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NCT03794323

A Study in Healthy Men to Find Out How Well Different Doses of BI 764122 Are Tolerated and Whether Food Affects the Amount of BI 764122 in the Blood

Completed Phase 1 Results posted Last updated 1 May 2023
What this trial tests

Phase 1 trial testing BI 764122 in Healthy in 76 participants. Completed in 12 August 2019.

Timeline
30 January 2019
Primary endpoint
12 August 2019
12 August 2019

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingsingle
Primary purposetreatment
Enrollment76
Start date30 January 2019
Primary completion12 August 2019
Estimated completion12 August 2019
Sites1 location across Belgium

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 18 to 50, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Percentage of Subjects With Drug-related Adverse Events Primary · From drug administration until 11 days thereafter for both single rising doses and food effect parts.

Percentage of subjects with drug-related adverse events.

GroupValue95% CI
Placebo6.3
4 mg BI 7641220.0
12 mg BI 76412216.7
25 mg BI 7641220.0
50 mg BI 7641220.0
100 mg BI 7641220.0
200 mg BI 7641220.0
300 mg BI 7641220.0
400 mg BI 7641220.0
50 mg BI 764122 Fasted8.3
50 mg BI 764122 Fed8.3
Area Under the Concentration-time Curve of BI 764122 in Plasma Over the Time Interval From 0 Extrapolated to Infinity (AUC0-inf) Secondary · Within 30 minutes (min) before and 10, 20, 30, 45min and 1 hour (h), 1h 30min, 2, 3, 4, 6, 8, 10, 12, 24, 34, 48, 72, 96 and 120 h post administration.

Area under the concentration-time curve of BI 764122 in plasma over the time interval from 0 extrapolated to infinity (AUC0-inf).

GroupValue95% CI
4 mg BI 764122534± 19.0
12 mg BI 7641221530± 33.3
25 mg BI 7641222850± 15.1
50 mg BI 7641225260± 23.5
100 mg BI 7641229810± 14.1
200 mg BI 76412219400± 14.4
300 mg BI 76412229600± 12.2
400 mg BI 76412245700± 17.4
50 mg BI 764122 Fasted6000± 20.5
50 mg BI 764122 Fed5810± 20.5
Maximum Measured Concentration of BI 764122 in Plasma (Cmax) Secondary · Within 30 minutes (min) before and 10, 20, 30, 45min and 1 hour (h), 1h 30min, 2, 3, 4, 6, 8, 10, 12, 24, 34, 48, 72, 96 and 120 h post administration.

Maximum measured concentration of BI 764122 in plasma (Cmax).

GroupValue95% CI
4 mg BI 764122154± 22.9
12 mg BI 764122565± 16.7
25 mg BI 7641221280± 35.3
50 mg BI 7641222550± 24.9
100 mg BI 7641224410± 45.6
200 mg BI 7641228090± 19.3
300 mg BI 76412213300± 48.4
400 mg BI 76412218600± 21.1
50 mg BI 764122 Fasted2610± 46.3
50 mg BI 764122 Fed1510± 35.3

Adverse events — posted to ClinicalTrials.gov

Time frame: From drug administration until 11 days thereafter for both single rising doses and food effect parts.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Placebo
Serious: 0/16 (0%)
Deaths: 0/16
4 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
12 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
25 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
50 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
100 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
200 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
300 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
400 mg BI 764122
Serious: 0/6 (0%)
Deaths: 0/6
50 mg BI 764122 Fasted
Serious: 0/12 (0%)
Deaths: 0/12
50 mg BI 764122 Fed
Serious: 0/12 (0%)
Deaths: 0/12
Other adverse events (16 terms — click to expand)

ReactionSystemPlacebo4 mg BI 76412212 mg BI 76412225 mg BI 76412250 mg BI 764122100 mg BI 764122200 mg BI 764122300 mg BI 764122400 mg BI 76412250 mg BI 764122 Fasted50 mg BI 764122 Fed
HeadacheNervous system disorders
Abdominal discomfortGastrointestinal disorders
DiarrhoeaGastrointestinal disorders
Epigastric discomfortGastrointestinal disorders
Abdominal distensionGastrointestinal disorders
Abdominal painGastrointestinal disorders
AstheniaGeneral disorders
Vessel puncture site haematomaGeneral disorders
Influenza like illnessGeneral disorders
ConjunctivitisInfections and infestations
Neck painMusculoskeletal and connective tissue disorders
DizzinessNervous system disorders
ParaesthesiaNervous system disorders
Skin irritationSkin and subcutaneous tissue disorders
Supraventricular tachycardiaCardiac disorders
EpistaxisRespiratory, thoracic and mediastinal disorders

Data from ClinicalTrials.gov NCT03794323 adverse events section.

Sponsor's own description

The main objectives of this trial are to investigate safety, tolerability and pharmacokinetics (PK) of BI 764122 in healthy male subjects following oral administration of single rising doses. The objective of the food effect (FE) part is to investigate the relative bioavailability of BI 764122 under fed and fasted conditions.

Publications & conference data

No peer-reviewed publications indexed yet for this trial. Completed trials usually publish results within 12-18 months.

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing