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NCT06186427: 68Ga-GPFAPI

A Novel 68Ga Labeled FAP Ligand PET/CT in Patients With Various Malignant Tumors

Status unknown NA Last updated 22 January 2024
What this trial tests

NA trial testing 68Ga-DOTA-GPFAPI-04 PET/CT in Cancer in 30 participants. Status unknown.

Timeline
13 January 2024
Primary endpoint
31 August 2025
31 December 2025

Quick facts

Lead sponsorGuangdong Provincial People's Hospital
PhaseNA
StatusStatus unknown
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposediagnostic
Enrollment30
Start date13 January 2024
Primary completion31 August 2025
Estimated completion31 December 2025
Sites1 location across China

Drugs / interventions tested

Conditions studied

Sponsor

Guangdong Provincial People's Hospital

Who can join

Adults 18 to 80, any sex, with Cancer or Malignant Neoplasm. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

The investigators designed and synthesized a novel fibroblast activation protein (FAP) ligand (DOTA-GPFAPI-04) by assembling three functional moieties: a quinoline-based FAP inhibitor for specifically targeting FAP, a FAP substrate Gly-Pro as a linker for increasing the FAP protein interaction, and a 2,2',2",2‴-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetraacetic acid (DOTA) chelator for radiolabeling with different radionuclides. Molecular docking studies investigated the FAP targeting ability of DOTA-GPFAPI-04. DOTA-GPFAPI-04 was then radiolabeled with 68Ga to give 68Ga-DOTA-GPFAPI-04 for positron emission tomography (PET) imaging. The investigators found that the 68Ga-DOTA-GPFAPI-04 has high stability, targeted specificity, and longer retention time. The tumor-to-muscle (T/M) ratio for 68Ga-DOTA-GPFAPI-04 reached 9.15.

Publications & conference data

No peer-reviewed publications indexed yet for this trial.

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Other recruiting trials for Cancer

Currently open trials in the same condition.

Other Guangdong Provincial People's Hospital trials

Trials by the same sponsor.

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Data sources for this page

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