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NCT05176379

Endothelial Derived Hyperpolarization Factor and Regulation of Cerebral and Muscle Blood Flow

Recruiting now Phase 4 Last updated 19 July 2024
What this trial tests

Phase 4 trial testing Fluconazole 150 mg in Healthy in 30 participants. Currently enrolling.

Timeline
19 February 2022
Primary endpoint
1 December 2024
1 May 2025

Quick facts

Lead sponsorUniversity of Oklahoma
PhasePhase 4
StatusRecruiting now
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingsingle
Primary purposebasic science
Enrollment30
Start date19 February 2022
Primary completion1 December 2024
Estimated completion1 May 2025
Sites1 location across United States

Drugs / interventions tested

Conditions studied

Sponsor

University of Oklahoma

Who can join

Adults 18 to 30, any sex, with Healthy. Healthy volunteers can join.

What's being measured

Primary outcomes are the specific endpoints the trial is designed to prove or disprove.

Sponsor's own description

Most cardiometabolic diseases are characterized by increased muscle sympathetic nerve activity (MSNA) during rest and exercise which contributes to poor health outcomes. In healthy humans during muscle contraction, there is a blunting of skeletal muscle vascular responsiveness to increases in MSNA. However, the exact mechanisms involved are unknown although, best evidence suggests that the mechanism is endothelium derived, but nitric oxide (NO) and prostaglandin (PG) independent. Endothelium-derived hyperpolarizing factor (EDHF) is a NO and PG independent vasodilator in both cerebral and skeletal muscle circulations, however, it is unknown if EDHF contributes to vascular responsiveness during elevated MSNA. The application of lower body negative pressure (LBNP) is a safe and non-invasive manipulation that can be used to increase MSNA causing vasoconstriction in humans. Therefore, the purpose of this experiment is to determine if acute inhibition of EDHF alters central and peripheral vascular responses to LBNP at rest and during dynamic exercise. Thereby, providing evidence by which EDHF contributes to vascular control in healthy humans and identify it's potential as a therapeutic target for cardiometabolic diseases that are characterized by elevated MSNA

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. The effects of CYP450 inhibition on cerebrovascular control during rest and mild hypovolemia: An exploratory study in young, healthy adults.
    Matney JE, Buelow AA, Mixon C, Skillett SM, et al · · 2025 · cited 1× · PMID 41420405 · DOI 10.14814/phy2.70712

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Other trials of Fluconazole 150 mg

Trials testing the same drug.

Other recruiting trials for Healthy

Currently open trials in the same condition.

Other University of Oklahoma trials

Trials by the same sponsor.

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT05176379.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing