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Acepromethazine — Competitive Intelligence Brief
phase 2
Histamine H1 receptor
Neuroscience
Small molecule
Live · refreshed every 30 min
Target snapshot
Acepromethazine (ACEPROMETAZINE). Acepromethazine works by blocking histamine receptors in the brain to promote sleep.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Acepromethazine TARGET | ACEPROMETAZINE | phase 2 | Histamine H1 receptor | |||
| Lastacaft | ALCAFTADINE | AbbVie | marketed | Histamine-1 Receptor Antagonist [EPC] | Histamine H1 receptor | 2010-01-01 |
| Xyzal | LEVOCETIRIZINE | Sanofi | marketed | Histamine-1 Receptor Antagonist | Histamine H1 receptor | 2007-01-01 |
| Elestat | EPINASTINE | AbbVie | marketed | Adrenergic Receptor Agonist | Histamine H1 receptor | 2003-01-01 |
| Rupax | RUPATADINE | Teikoku Seiyaku | marketed | rupatadine | Histamine H1 receptor | 2001-01-01 |
| Zaditor | KETOTIFEN | marketed | Histamine-1 Receptor Inhibitor | Histamine H1 receptor | 1999-01-01 | |
| Mizollen | MIZOLASTINE | Sanofi | marketed | mizolastine | Histamine H1 receptor | 1998-01-01 |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape
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Cite this brief
Drug Landscape (2026). Acepromethazine — Competitive Intelligence Brief. https://druglandscape.com/ci/aceprometazine. Accessed 2026-06-10.
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