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NCT05732454

A Study to Learn About the Study Medicine Etrasimod in Adults With Moderate to Severe Atopic Dermatitis (AD) Who Have Already Tried Treatments Taken by Mouth or by Injection

Terminated Phase 2, PHASE3 Results posted Last updated 8 May 2025
What this trial tests

Phase 2, PHASE3 trial testing etrasimod in Atopic Dermatitis in 58 participants. Terminated before completion.

Timeline
18 January 2023
Primary endpoint
29 April 2024
29 April 2024

Quick facts

Lead sponsorPfizer
PhasePhase 2, PHASE3
StatusTerminated
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingquadruple
Primary purposetreatment
Enrollment58
Start date18 January 2023
Primary completion29 April 2024
Estimated completion29 April 2024
Sites74 locations across Canada, United States, Poland, Czechia

Drugs / interventions tested

Conditions studied

Sponsor

Pfizer — full company profile →

Who can join

Adults 18 to 80, any sex, with Atopic Dermatitis or Atopic Dermatitis, Unspecified. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Part 1, DB Period: Percentage of Participants Achieving Investigator's Global Assessment (IGA) Response at Week 16 Primary · DB Period: Week 16

IGA measured AD severity, based on a 5-point scale (0-4); 0= AD is clear, 1= AD is almost clear, 2= mild AD, 3= moderate AD and 4= severe AD. IGA response was defined as participants achieving IGA 0 (clear) or 1 (almost clear) and a reduction of \>=2 points from baseline.

GroupValue95% CI
DB Period: Etrasimod 2 mg3.3
DB Period: Placebo7.1
Part 1, DB Period: Percentage of Participants Who Achieved >=75% Reduction From Baseline in Eczema Area and Severity Index (EASI) Score (EASI-75) at Week 16 Secondary · DB Period: Week 16

EASI-75 response was defined as a 75% reduction or greater in EASI score from Baseline to Week 16. EASI quantified severity of AD based on severity of lesion clinical signs and percentage (%) of body surface area (BSA) affected. Severity of clinical signs of AD lesions (erythema \[E\], induration/papulation \[I\], excoriation \[Ex\] and lichenification \[L\]) were scored separately for each of 4 body regions (head and neck, upper limbs, trunk \[including axillae and groin)\] and lower limbs \[including buttocks\]) on a 4-point scale: 0= absent; 1= mild; 2= moderate; 3= severe. EASI area score

GroupValue95% CI
DB Period: Etrasimod 2 mg23.3
DB Period: Placebo14.3
Part 1, DB Period: Percent Change From Baseline in EASI Score at Week 16 Secondary · DB Period: Baseline, Week 16

EASI quantified severity of AD based on severity of lesion clinical signs and percentage (%) of body surface area (BSA) affected. Severity of clinical signs of AD lesions (erythema \[E\], induration/papulation \[I\], excoriation \[Ex\] and lichenification \[L\]) were scored separately for each of 4 body regions (head and neck, upper limbs, trunk \[including axillae and groin)\] and lower limbs \[including buttocks\]) on a 4-point scale: 0= absent; 1= mild; 2= moderate; 3= severe. EASI area score was based on % BSA with AD in body region: 0 (0%), 1 (\>0 to \<10%), 2 (10 to \<30%), 3 (30 to \<50

GroupValue95% CI
DB Period: Etrasimod 2 mg-53.87± 9.007
DB Period: Placebo-24.65± 9.533
Part 1, DB Period: Number of Participants With Treatment Emergent Adverse Events (TEAEs) (All Causality) Primary · DB Period: From first dose of study drug up to 16 Weeks of treatment

An adverse event (AE) was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state.

GroupValue95% CI
DB Period: Etrasimod 2 mg16
DB Period: Placebo8
Part 1, DB Period: Number of Participants With TEAEs (All Causality) Leading to Study Treatment Discontinuation Primary · DB Period: From first dose of study drug up to 16 Weeks of treatment

An AE was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state.

GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
Part 1, DB Period: Number of Participants With Treatment Emergent Serious Adverse Events (SAEs) (All Causality) Primary · DB Period: From first dose of study drug up to 16 Weeks of treatment

An AE was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state. SAE was an AE resulting in any of the following outcomes or deemed significant for any other reason: death; life-threatening experience (immediate risk of death); new or prolonged inpatient hospitalization; persistent or significant disability/incapacity;

GroupValue95% CI
DB Period: Etrasimod 2 mg0
DB Period: Placebo0
Part 1, DB Period: Number of Participants With Treatment Emergent AEs of Special Interest (AESIs) (All Causality) Primary · DB Period: From first dose of study drug up to 16 Weeks of treatment

An AE was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state. AESIs included here were cardiovascular events (i.e., bradycardia, Atrioventricular (AV) conduction delay, and hypertension); macular edema, pulmonary events (airflow obstruction or decreased gas exchange); infections (severe infections, opportunistic inf

GroupValue95% CI
DB Period: Etrasimod 2 mg2
DB Period: Placebo1
Part 1, DB Period: Number of Participants With Laboratory Test Abnormalities Primary · DB Period: From first dose of study drug up to 16 Weeks of treatment

Laboratory assessments included hematology, clinical chemistry, urinalysis, other parameters and reflex tests. Number of participants with abnormalities in any of laboratory parameters is reported.

GroupValue95% CI
DB Period: Etrasimod 2 mg22
DB Period: Placebo13
Part 1, DB Period: Number of Participants With Markedly Abnormal 12-Lead Electrocardiogram Measurements and AV Blocks Primary · DB Period: Pre-dose and 4 hours (hrs) post-dose on Day 1/Week 0; Pre-dose and 4 hrs post-dose on Day 113/Week 16

Standard 12-lead ECGs utilizing limb leads were used to measure PR interval, QT interval, QTc corrected using Fridericia's formula (QTcF), and QRS complex. Number of participants with non-zero ECG abnormalities and AV blocks are reported in this outcome measure.

Pre-dose/Day 1: AV conduction: First-degree AV Block
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
4 hrs post-dose/Day 1: QTCF (msec), single beat:>= 450 (male) or >= 470 (female)
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
4 hrs post-dose/Day 1: Change From Baseline (CFB) in QT: >30 msec increase
GroupValue95% CI
DB Period: Etrasimod 2 mg9
DB Period: Placebo0
4 hrs post-dose/Day 1: AV conduction: First degree AV Block
GroupValue95% CI
DB Period: Etrasimod 2 mg3
DB Period: Placebo0
Pre-dose/Week 16: CFB in QT: >30 msec increase
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
Pre-dose/Week 16: CFB in QT: >60 msec increase
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
Pre-dose/Week 16: CFB in QTcF: >30 msec increase
GroupValue95% CI
DB Period: Etrasimod 2 mg2
DB Period: Placebo0
4 hrs post-dose/Week 16: CFB in QTcF: >30 msec increase
GroupValue95% CI
DB Period: Etrasimod 2 mg2
DB Period: Placebo0
Part 1, DB Period: Number of Participants With Markedly Abnormal Vital Sign Primary · DB Period: Pre-dose and 1, 2, 3, 4 hours (hrs) post-dose on Day 1/Week 0; Day 29/Week 4; Day 57/Week 8; Day 85/Week 12; Pre-dose and 1, 2, 3, 4, 5 and 6 hrs post-dose on Day 113/Week 16

Vital signs evaluation included systolic blood pressure (SBP), diastolic blood pressure (DBP), pulse rate. Number of participants with non-zero vital signs abnormalities are reported in this outcome measure.

Pre-dose/Day 1: DBP >90 mmHg
GroupValue95% CI
DB Period: Etrasimod 2 mg0
DB Period: Placebo1
Pre-dose/Day 1: Pulse rate: <60 bpm
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo3
Pre-dose/Day 1: Pulse rate >100 bpm
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
1 hr post-dose/Day 1: SBP: Change >=30 mmHg decrease
GroupValue95% CI
DB Period: Etrasimod 2 mg0
DB Period: Placebo1
1 hr post-dose/Day 1: DBP >90 mmHg
GroupValue95% CI
DB Period: Etrasimod 2 mg2
DB Period: Placebo2
1 hr post-dose/Day 1: Pulse rate: <50 bpm
GroupValue95% CI
DB Period: Etrasimod 2 mg1
DB Period: Placebo0
1 hr post-dose/Day 1: Pulse rate: <60 bpm
GroupValue95% CI
DB Period: Etrasimod 2 mg7
DB Period: Placebo3
2 hrs post-dose/Day 1: SBP: >150 mmHg
GroupValue95% CI
DB Period: Etrasimod 2 mg0
DB Period: Placebo2
Part 1, OLE Period: Number of Participants With TEAEs (All Causality) Primary · OLE Period: First dose of study drug in OLE period up to 4 weeks after last dose in OLE period (up to maximum of 56 Weeks)

An AE was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state.

GroupValue95% CI
OLE Period: Etrasimod 2 mg (Etrasimod 2 mg in DB Period)9
OLE Period: Etrasimod 2 mg (Placebo in DB Period)5
Part 1, OLE Period: Number of Participants With Treatment Emergent AEs (All Causality) Leading to Study Treatment Discontinuation Primary · OLE Period: First dose of study drug in OLE period up to 4 weeks after last dose in OLE period (up to maximum of 56 Weeks)

An AE was any untoward medical occurrence in a participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention. Treatment-emergent are events between first dose of study drug and up to last dose that were absent before treatment or that worsened relative to pretreatment state.

