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NCT05266586: ROSE2

Study to Evaluate the Effect of Obicetrapib in Combination With Ezetimibe as an Adjunct to HIS Therapy

Completed Phase 2 Results posted Last updated 3 July 2024
What this trial tests

Phase 2 trial testing Obicetrapib in Dyslipidemias in 119 participants. Completed in 8 September 2022.

Timeline
9 March 2022
Primary endpoint
12 August 2022
8 September 2022

Quick facts

Lead sponsorNewAmsterdam Pharma
PhasePhase 2
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingquadruple
Primary purposetreatment
Enrollment119
Start date9 March 2022
Primary completion12 August 2022
Estimated completion8 September 2022
Sites16 locations across United States

Drugs / interventions tested

Conditions studied

Sponsor

NewAmsterdam Pharma — full company profile →

Who can join

Adults 18 to 75, any sex, with Dyslipidemias or High Cholesterol. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [Friedewald] Primary · 12-weeks

Mean percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-0.83± 24.514
Combination Therapy-59.07± 14.814
Median Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [Friedewald] Primary · 12-Weeks

Median percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-6.35-36.4 – 96.7
Combination Therapy-63.40-83.7 – -29.7
LS Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [Friedewald] Primary · 12-Weeks

LS Mean percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-0.85± 3.472
Combination Therapy-59.23± 3.786
Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [PUC] Primary · 12-Weeks

Mean percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-1.49± 23.762
Combination Therapy-59.51± 15.192
Median Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [PUC] Primary · 12-Weeks

Median percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-3.95-34.3 – 91.8
Combination Therapy-62.80-82.3 – -31.0
LS Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Combination Treatment Group Compared With the Placebo Group [PUC] Primary · 12-Weeks

LS Mean percent change from Day 1 to Day 84 in Low-Density Lipoprotein Cholesterol (LDL-C) for the obicetrapib 10 mg + ezetimibe 10 mg combination treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-1.54± 3.533
Combination Therapy-59.69± 3.811
Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [Friedewald] Secondary · 12-weeks

Mean percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-0.83± 24.514
Monotherapy-39.35± 22.602
Median Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [Friedewald] Secondary · 12-Weeks

Median percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-6.35-36.4 – 96.7
Monotherapy-43.50-78.4 – 22.6
LS Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [Friedewald] Secondary · 12-Weeks

LS Mean percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C was calculated using the Friedewald equation unless TG ≥400 mg/dL or LDL-C ≤50 mg/dL; if TG ≥400 mg/dL or LDL-C ≤50 mg/dL, then LDL-C level was measured directly by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-0.85± 3.472
Monotherapy-39.20± 4.133
Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [PUC] Secondary · 12-Weeks

Mean percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-1.49± 23.762
Monotherapy-39.04± 23.456
Median Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [PUC] Secondary · 12-Weeks

Median percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-3.95-34.3 – 91.8
Monotherapy-43.55-78.4 – 20.4
LS Mean Percent Change in Low-Density Lipoprotein Cholesterol (LDL-C) for Obicetrapib 10 mg Monotherapy Compared With Placebo [PUC] Secondary · 12-Weeks

LS Mean percent change in Low-Density Lipoprotein Cholesterol (LDL-C) from day 1 to day 84 for obicetrapib 10 mg monotherapy treatment group compared with the placebo group. LDL-C level was measured by preparative ultracentrifugation (PUC).

GroupValue95% CI
Placebo-1.54± 3.533
Monotherapy-38.75± 4.166

Adverse events — posted to ClinicalTrials.gov

Time frame: From first dose of study drug through Week 16. Reporting threshold: 0%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Placebo
Serious: 1/40 (3%)
Deaths: 0/40
Monotherapy
Serious: 1/39 (3%)
Deaths: 0/39
Combination Therapy
Serious: 0/40 (0%)
Deaths: 0/40

Serious adverse events (2 terms)

ReactionSystemPlaceboMonotherapyCombination Therapy
Acute myocardial infarctionCardiac disorders
Cerebrovascular accidentNervous system disorders
Other adverse events (42 terms — click to expand)

ReactionSystemPlaceboMonotherapyCombination Therapy
Urinary tract infectionInfections and infestations
NauseaGastrointestinal disorders
HeadacheNervous system disorders
MyalgiaMusculoskeletal and connective tissue disorders
COVID-19Infections and infestations
Acute sinusitisInfections and infestations
BronchitisInfections and infestations
NasopharyngitisInfections and infestations
PharyngitisInfections and infestations
Tooth infectionInfections and infestations
Abdominal painGastrointestinal disorders
Abdominal pain upperGastrointestinal disorders
DiarrhoeaGastrointestinal disorders
Gastrooesophageal reflux diseaseGastrointestinal disorders
VomitingGastrointestinal disorders
Foot fractureInjury, poisoning and procedural complications
Muscle strainInjury, poisoning and procedural complications
FallInjury, poisoning and procedural complications
Rib fractureInjury, poisoning and procedural complications
Road traffic accidentInjury, poisoning and procedural complications
Skin lacerationInjury, poisoning and procedural complications
Vaccination complicationInjury, poisoning and procedural complications
DizzinessNervous system disorders
Burning sensationNervous system disorders
Cerebrovascular accidentNervous system disorders
Dizziness posturalNervous system disorders
MigraineNervous system disorders
TremorNervous system disorders
Blood creatine phosphokinase increasedInvestigations
Blood lactate dehydrogenase increasedInvestigations
Haemoglobin decreasedInvestigations
Hepatic enzyme increasedInvestigations
Weight increasedInvestigations
ArthralgiaMusculoskeletal and connective tissue disorders
Muscle spasmsMusculoskeletal and connective tissue disorders
Acute myocardial infarctionCardiac disorders
Coronary artery diseaseCardiac disorders
TachycardiaCardiac disorders
AnaemiaBlood and lymphatic system disorders
ThrombocytosisBlood and lymphatic system disorders

Most-reported serious reactions: Acute myocardial infarction, Cerebrovascular accident.

Data from ClinicalTrials.gov NCT05266586 adverse events section.

Sponsor's own description

This study will be a placebo-controlled, double-blind, randomized, phase 2 study to evaluate the efficacy, safety, and tolerability of obicetrapib 10 mg, both in combination with ezetimibe 10 mg and as monotherapy, as an adjunct to high-intensity statin therapy.

Publications & conference data

3 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Roles of peripheral lipoproteins and cholesteryl ester transfer protein in the vascular contributions to cognitive impairment and dementia.
    Poliakova T, Wellington CL. · · 2023 · cited 24× · PMID 37974180 · DOI 10.1186/s13024-023-00671-y
  2. Obicetrapib exhibits favorable physiochemical and pharmacokinetic properties compared to previous cholesteryl ester transfer protein inhibitors: An integrated summary of results from non-human primate studies and clinical trials.
    Nicholls SJ, Nelson AJ, Kastelein JJP, Ditmarsch M, et al · · 2024 · cited 7× · PMID 39425271 · DOI 10.1002/prp2.70010
  3. Existing and Potential Therapeutic Strategies for Lowering Lipoprotein(a) Levels: An Update.
    Domański I, Kozieł A, Domański J, Trocha M. · · 2026 · PMID 41899103 · DOI 10.3390/jcm15062179

Verify or expand the search:

Other trials of Obicetrapib

Trials testing the same drug.

Other recruiting trials for Dyslipidemias

Currently open trials in the same condition.

Other NewAmsterdam Pharma trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT05266586.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing