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Abiraterone Acetate (AA) — Competitive Intelligence Brief
phase 3
CYP17A1 inhibitor
CYP17A1 (17α-hydroxylase/17,20-lyase)
Oncology
Small molecule
Live · refreshed every 30 min
Target snapshot
Abiraterone Acetate (AA) (Abiraterone Acetate (AA)) — Janssen Research & Development, LLC. Abiraterone acetate inhibits CYP17A1, a key enzyme in androgen synthesis, thereby reducing testosterone production in patients with castration-resistant prostate cancer.
Comparator set (5 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Abiraterone Acetate (AA) TARGET | Abiraterone Acetate (AA) | Janssen Research & Development, LLC | phase 3 | CYP17A1 inhibitor | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone acetate and prednisone | Abiraterone acetate and prednisone | Janssen Research & Development, LLC | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Abiraterone + Prednisolone/Prednisone | Abiraterone + Prednisolone/Prednisone | AstraZeneca | phase 3 | CYP17A1 inhibitor (androgen synthesis inhibitor) + glucocorticoid | CYP17A1 (17α-hydroxylase/17,20-lyase) | |
| Enzalutamide, Abiraterone | Enzalutamide, Abiraterone | Veru Inc. | phase 3 | Androgen receptor antagonist + CYP17A1 inhibitor combination | Androgen receptor (AR) and CYP17A1 | |
| Abiraterone with Prednisone or Enzalutamide | Abiraterone with Prednisone or Enzalutamide | Curium US LLC | phase 3 | CYP17A1 inhibitor (abiraterone) + androgen receptor antagonist (enzalutamide) + glucocorticoid (prednisone) | CYP17A1 (abiraterone); androgen receptor (enzalutamide); glucocorticoid receptor (prednisone) | |
| Fuzuloparib , Abiraterone acetate and Prednisone | Fuzuloparib , Abiraterone acetate and Prednisone | Jiangsu HengRui Medicine Co., Ltd. | phase 3 | PARP inhibitor (fuzuloparib) combined with CYP17A1 inhibitor (abiraterone acetate) and glucocorticoid (prednisone) | PARP1/PARP2 (fuzuloparib); CYP17A1 (abiraterone acetate); glucocorticoid receptor (prednisone) |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (CYP17A1 inhibitor class)
- Assistance Publique - Hôpitaux de Paris · 1 drug in this class
- Janssen Research & Development, LLC · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Abiraterone Acetate (AA) — Competitive Intelligence Brief. https://druglandscape.com/ci/abiraterone-acetate-aa. Accessed 2026-06-10.
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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing