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NCT05817708

A Study of Silmitasertib (CX-4945) in Healthy Subject

Completed Phase 1 Results posted Last updated 27 January 2025
What this trial tests

Phase 1 trial testing CX-4945 in COVID-19 in 30 participants. Completed in 20 June 2023.

Timeline
28 November 2022
Primary endpoint
23 March 2023
20 June 2023

Quick facts

Lead sponsorSenhwa Biosciences, Inc.
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designparallel
Maskingnone
Primary purposetreatment
Enrollment30
Start date28 November 2022
Primary completion23 March 2023
Estimated completion20 June 2023
Sites1 location across Taiwan

Drugs / interventions tested

Conditions studied

Sponsor

Senhwa Biosciences, Inc. — full company profile →

Who can join

Adults 20 to 55, any sex, with COVID-19. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Number of Participants With Treatment-emergent Adverse Events (TEAT) Primary · Day 1 to Day 5

Evaluate the number adverse events occurring from Day 1 to Day 5 as characterized by type, frequency, severity \[as graded by the National Cancer Institute Common Terminology Criteria for Adverse Events \[CTCAE\] version 5.0\], timing, seriousness, and relationship to study therapy after administration of 200mg QD, 200mg BID and 400mg BID for continuously 5 days to healthy subjects.

GroupValue95% CI
CX-4945 200mg QD1
CX-4945 200mg BID3
CX-4945 400mg BID7
Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes ALP in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD-2.1± 5.78
CX-4945 200mg BID-0.3± 6.62
CX-4945 400mg BID3.4± 2.84
Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes AST in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD-3.9± 5.11
CX-4945 200mg BID-2.4± 3.72
CX-4945 400mg BID0.1± 3.35
To Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes ALT in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD-4.0± 6.15
CX-4945 200mg BID-1.4± 5.19
CX-4945 400mg BID0.9± 4.77
To Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes LDH in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD-17.0± 17.17
CX-4945 200mg BID-26.2± 10.75
CX-4945 400mg BID-28.2± 14.33
To Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes CPK in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD-24.3± 19.35
CX-4945 200mg BID-54.0± 63.71
CX-4945 400mg BID-65.1± 71.37
To Evaluate Changes in Blood Chemistry. Secondary · Day 1 to Day 6

Changes CRP in blood chemistry assessment from Day 1(Baseline) to Day 6 morning.

GroupValue95% CI
CX-4945 200mg QD0.003± 0.1341
CX-4945 200mg BID-0.071± 0.2497
CX-4945 400mg BID0.002± 0.0447
Number of Participants Evaluated as Having Abnormalities (CS or NCS) in Their ECG Secondary · Screening, Day 1, Day 3, Day 5, and Day 6

ECG assessments were done during Screening, Day 1, Day 3, Day 5, and Day 6. A 12-lead ECG was performed at baseline (Day1), Day 3, Day 5, and Day 6 and categorized as normal, abnormal and not clinically significant (abnormal NCS) or abnormal and clinically significant (abnormal CS).

Screening
GroupValue95% CI
CX-4945 200mg QD7
CX-4945 200mg BID6
CX-4945 400mg BID6
Day 1 (Baseline)
GroupValue95% CI
CX-4945 200mg QD3
CX-4945 200mg BID4
CX-4945 400mg BID8
Day 3
GroupValue95% CI
CX-4945 200mg QD7
CX-4945 200mg BID9
CX-4945 400mg BID6
Day 5
GroupValue95% CI
CX-4945 200mg QD5
CX-4945 200mg BID6
CX-4945 400mg BID7
Day 6
GroupValue95% CI
CX-4945 200mg QD6
CX-4945 200mg BID6
CX-4945 400mg BID6

Adverse events — posted to ClinicalTrials.gov

Time frame: from Day 1 to Day 6. Reporting threshold: 0%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

CX-4945 200mg BID
Serious: 0/10 (0%)
Deaths: 0/10
CX-4945 200mg QD
Serious: 0/10 (0%)
Deaths: 0/10
CX-4945 400mg BID
Serious: 0/10 (0%)
Deaths: 0/10
Other adverse events (8 terms — click to expand)

ReactionSystemCX-4945 200mg BIDCX-4945 200mg QDCX-4945 400mg BID
DirrhoeaGastrointestinal disorders
C-reactive protein abnormalInvestigations
NauseaGastrointestinal disorders
Alanine aminotransferase increasedInvestigations
Aspartate aminotransferase increasedInvestigations
Blood creatine phosphokinase increasedInvestigations
Gamma-glutamyltransferase increasedInvestigations
HypertriglyceridaemiaMetabolism and nutrition disorders

Data from ClinicalTrials.gov NCT05817708 adverse events section.

Sponsor's own description

This is a Phase I single center, open-label, parallel design in 30 subjects to evaluate safety and tolerability of CX-4945 200mg QD, 200 mg BID and 400mg BID doses (10 subjects in each regimen) for continuously 5 days in healthy subjects for dose selection.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. VTA dopamine neurons are hyperexcitable in 3xTg-AD mice due to casein kinase 2-dependent SK channel dysfunction.
    Blankenship HE, Carter KA, Pham KD, Cassidy NT, et al · · 2024 · cited 15× · PMID 39516200 · DOI 10.1038/s41467-024-53891-1

Verify or expand the search:

Other trials of CX-4945

Trials testing the same drug.

Other recruiting trials for COVID-19

Currently open trials in the same condition.

Other Senhwa Biosciences, Inc. trials

Trials by the same sponsor.

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT05817708.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing