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NCT03588390

This Study in Healthy Men Tests How Different Doses of BI 1323495 Are Taken up in the Body and How Well They Are Tolerated.

Completed Phase 1 Results posted Last updated 22 February 2024
What this trial tests

Phase 1 trial testing BI 1323495 in Healthy in 63 participants. Completed in 14 November 2018.

Timeline
31 July 2018
Primary endpoint
14 November 2018
14 November 2018

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingsingle
Primary purposetreatment
Enrollment63
Start date31 July 2018
Primary completion14 November 2018
Estimated completion14 November 2018
Sites1 location across Germany

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 18 to 45, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Percentage of Participants With Drug-related Adverse Events Primary · From drug administration until end of trial, up to 15 days.

Percentage of participants with drug-related adverse events.

GroupValue95% CI
Placebo Matching BI 13234956.7
BI 1323495 Dose Group 150.0
BI 1323495 Dose Group 233.3
BI 1323495 Dose Group 30.0
BI 1323495 Dose Group 416.7
BI 1323495 Dose Group 50.0
BI 1323495 Dose Group 616.7
BI 1323495 Dose Group 750.0
BI 1323495 Dose Group 816.7
Area Under the Concentration-time Curve of BI 1323495 in Plasma Over the Time Interval From 0 Extrapolated to Infinity (AUC0-∞) Secondary · 1 hour (h) before drug administration and 1, 2, 3, 4, 6, 7, 8, 9, 10, 12, 24, 34, 48, 72 and 96 h and additionally 4.75, 5.5, 6.5, 7.5 h for dose group 1/2/3 and 0.333, 0.667, 1.5, 5 h for dose group 4/5/6/7/8 after drug administration.

Area under the concentration-time curve of BI 1323495 in plasma over the time interval from 0 extrapolated to infinity (AUC0-∞) after single oral administration of BI 1323495.

GroupValue95% CI
BI 1323495 Dose Group 1143± 102.0
BI 1323495 Dose Group 2883± 118.0
BI 1323495 Dose Group 3824± 77.7
BI 1323495 Dose Group 42360± 73.5
BI 1323495 Dose Group 53710± 69.4
BI 1323495 Dose Group 63120± 140.0
BI 1323495 Dose Group 71780± 102.0
BI 1323495 Dose Group 83820± 71.9
Maximum Measured Concentration of BI 1323495 in Plasma (Cmax) Secondary · 1 hour (h) before drug administration and 1, 2, 3, 4, 6, 7, 8, 9, 10, 12, 24, 34, 48, 72 and 96 h and additionally 4.75, 5.5, 6.5, 7.5 h for dose group 1/2/3 and 0.333, 0.667, 1.5, 5 h for dose group 4/5/6/7/8 after drug administration.

Maximum measured concentration of BI 1323495 in plasma (Cmax) after single oral administration of BI 1323495.

GroupValue95% CI
BI 1323495 Dose Group 110.5± 66.3
BI 1323495 Dose Group 259.4± 147.0
BI 1323495 Dose Group 3145.0± 74.8
BI 1323495 Dose Group 4229.0± 127.0
BI 1323495 Dose Group 5179.0± 152.0
BI 1323495 Dose Group 6136.0± 74.2
BI 1323495 Dose Group 7195.0± 90.8
BI 1323495 Dose Group 8195.0± 90.8

Adverse events — posted to ClinicalTrials.gov

Time frame: From drug administration until end of trial, up to 15 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Placebo Matching BI 1323495
Serious: 0/15 (0%)
Deaths: 0/15
BI 1323495 Dose Group 1
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 2
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 3
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 4
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 5
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 6
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 7
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Dose Group 8
Serious: 0/6 (0%)
Deaths: 0/6
BI 1323495 Total
Serious: 0/48 (0%)
Deaths: 0/48
Other adverse events (10 terms — click to expand)

ReactionSystemPlacebo Matching BI 1323495BI 1323495 Dose Group 1BI 1323495 Dose Group 2BI 1323495 Dose Group 3BI 1323495 Dose Group 4BI 1323495 Dose Group 5BI 1323495 Dose Group 6BI 1323495 Dose Group 7BI 1323495 Dose Group 8BI 1323495 Total
HeadacheNervous system disorders
DiarrhoeaGastrointestinal disorders
FatigueGeneral disorders
MalaiseGeneral disorders
Unevaluable eventGeneral disorders
NasopharyngitisInfections and infestations
RhinitisInfections and infestations
Alanine aminotransferase increasedInvestigations
Glutamate dehydrogenase increasedInvestigations
Musculoskeletal stiffnessMusculoskeletal and connective tissue disorders

Data from ClinicalTrials.gov NCT03588390 adverse events section.

Sponsor's own description

The primary objective of this trial is to investigate the safety and tolerability of BI 1323495 in healthy male subjects following oral administration of single rising doses. Secondary objectives are the exploration of the pharmacokinetics (PK) including dose proportionality and pharmacodynamics (PD) of BI 1323495 after single dosing and the assessment of the PK/PD relationship.

Publications & conference data

No peer-reviewed publications indexed yet for this trial. Completed trials usually publish results within 12-18 months.

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Other trials of BI 1323495

Trials testing the same drug.

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Other Boehringer Ingelheim trials

Trials by the same sponsor.

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