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Aliskiren 3.125 mini-tablets — Competitive Intelligence Brief
phase 1
Renin inhibitor
Renin
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Aliskiren 3.125 mini-tablets (Aliskiren 3.125 mini-tablets) — Novartis. Aliskiren is a direct renin inhibitor that blocks the conversion of angiotensinogen to angiotensin I, reducing blood pressure.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Aliskiren 3.125 mini-tablets TARGET | Aliskiren 3.125 mini-tablets | Novartis | phase 1 | Renin inhibitor | Renin | |
| Tekturna | ALISKIREN | Lxo Ireland | marketed | Renin Inhibitor | Renin | 2007-01-01 |
| Capozide 25/15 | CAPTOPRIL | Aarxion Anda Hlding | marketed | Thiazide Diuretic [EPC] | Renin | 1981-01-01 |
| Early sequential nephron blockade | Early sequential nephron blockade | University of Parma | marketed | RAAS inhibitor combination strategy | Renin-angiotensin-aldosterone system (multiple targets) | |
| ALIS | ALIS | Lxo Ireland | marketed | Multidrug resistance protein 1, Cytochrome P450 3A4, Renin | ||
| Aliskiren Hydrochlorothiazide | Aliskiren Hydrochlorothiazide | Novartis | marketed | Direct renin inhibitor / thiazide diuretic combination | Renin; sodium-chloride cotransporter (NCCT) | |
| Keverprazan 14 days | Keverprazan 14 days | Second Affiliated Hospital, School of Medicine, Zhejiang University | marketed | direct renin inhibitor | renin |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Renin inhibitor class)
- Novartis · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Aliskiren 3.125 mini-tablets — Competitive Intelligence Brief. https://druglandscape.com/ci/aliskiren-3-125-mini-tablets. Accessed 2026-05-16.
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