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NCT04971837

Interaction Between Cannabidiol, Meal Ingestion, and Liver Function

Completed NA Results posted Last updated 15 November 2024
What this trial tests

NA trial testing Cannabidiol (CBD) powder formulation in Metabolism in 26 participants. Completed in 9 December 2021.

Timeline
20 May 2021
Primary endpoint
9 December 2021
9 December 2021

Quick facts

Lead sponsorColorado State University
PhaseNA
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingsingle
Primary purposebasic science
Enrollment26
Start date20 May 2021
Primary completion9 December 2021
Estimated completion9 December 2021
Sites1 location across United States

Drugs / interventions tested

Conditions studied

Sponsor

Colorado State University

Who can join

18 and older, any sex, with Metabolism or Liver Function. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Pharmacokinetic Time to Maximum Concentration- (Tmax) for Different Formulations of CBD Primary · Venous blood will be sampled at standardized intervals: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate Tmax (minutes).

GroupValue95% CI
Formulation 088116.3± 76
Formulation 12635.4± 13.5
Formulation 21351.8± 24.2
Formulation 625129.5± 89.6
Formulation 72538.2± 24.9
Pharmacokinetic Maximum Concentration-(Cmax) for Different Formulations of CBD Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate Cmax (ng/mL).

GroupValue95% CI
Formulation 0880.5± 0.2
Formulation 1263.1± 2.1
Formulation 2132.2± 2.0
Formulation 6250.4± 0.6
Formulation 7251.8± 1.5
Pharmacokinetic Area Under the Curve Representing Total Cannabidiol Exposure Between 0 and 4 h (AUC 0-4) for Different Formulations of CBD Primary · Venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate AUC 0-4 (min x ng/mL).

GroupValue95% CI
Formulation 08862.8± 29.7
Formulation 126272.3± 176
Formulation 213208.6± 151.1
Formulation 62546± 59.4
Formulation 725177.3± 104.8
Pharmacokinetic Area Under the Curve an Estimate of Total Exposure to CBD Over Time (AUC 0-inf) for Different Formulations of CBD Primary · Venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate AUC 0-inf (mins x ng/mL).

GroupValue95% CI
Formulation 126385.2± 226.6
Formulation 213367.6± 217.1
Formulation 725301.6± 221.9
Pharmacokinetic Amount of Time it Takes to Decrease the Circulating Concentration to Half of Its Initial Value (t1/2) for Different Formulations of CBD Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate t1/2 (mins).

GroupValue95% CI
Formulation 088280.7± 141.5
Formulation 126171.0± 129.2
Formulation 213140.5± 96.6
Formulation 625442.7± 451.0
Formulation 725133.1± 26.7
Pharmacokinetic Rate at Which CBD is Removed From the Body (Ke) for Different Formulations of CBD Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate Ke (1/h).

GroupValue95% CI
Formulation 08800.003± .001
Formulation 126.006± .003
Formulation 213.006± .002
Formulation 6250.003± .002
Formulation 7250.005± .001
CBD Pharmacokinetic Volume of Distribution- (Vd) for Different Formulations of CBD Primary · Venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

The different formulations will be standardized for CBD dose (30 mg) but will differ in their preparation (e.g. water vs. fat-soluble). At the 5 randomized Visits Not Including A Test Meal venous blood will be sampled at standardized intervals over 4-hours to calculate Vd (L).

GroupValue95% CI
Formulation 12611836405± 7642484
Formulation 21313130100± 6339554
Formulation 72522687960± 16435999
Pharmacokinetic Parameter Tmax of a Formulation 725 After a Standardized Meal Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

At the 2 randomized visits Including a Test Meal, determine if a high-fat meal impacts the time to attain peak circulating concentration Tmax (mins).

GroupValue95% CI
Formulation 725113.6± 70.5
Pharmacokinetic Parameter Cmax of a Formulation 725 After a Standardized Meal Primary · venous blood will be sampled at standardized intervals over: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

At the 2 randomized visits Including a Test Meal, determine if a high-fat meal impacts maximal concentration of circulating CBD Cmax (ng/L).

GroupValue95% CI
Formulation 7252.9± 1.3
Pharmacokinetic Parameter AUC 0-4 of Formulation 725 After a Standardized Meal Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

At the 2 randomized visits Including a Test Meal, determine if a high-fat meal impacts maximal concentration of circulating CBD AUC 0-4 (min x ng/mL).

GroupValue95% CI
Formulation 725397± 167
Pharmacokinetic Parameter t1/2 of Formulation 725 After a Standardized Meal Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

At the 2 randomized visits Including a Test Meal, determine if a high-fat meal impacts maximal concentration of circulating CBD t1/2 (h).

GroupValue95% CI
Formulation 725248.6± 304.6
Pharmacokinetic Parameter Ke of Formulation 725 After a Standardized Meal Primary · venous blood will be sampled at standardized intervals over 4-hours: 0, 10, 20, 30, 45, 60, 120, 180, and 240 minutes and will be analyzed to compare circulating CBD concentration.

At the 2 randomized visits Including a Test Meal, determine if a high-fat meal impacts maximal concentration of circulating CBD Ke (1/h).

GroupValue95% CI
Formulation 7250.005± 0.002

Sponsor's own description

According to a recent consumer poll, over 20 million Americans regularly use cannabidiol (CBD). Moreover, 64 million Americans (over 25% of the population) report trying CBD at least once within the previous 2 years. Since the passing of the 2018 Agriculture Improvement Act, the use of hemp-derived products, such as CBD, is highly prevalent across North America. The acceleration of the use of CBD has outpaced our understanding of the associated potential risks and benefits, and the way it is processed within the body. In the current proposed project, investigators wish to continue our ongoing collaboration with Caliper Foods, a Colorado-based manufacturer of CBD products. The focus of this project is three-fold: (1) investigators will compare the pharmacokinetics of different formulations of ingestible CBD; (2) investigators will examine the potential two-way interaction between a meal and one formulation of ingestible CBD; and, (3) investigators will examine the influence of different formulations of CBD on markers of liver function.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. Cannabidiol and Cannabidiol Metabolites: Pharmacokinetics, Interaction with Food, and Influence on Liver Function.
    Abbotts KSS, Ewell TR, Butterklee HM, Bomar MC, et al · · 2022 · cited 40× · PMID 35631293 · DOI 10.3390/nu14102152

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Other trials of Cannabidiol (CBD) powder formulation

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