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Angiotensin II Receptor Blockers — Competitive Intelligence Brief
phase 3
Angiotensin II Receptor Blocker (ARB)
AT1 receptor (Angiotensin II Type 1 Receptor)
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Angiotensin II Receptor Blockers (Angiotensin II Receptor Blockers) — Ottawa Heart Institute Research Corporation. Angiotensin II Receptor Blockers (ARBs) block the angiotensin II type 1 receptor, preventing vasoconstriction and aldosterone release to lower blood pressure.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Angiotensin II Receptor Blockers TARGET | Angiotensin II Receptor Blockers | Ottawa Heart Institute Research Corporation | phase 3 | Angiotensin II Receptor Blocker (ARB) | AT1 receptor (Angiotensin II Type 1 Receptor) | |
| Allisartan Isoproxil | Allisartan Isoproxil | Guangdong Provincial People's Hospital | marketed | Angiotensin II receptor blocker (ARB) | AT1 receptor (Angiotensin II type 1 receptor) | |
| Placebo to Telmisartan | Placebo to Telmisartan | Novartis | marketed | Angiotensin II receptor blocker (ARB) | AT1 receptor (Angiotensin II type 1 receptor) | |
| Valsartan+/- Hydrochlorothiazide | Valsartan+/- Hydrochlorothiazide | Novartis | marketed | Angiotensin II receptor blocker (ARB); combination with thiazide diuretic when applicable | AT1 receptor (angiotensin II type 1 receptor); sodium-chloride cotransporter (thiazide component) | |
| losartan/amlodpine | losartan/amlodpine | University of Pavia | marketed | Angiotensin II receptor blocker (ARB) / Calcium channel blocker (CCB) | Angiotensin II receptors (AT1) and L-type calcium channels | |
| Diovan (Valsartan) | Diovan (Valsartan) | Bayer | marketed | Angiotensin II receptor blocker (ARB) | AT1 receptor (Angiotensin II type 1 receptor) | |
| Cozzar tablet | Cozzar tablet | Chong Kun Dang Pharmaceutical | marketed | Angiotensin II receptor blocker (ARB) | AT1 receptor (angiotensin II type 1 receptor) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Angiotensin II Receptor Blocker (ARB) class)
- Ottawa Heart Institute Research Corporation · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Angiotensin II Receptor Blockers — Competitive Intelligence Brief. https://druglandscape.com/ci/angiotensin-ii-receptor-blockers. Accessed 2026-05-17.
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