Last reviewed · How we verify

NCT05483998

A Study to Evaluate Single and Multiple Doses of TLC-2716 in Healthy Participants

Completed Phase 1 Last updated 20 May 2024
What this trial tests

Phase 1 trial testing TLC-2716 in Healthy Subjects in 100 participants. Completed in 18 June 2023.

Timeline
9 September 2022
Primary endpoint
13 April 2023
18 June 2023

Quick facts

Lead sponsorOrsoBio, Inc
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designsequential
Maskingdouble
Primary purposetreatment
Enrollment100
Start date9 September 2022
Primary completion13 April 2023
Estimated completion18 June 2023
Sites1 location across New Zealand

Drugs / interventions tested

Conditions studied

Sponsor

OrsoBio, Inc — full company profile →

Who can join

Adults 18 to 55, any sex, with Healthy Subjects. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

This phase 1 study is designed to evaluate the safety, tolerability, pharmacokinetics, and pharmacodynamics of TLC-2716 after single- and multiple-ascending doses in healthy subjects.

Publications & conference data

3 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Development of LXR inverse agonists to treat MAFLD, NASH, and other metabolic diseases.
    Griffett K, Burris TP. · · 2023 · cited 26× · PMID 36817797 · DOI 10.3389/fmed.2023.1102469
  2. An oral, liver-restricted LXR inverse agonist for dyslipidemia: preclinical development and phase 1 trial.
    Li X, Benegiamo G, Vijayakumar A, Sroda N, et al · · 2026 · cited 1× · PMID 41545590 · DOI 10.1038/s41591-025-04169-6
  3. Nuclear receptors as therapeutic targets in metabolic and cardiovascular disorders.
    Li F, Chen Q, Dai Y, Lu L. · · 2025 · PMID 41438090 · DOI 10.1016/j.isci.2025.114042

Verify or expand the search:

Other recruiting trials for Healthy Subjects

Currently open trials in the same condition.

Other OrsoBio, Inc trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT05483998.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing