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ApatinibMesylateTablets — Competitive Intelligence Brief

ApatinibMesylateTablets (ApatinibMesylateTablets) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Tyrosine kinase inhibitor. Area: Oncology.

phase 2 Tyrosine kinase inhibitor VEGFR2 Oncology Small molecule Live · refreshed every 30 min

Target snapshot

ApatinibMesylateTablets (ApatinibMesylateTablets) — Chang-Ming Huang, Prof.. Tyrosine kinase inhibitor

Comparator set (6 drugs)

Auto-detected by same drug class / molecular target / therapeutic area, ranked by phase + recency. Override with ?vs=slug1,slug2,….

DrugGenericSponsorPhaseClassTargetApproval / PDUFA
ApatinibMesylateTablets TARGET ApatinibMesylateTablets Chang-Ming Huang, Prof. phase 2 Tyrosine kinase inhibitor VEGFR2
REGORAFENIB REGORAFENIB marketed RET, VEGFR1, VEGFR2, VEGFR3, KIT, PDGFR-alpha, PDGFR-beta, FGFR1, FGFR2, TIE2, DDR2, TrkA, Eph2A, RAF-1, BRAF, BRAF V600E, SAPK2, PTK5, Abl, CSF1R 2012-01-01
Sutent Sunitinib Malate Pfizer marketed Small molecule kinase inhibitor Receptor tyrosine kinases (RTKs): PDGFRα, PDGFRβ, VEGFR1, VEGFR2, VEGFR3, KIT, FLT3, CSF-1R, RET 2006-01-01
Apatinib+Capecitabine Apatinib+Capecitabine Huazhong University of Science and Technology phase 3 Tyrosine kinase inhibitor + Fluoropyrimidine antimetabolite VEGFR2 (apatinib); Thymidylate synthase (capecitabine)
Ramucirumab+ paclitaxel Ramucirumab+ paclitaxel AstraZeneca phase 3 Angiogenesis inhibitor, Microtubule inhibitor VEGFR2
Rivoceranib (Apatinib) Rivoceranib (Apatinib) Jiangsu HengRui Medicine Co., Ltd. phase 3 tyrosine kinase inhibitor VEGFR2
Ramucirumab / Paclitaxel/ Docetaxel/ Irinotecan Ramucirumab / Paclitaxel/ Docetaxel/ Irinotecan Jiangsu HengRui Medicine Co., Ltd. phase 3 Monoclonal antibody (ramucirumab) + chemotherapy combination VEGF receptor 2 (VEGFR2); tubulin (taxanes) / topoisomerase I (irinotecan)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Tyrosine kinase inhibitor class)

  1. Jiangsu HengRui Medicine Co., Ltd. · 5 drugs in this class
  2. Centre Leon Berard · 2 drugs in this class
  3. AB Science · 2 drugs in this class
  4. Chia Tai Tianqing Pharmaceutical Group Co., Ltd. · 2 drugs in this class
  5. Betta Pharmaceuticals Co., Ltd. · 1 drug in this class
  6. Angion Biomedica Corp · 1 drug in this class
  7. Beijing InnoCare Pharma Tech Co., Ltd. · 1 drug in this class
  8. Chang-Ming Huang, Prof. · 1 drug in this class
  9. Deciphera Pharmaceuticals, LLC · 1 drug in this class
  10. AstraZeneca · 1 drug in this class

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Cite this brief

Drug Landscape (2026). ApatinibMesylateTablets — Competitive Intelligence Brief. https://druglandscape.com/ci/apatinibmesylatetablets. Accessed 2026-06-10.

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing