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NCT03693625

A Study to Evaluate the Long-term Safety and Efficacy of Fenebrutinib in Participants Previously Enrolled in a Fenebrutinib Chronic Spontaneous Urticaria (CSU) Study

Terminated Phase 2 Results posted Last updated 25 September 2020
What this trial tests

Phase 2 trial testing GDC-0853 in Urticaria in 31 participants. Terminated before completion.

Timeline
27 September 2018
Primary endpoint
23 October 2019
23 October 2019

Quick facts

Lead sponsorGenentech, Inc.
PhasePhase 2
StatusTerminated
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment31
Start date27 September 2018
Primary completion23 October 2019
Estimated completion23 October 2019
Sites10 locations across United States

Drugs / interventions tested

Conditions studied

Sponsor

Genentech, Inc. — full company profile →

Who can join

Adults 18 to 75, any sex, with Urticaria. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Percentage of Participants With Adverse Events (AEs) Primary · Baseline up until 4 weeks after the last dose of study drug (up to 10 months).

An Adverse Event (AE) is any untoward medical occurrence in a participant administered a pharmaceutical product and which does not necessarily have to have a causal relationship with the treatment. An Adverse Event can therefore be any unfavorable and unintended sign (including abnormal laboratory values or abnormal clinical test results), symptom, or disease temporally associated with the use of a pharmaceutical product, whether or not considered related to the pharmaceutical product. Preexisting conditions which worsen during a study are also considered as Adverse Events.

GroupValue95% CI
Parent Study: GDC-085360.9
Parent Study: Placebo62.5
Plasma Concentrations of Fenebrutinib (GDC-0853) at Specified Timepoints Secondary · Week 1 Day 1; Weeks 12 and 24; Study Completion/Early Discontinuation

Plasma Concentration Data for fenebrutinib (GDC-0853) will be tabulated and summarised by visits. Descriptive summary statistics for Arithmetic Mean and Standard Deviation will be presented.

Week 1 Day 1
GroupValue95% CI
Parent Study: GDC-0853NA± NA
Parent Study: PlaceboNA± NA
Week 12
GroupValue95% CI
Parent Study: GDC-0853192± 181
Parent Study: Placebo190± 278
Week 24
GroupValue95% CI
Parent Study: GDC-0853130± 63.8
Parent Study: Placebo467± 480
Study Completion/Early Discontinuation
GroupValue95% CI
Parent Study: GDC-0853NA± NA
Parent Study: PlaceboNA± NA

Adverse events — posted to ClinicalTrials.gov

Time frame: Baseline up until 4 weeks after the last dose of study drug (up to 10 months).. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Parent Study: GDC-0853
Serious: 0/23 (0%)
Deaths: 0/23
Parent Study: Placebo
Serious: 0/8 (0%)
Deaths: 0/8
Other adverse events (20 terms — click to expand)

ReactionSystemParent Study: GDC-0853Parent Study: Placebo
URTICARIASkin and subcutaneous tissue disorders
INCREASED TENDENCY TO BRUISEBlood and lymphatic system disorders
DIARRHOEAGastrointestinal disorders
DYSPEPSIAGastrointestinal disorders
GASTROOESOPHAGEAL REFLUX DISEASEGastrointestinal disorders
ABSCESS LIMBInfections and infestations
ORAL HERPESInfections and infestations
SKIN INFECTIONInfections and infestations
ALANINE AMINOTRANSFERASE INCREASEDInvestigations
ASPARTATE AMINOTRANSFERASE INCREASEDInvestigations
BLOOD CREATINE PHOSPHOKINASE INCREASEDInvestigations
BACK PAINMusculoskeletal and connective tissue disorders
MUSCULOSKELETAL CHEST PAINMusculoskeletal and connective tissue disorders
MYALGIAMusculoskeletal and connective tissue disorders
HEADACHENervous system disorders
MIGRAINENervous system disorders
HAEMATURIARenal and urinary disorders
COUGHRespiratory, thoracic and mediastinal disorders
PRURITUSSkin and subcutaneous tissue disorders
RASHSkin and subcutaneous tissue disorders

Data from ClinicalTrials.gov NCT03693625 adverse events section.

Sponsor's own description

This is a Phase II, multicenter, open-label extension (OLE) study to evaluate the long-term safety and efficacy of fenebrutinib in participants with Chronic Spontaneous Urticaria (CSU) who have completed the treatment period in a fenebrutinib CSU parent study. Participants may enroll in this OLE study at any time after completing the treatment period of the parent study. Participants will receive open-label fenebrutinib at a dose of 200 milligram (mg) orally twice a day. Treatment may continue until the end of the study.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Small Molecule NF-κB Pathway Inhibitors in Clinic.
    Ramadass V, Vaiyapuri T, Tergaonkar V. · · 2020 · cited 154× · PMID 32708302 · DOI 10.3390/ijms21145164
  2. Bruton's Tyrosine Kinase (BTK) Inhibitors and Autoimmune Diseases: Making Sense of BTK Inhibitor Specificity Profiles and Recent Clinical Trial Successes and Failures.
    Ringheim GE, Wampole M, Oberoi K. · · 2021 · cited 100× · PMID 34803999 · DOI 10.3389/fimmu.2021.662223
  3. Bruton's tyrosine kinase inhibition-An emerging therapeutic strategy in immune-mediated dermatological conditions.
    Mendes-Bastos P, Brasileiro A, Kolkhir P, Frischbutter S, et al · · 2022 · cited 67× · PMID 35175630 · DOI 10.1111/all.15261
  4. The Development of BTK Inhibitors: A Five-Year Update.
    Tasso B, Spallarossa A, Russo E, Brullo C. · · 2021 · cited 40× · PMID 34885993 · DOI 10.3390/molecules26237411
  5. Btk Inhibitors: A Medicinal Chemistry and Drug Delivery Perspective.
    Brullo C, Villa C, Tasso B, Russo E, et al · · 2021 · cited 36× · PMID 34299259 · DOI 10.3390/ijms22147641
  6. Bruton's Tyrosine Kinase Inhibition in Multiple Sclerosis.
    Schneider R, Oh J. · · 2022 · cited 30× · PMID 36301434 · DOI 10.1007/s11910-022-01229-z
  7. Current and emerging treatments for chronic spontaneous urticaria.
    Johal KJ, Saini SS. · · 2020 · cited 26× · PMID 31494233 · DOI 10.1016/j.anai.2019.08.465
  8. Emerging Therapies in Chronic Spontaneous Urticaria.
    Min TK, Saini SS. · · 2019 · cited 21× · PMID 31172716 · DOI 10.4168/aair.2019.11.4.470

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