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Apatinib+Capecitabine — Competitive Intelligence Brief
phase 3
Tyrosine kinase inhibitor + Fluoropyrimidine antimetabolite
VEGFR2 (apatinib); Thymidylate synthase (capecitabine)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Apatinib+Capecitabine (Apatinib+Capecitabine) — Huazhong University of Science and Technology. Apatinib inhibits vascular endothelial growth factor receptor 2 (VEGFR2) to block tumor angiogenesis, while capecitabine is a fluoropyrimidine that inhibits thymidylate synthase to disrupt DNA synthesis in cancer cells.
Comparator set
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Apatinib+Capecitabine TARGET | Apatinib+Capecitabine | Huazhong University of Science and Technology | phase 3 | Tyrosine kinase inhibitor + Fluoropyrimidine antimetabolite | VEGFR2 (apatinib); Thymidylate synthase (capecitabine) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Tyrosine kinase inhibitor + Fluoropyrimidine antimetabolite class)
- Huazhong University of Science and Technology · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Apatinib+Capecitabine — Competitive Intelligence Brief. https://druglandscape.com/ci/apatinib-capecitabine. Accessed 2026-05-16.
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