GroupValue95% CI
OLE Period: Etrasimod 2 mg (Etrasimod 2 mg in DB Period)0
OLE Period: Etrasimod 2 mg (Placebo in DB Period)1

Adverse events — posted to ClinicalTrials.gov

Time frame: Part 1, DB Period: Day 1 to Week 16; Part 1, OLE Period: Week 20 to Week 68; Part 1, DB +OLE Period: Day 1 to Week 68. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

DB Period: Etrasimod 2 mg
Serious: 0/30 (0%)
Deaths: 0/30
DB Period: Placebo
Serious: 0/28 (0%)
Deaths: 0/28
OLE Period: Etrasimod 2 mg (Etrasimod 2 mg in DB Period)
Serious: 1/30 (3%)
Deaths: 0/30
OLE Period: Etrasimod 2 mg (Placebo in DB Period)
Serious: 0/28 (0%)
Deaths: 0/28
DB Etrasimod 2 mg Then OLE Etrasimod 2 mg
Serious: 1/30 (3%)
Deaths: 0/30
DB Placebo Then OLE Etrasimod 2 mg
Serious: 0/28 (0%)
Deaths: 0/28

Serious adverse events (1 terms)

ReactionSystemDB Period: Etrasimod 2 mgDB Period: PlaceboOLE Period: Etrasimod 2 mg…OLE Period: Etrasimod 2 mg…DB Etrasimod 2 mg Then OLE…DB Placebo Then OLE Etrasi…
Pneumothorax spontaneousRespiratory, thoracic and mediastinal disorders
Other adverse events (5 terms — click to expand)

ReactionSystemDB Period: Etrasimod 2 mgDB Period: PlaceboOLE Period: Etrasimod 2 mg…OLE Period: Etrasimod 2 mg…DB Etrasimod 2 mg Then OLE…DB Placebo Then OLE Etrasi…
HypertensionVascular disorders
COVID-19Infections and infestations
NasopharyngitisInfections and infestations
Dermatitis atopicSkin and subcutaneous tissue disorders
Respiratory tract infectionInfections and infestations

Most-reported serious reactions: Pneumothorax spontaneous.

Data from ClinicalTrials.gov NCT05732454 adverse events section.

Sponsor's own description

The purpose of this study is to learn about the safety and effects of the study medicine called etrasimod for the possible treatment of atopic dermatitis (AD), also called eczema, in adults who have already tried AD treatments taken by mouth or by injection that work all over the body. These adults can have moderate to severe AD. This study is seeking participants who: * have AD for at least 1 year * have moderate-to-severe AD * have tried treatments that work all over the body and saw no effects * are willing to apply a moisturizer at least once daily during the study This is a 2-part study that is only selecting about 60 participants for Part 1 as of now. In Part 1, half of the participants will receive etrasimod, a pill to be taken by mouth once daily. The other half will receive a placebo, a pill that looks like etrasimod but has no medicine also taken by mouth once daily. No one will know what treatment the participant is taking. The Sponsor will compare participant experiences of those taking etrasimod to those taking placebo for 16 weeks. This will help determine if the study medicine is safe and effective. After the first 16 weeks, some participants may continue the study knowing they are taking etrasimod for an additional 52 weeks. Those participating for just the first 16-weeks, will need to visit the study clinic at least 6 times during the study (about every 4 weeks), and will have to come for 2 safety follow up visits at 2nd and 4th week after the last dose of study medicine. People who want to and can continue for an additional 52 weeks will need to visit the study clinic for at least 6 more visits making 12 total visits over 68 weeks followed by 2 safety follow up visits at the 2nd and 4th week after the last dose of study medicine. In Part 2 of the study, around 340 more participants will be participating. Everyone will receive etrasimod pills once daily for 52 weeks. Participants will need to go to the study clinic at least 9 times after which they will have to go for 2 more safety follow up visits at the 2nd and 4th weeks after the last dose of study medicine. At every study visit in Part 1 and Part 2, the focus will be on signs and symptoms of AD (like lesions, itch, and pain) as well as general health and overall side effects. Blood samples and vital signs will be taken at every visit. Due to the way the study medicine works, the in-study clinic visit will last at least 4 hours on Day 1 (Part 1 and Part 2) and Week 16 (Part 1).

Publications & conference data

2 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Atopic dermatitis: a comprehensive updated review of this intriguing disease with futuristic insights.
    Abdel-Mageed HM. · · 2025 · cited 16× · PMID 39918744 · DOI 10.1007/s10787-025-01642-z
  2. T cell trafficking in human chronic inflammatory diseases.
    Giovenzana A, Codazzi V, Pandolfo M, Petrelli A. · · 2024 · cited 5× · PMID 39171290 · DOI 10.1016/j.isci.2024.110528

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT05732454.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing