2 | |
| REGORAFENIB | REGORAFENIB | marketed | RET, VEGFR1, VEGFR2, VEGFR3, KIT, PDGFR-alpha, PDGFR-beta, FGFR1, FGFR2, TIE2, DDR2, TrkA, Eph2A, RAF-1, BRAF, BRAF V600E, SAPK2, PTK5, Abl, CSF1R | 2012-01-01 | ||
| Sutent | Sunitinib Malate | Pfizer | marketed | Small molecule kinase inhibitor | Receptor tyrosine kinases (RTKs): PDGFRα, PDGFRβ, VEGFR1, VEGFR2, VEGFR3, KIT, FLT3, CSF-1R, RET | 2006-01-01 |
| Apatinib+Capecitabine | Apatinib+Capecitabine | Huazhong University of Science and Technology | phase 3 | Tyrosine kinase inhibitor + Fluoropyrimidine antimetabolite | VEGFR2 (apatinib); Thymidylate synthase (capecitabine) | |
| Ramucirumab+ paclitaxel | Ramucirumab+ paclitaxel | AstraZeneca | phase 3 | Angiogenesis inhibitor, Microtubule inhibitor | VEGFR2 | |
| Rivoceranib (Apatinib) | Rivoceranib (Apatinib) | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | tyrosine kinase inhibitor | VEGFR2 | |
| Ramucirumab / Paclitaxel/ Docetaxel/ Irinotecan | Ramucirumab / Paclitaxel/ Docetaxel/ Irinotecan | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | Monoclonal antibody (ramucirumab) + chemotherapy combination | VEGF receptor 2 (VEGFR2); tubulin (taxanes) / topoisomerase I (irinotecan) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Tyrosine kinase inhibitor class)
- Jiangsu HengRui Medicine Co., Ltd. · 5 drugs in this class
- Centre Leon Berard · 2 drugs in this class
- AB Science · 2 drugs in this class
- Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 2 drugs in this class
- Betta Pharmaceuticals Co., Ltd. · 1 drug in this class
- Angion Biomedica Corp · 1 drug in this class
- Beijing InnoCare Pharma Tech Co., Ltd. · 1 drug in this class
- Chang-Ming Huang, Prof. · 1 drug in this class
- Deciphera Pharmaceuticals, LLC · 1 drug in this class
- AstraZeneca · 1 drug in this class
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Cite this brief
Drug Landscape (2026). ApatinibMesylateTablets — Competitive Intelligence Brief. https://druglandscape.com/ci/apatinibmesylatetablets. Accessed 2026-06-10.
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