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NCT03907280

A Study in Healthy Men That Tests if Taking BI 1265162 by Mouth, Intravenously, or Inhaled Influences the Amount of BI 1265162 in the Blood

Completed Phase 1 Results posted Last updated 6 July 2022
What this trial tests

Phase 1 trial testing BI 1265162 (T1) in Healthy in 12 participants. Completed in 6 December 2019.

Timeline
23 April 2019
Primary endpoint
6 December 2019
6 December 2019

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingnone
Primary purposetreatment
Enrollment12
Start date23 April 2019
Primary completion6 December 2019
Estimated completion6 December 2019
Sites1 location across Germany

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 18 to 50, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Area Under the Concentration-time Curve of BI 1265162 in Plasma Over the Time Interval From 0 Extrapolated to Infinity, Dose-normalized, (AUC0-∞, Norm) Primary · Up to 24 hours following administration of the trial drug, see detailed time frame in the endpoint description.

Area under the concentration-time curve of BI 1265162 in plasma over the time interval from 0 extrapolated to infinity, dose-normalized to 1 µg BI 1265162, (AUC0-∞, norm). Time frame for treatment T1: Within 3 hours before and 30 and 45 minutes, 1, 2, 3, 4, 6, 8, 12 and 24 hours following administration of the trial drug. Time frame for treatment T2 and T3: Within 3 hours before and 2, 5, 10, 15 and 40 minutes, 1, 2, 4, 8, 10, 12 and 24 hours following administration of the trial drug. Time frame for treatment R: Within 3 hours (h) before and 5, 30 and 59 minutes (min), 1 h 5 min, 1 h 10

GroupValue95% CI
BI 1265162 as Infusion (R)44.63± NA
BI 1265162 as Oral Solution (T1)0.22± NA
BI 1265162 for Inhalation With Activated Charcoal (T2)17.97± NA
BI 1265162 for Inhalation Without Activated Charcoal (T3)17.96± NA

Adverse events — posted to ClinicalTrials.gov

Time frame: For Serious and Other Adverse Events: On-treatment period, that is, from administration of the respective formulation of BI 1265162 until the end of the residual effect period, up to 2 days. For All-Cause Mortality: Each on-treatment period + Follow-up period, i.e. up to 48 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

BI 1265162 as Infusion (R)
Serious: 0/12 (0%)
Deaths: 0/12
BI 1265162 as Oral Solution (T1)
Serious: 1/12 (8%)
Deaths: 0/12
BI 1265162 for Inhalation With Activated Charcoal (T2)
Serious: 0/11 (0%)
Deaths: 0/11
BI 1265162 for Inhalation Without Activated Charcoal (T3)
Serious: 0/12 (0%)
Deaths: 0/12

Serious adverse events (1 terms)

ReactionSystemBI 1265162 as Infusion (R)BI 1265162 as Oral Solutio…BI 1265162 for Inhalation …BI 1265162 for Inhalation …
Vestibular disorderEar and labyrinth disorders
Other adverse events (2 terms — click to expand)

ReactionSystemBI 1265162 as Infusion (R)BI 1265162 as Oral Solutio…BI 1265162 for Inhalation …BI 1265162 for Inhalation …
VomitingGastrointestinal disorders
HeadacheNervous system disorders

Most-reported serious reactions: Vestibular disorder.

Data from ClinicalTrials.gov NCT03907280 adverse events section.

Sponsor's own description

The main objective of this trial is to investigate the absolute bioavailability of BI 1265162 following administration of oral solution and inhaled (with and without charcoal) via Respimat.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. First clinical trials of the inhaled epithelial sodium channel inhibitor BI 1265162 in healthy volunteers.
    Mackie A, Rascher J, Schmid M, Endriss V, et al · · 2021 · cited 8× · PMID 33569494 · DOI 10.1183/23120541.00447-2020

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT03907280.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing