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NCT03179436

Study of Quavonlimab (MK-1308) in Combination With Pembrolizumab (MK-3475) in Advanced Solid Tumors (MK-1308-001)

Completed Phase 1, PHASE2 Results posted Last updated 8 April 2025
What this trial tests

Phase 1, PHASE2 trial testing Quavonlimab in Advanced Solid Tumors in 415 participants. Completed in 8 April 2024.

Timeline
2 July 2017
Primary endpoint
8 April 2024
8 April 2024

Quick facts

Lead sponsorMerck Sharp & Dohme LLC
PhasePhase 1, PHASE2
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designparallel
Maskingnone
Primary purposetreatment
Enrollment415
Start date2 July 2017
Primary completion8 April 2024
Estimated completion8 April 2024
Sites53 locations across France, Italy, Japan, New Zealand, Greece, South Africa, Chile, Sweden

Drugs / interventions tested

Conditions studied

Sponsor

Merck Sharp & Dohme LLC — full company profile →

Who can join

18 and older, any sex, with Advanced Solid Tumors. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Percentage of Participants With ≥1 Dose Limiting Toxicity (DLT) Primary · Up to 6 weeks

DLT was defined as toxicity that is possibly, probably, or definitely related to study therapy and may result in a change in the given dose. DLTs include Grade (Gr)4 non-hematologic toxicity (not laboratory); Gr 4 hematologic toxicity lasting ≥7 days (except thrombocytopenia); most non-hematologic AEs ≥ Gr 3 in severity; any Gr 3 or Gr 4 non-hematologic laboratory value that requires clinically significant medical intervention, leads to hospitalization, persists for \>1 week, or results in a drug-induced liver injury; Gr 3 or Gr 4 febrile neutropenia; a prolonged delay in initiating Cycle 2 or

GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W0.00.0 – 10.9
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W13.34.9 – 26.6
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W0.00.0 – 18.2
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W7.53.3 – 14.0
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W5.01.7 – 10.8
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W10.05.0 – 17.1
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W10.05.0 – 17.1
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W7.11.4 – 19.4
Number of Participants With ≥1 Adverse Event (AE) Primary · Up to approximately 77 months

An AE is defined as any untoward medical occurrence in a participant administered a pharmaceutical product temporally associated with the use of study treatment, whether or not considered related to the study treatment. Per protocol, no analysis was planned for the cross over phase. The number of participants who experienced an AE are presented.

GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W14
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W17
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W8
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W39
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W38
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W40
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W38
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W14
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin104
Arm G: MK-1308 25 mg Q6W37
Arm I: MK-1308A Q6W (Co-form)28
Arm K: MK-1308A Q6W (Co-form)18
Number of Participants Discontinuing Study Treatment Due to an AE Primary · Up to approximately 26 months

An AE is defined as any untoward medical occurrence in a participant administered a pharmaceutical product temporally associated with the use of study treatment, whether or not considered related to the study treatment. Per protocol, no analysis was planned for the cross over phase. The number of participants who discontinued study treatment due to an AE are presented.

GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W4
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W3
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W7
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W7
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W17
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W7
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W6
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin14
Arm G: MK-1308 25 mg Q6W1
Arm I: MK-1308A Q6W (Co-form)4
Arm K: MK-1308A Q6W (Co-form)2
Efficacy Expansion: Objective Response Rate (ORR) as Assessed by Blinded Independent Central Review (BICR) Based on Adjusted Response Evaluation Criteria in Solid Tumors Version 1.1 (RECIST v1.1) Primary · Up to approximately 72 months

ORR is defined as the percentage of participants with Complete Response (CR: disappearance of all target lesions) or Partial Response (PR: at least a 30% decrease in the sum of diameters of target lesions) per adjusted Response Evaluation Criteria In Solid Tumors Version 1.1 (RECIST 1.1). The percentage of participants who experience CR or PR in the concurrent randomized subset as assessed by Blinded Independent Central Review (BICR) will be presented. Per protocol, only data for arms F and G were presented for this endpoint.

GroupValue95% CI
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin4.90.6 – 16.5
Arm G: MK-1308 25 mg Q6W2.50.1 – 13.2
Area Under the Plasma Concentration Time Curve (AUC) of Pembrolizumab Secondary · At designated time points up to - Cohorts 1-3: Day 15 Cycle 3, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F: Day 21 Cycle 3, Arm I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

AUC was defined as a measure of pembrolizumab exposure that was calculated as the product of plasma drug concentration and time after drug administration. AUC determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for participants in arm G and cross over phase. AUC of pembrolizumab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 2 and 3. Arms A, B, C, D, E: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2, 3. Arm F: Predose and Postdose on Day 1 and 21

Cycle 1
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W608± 24.6
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W620± 25.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W627± 20.6
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W642± 23.9
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W554± 15.6
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin2050± 33.6
Arm I: MK-1308A Q6W (Co-form)2250± 18.7
Arm K: MK-1308A Q6W (Co-form)1610± 25.0
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W729± 18.3
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W546± 40.5
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W727± 24.5
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W788± 24.7
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W854± 19.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W822± 25.0
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W877± 28.3
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W794± 18.0
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin2370± 40.6
Arm I: MK-1308A Q6W (Co-form)2820± 29.7
Arm K: MK-1308A Q6W (Co-form)1770± 34.4
Cycle 3
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W911± 22.7
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W971± 22.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W944± 26.0
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W1050± 20.8
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W872± 16.3
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin2410± 29.5
Arm I: MK-1308A Q6W (Co-form)3410± 16.1
Arm K: MK-1308A Q6W (Co-form)2440± 39.8
Maximum Concentration (Cmax) of Pembrolizumab Secondary · At designated time points up to - Cohorts 1-3: Day 15 Cycle 3, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F: Day 21 Cycle 3, Arm I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

Cmax was defined as the maximum concentration of pembrolizumab observed in plasma. Cmax determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for participants in arm G and cross over phase. Cmax of pembrolizumab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 2 and 3. Arms A, B, C, D, E: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2, 3. Arm F: Predose and Postdose on Day 1 and 21 on Cycles 1, 2, 3. Arm I: Predose and Postdose on Day 1 and 21 on Cyc

Cycle 1
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W71.8± 24.0
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W77.1± 26.7
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W74.0± 27.8
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W73.6± 22.3
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W70.9± 35.3
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin149± 29.1
Arm I: MK-1308A Q6W (Co-form)149± 23.8
Arm K: MK-1308A Q6W (Co-form)128± 21.9
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W79.8± 31.3
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W82.3± 32.3
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W78.7± 32.4
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W82.9± 20.2
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W88.2± 20.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W83.9± 23.2
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W90.4± 23.7
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W84.8± 18.6
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin150± 28.9
Arm I: MK-1308A Q6W (Co-form)164± 22.8
Arm K: MK-1308A Q6W (Co-form)139± 20.5
Cycle 3
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W93.9± 21.0
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W74.9± 28.1
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W88.6± 12.2
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W84.2± 16.9
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W92.3± 27.5
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W91.8± 21.7
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W98.0± 27.4
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W84.5± 13.8
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin153± 22.1
Arm I: MK-1308A Q6W (Co-form)168± 22.3
Arm K: MK-1308A Q6W (Co-form)138± 31.1
Minimum Concentration (Cmin) of Pembrolizumab Secondary · At designated time points up to - Cohorts 1-3: Day 1 Cycle 4, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F: Day 21 Cycle 3, Arm I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

Cmin was defined as the minimum or "trough" concentration of pembrolizumab observed after its administration and just prior to the administration of a subsequent dose. Cmin determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for participants in arm G and cross over phase. Cmin of pembrolizumab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 2 and 3, Day 1 on Cycle 4. Arms A, B, C, D, E: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2, 3. Arm F: Pre

Cycle 1
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W13.30.00 – 22.3
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W13.13.93 – 24.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W14.35.59 – 90.4
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W15.66.35 – 35.9
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W11.54.77 – 18.0
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin21.91.89 – 143
Arm I: MK-1308A Q6W (Co-form)19.57.25 – 35.8
Arm K: MK-1308A Q6W (Co-form)14.45.74 – 26.0
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W18.311.3 – 27.8
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W11.30.00 – 28.1
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W19.09.21 – 24.6
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W19.66.62 – 37.4
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W24.39.06 – 34.6
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W20.49.19 – 44.9
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W25.210.1 – 55.1
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W18.98.52 – 25.5
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin23.10.0266 – 51.6
Arm I: MK-1308A Q6W (Co-form)30.016.2 – 60.4
Arm K: MK-1308A Q6W (Co-form)22.58.74 – 37.1
Cycle 3
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W25.713.7 – 40.3
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W27.512.4 – 42.2
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W25.511.3 – 98.2
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W29.310.4 – 56.7
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W27.714.5 – 30.5
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin24.52.22 – 127
Arm I: MK-1308A Q6W (Co-form)34.018.9 – 72.2
Arm K: MK-1308A Q6W (Co-form)26.67.74 – 32.6
Cycle 4
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W34.329.8 – 39.9
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W14.10.00 – 38.1
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W23.523.5 – 23.5
Area Under the Plasma Concentration Time Curve (AUC) of Quavonlimab (MK-1308) Secondary · At designated time points up to - Cohorts 1-3: Day 15 Cycle 3, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F, G, I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

AUC was defined as a measure of quavonlimab exposure that was calculated as the product of plasma drug concentration and time after drug administration. AUC determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for the cross over phase. AUC of quavonlimab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2 and 3. Arms A, B, C, D, E: Days 1, 8, 15 on Cycles 1, 2, 3. Arms F, G and I: Predose and Postdose on Day 1 and 21 on Cycles 1, 2, 3. Arm K: Days 1, 2,

Cycle 1
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W68.2± 17.7
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W160± 19.5
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W510± 25.7
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W55.0± 26.6
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W69.6± 33.5
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W199± 36.2
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W222± 39.7
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W178± 17.6
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin77.1± 32.7
Arm G: MK-1308 25 mg Q6W92.8± 38.1
Arm I: MK-1308A Q6W (Co-form)106± 34.7
Arm K: MK-1308A Q6W (Co-form)85.8± 24.2
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W91.5± 19.9
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W178± 53.9
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W751± 23.4
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W73.6± 26.4
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W192± 17.7
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin94.4± 43.9
Arm G: MK-1308 25 mg Q6W65.9± 27.8
Arm I: MK-1308A Q6W (Co-form)96.1± 39.7
Arm K: MK-1308A Q6W (Co-form)86.0± 47.7
Cycle 3
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W64.3± 56.5
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W59.4± 74.9
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W182± 75.1
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W193± 90.8
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W186± 22.1
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin95.2± 63.4
Arm G: MK-1308 25 mg Q6W95.0± 58.2
Arm I: MK-1308A Q6W (Co-form)72.1± 9.92
Arm K: MK-1308A Q6W (Co-form)92.3± 60.2
Maximum Concentration (Cmax) of Quavonlimab Secondary · At designated time points up to - Cohorts 1-3: Day 15 Cycle 3, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F, G, I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

Cmax was defined as the maximum concentration of quavonlimab observed in plasma. Cmax determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for the cross over phase. Cmax of quavonlimab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2 and 3. Arms A, B, C, D, E: Days 1, 8, 15 on Cycles 1, 2, 3. Arms F, G and I: Predose and Postdose on Day 1 and 21 on Cycles 1, 2, 3. Arm K: Days 1, 2, 8, 15, 21 on Cycles 1, 2; Days 1, 21 on Cycle 3. Each cycle is 21 day

Cycle 1
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W8.23± 26.1
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W22.5± 29.8
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W68.3± 17.2
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W7.28± 30.6
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W8.02± 29.5
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W23.4± 24.3
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W24.1± 30.1
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W25.0± 20.6
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin7.25± 26.4
Arm G: MK-1308 25 mg Q6W7.42± 30.4
Arm I: MK-1308A Q6W (Co-form)8.06± 26.5
Arm K: MK-1308A Q6W (Co-form)8.23± 26.7
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W9.41± 20.4
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W23.5± 25.1
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W71.9± 29.0
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W8.58± 22.4
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W26.3± 24.7
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin7.65± 25.3
Arm G: MK-1308 25 mg Q6W7.22± 29.3
Arm I: MK-1308A Q6W (Co-form)8.17± 26.2
Arm K: MK-1308A Q6W (Co-form)7.99± 29.7
Cycle 3
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W9.11± 24.7
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W23.3± 48.0
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W88.3± 16.0
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W7.72± 27.7
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W6.98± 43.7
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W22.7± 33.1
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W24.2± 50.4
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W27.2± 10.2
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin7.94± 29.6
Arm G: MK-1308 25 mg Q6W6.65± 32.7
Arm I: MK-1308A Q6W (Co-form)7.25± 21.9
Arm K: MK-1308A Q6W (Co-form)7.94± 35.4
Minimum Concentration (Cmin) of Quavonlimab Secondary · At designated time points up to - Cohorts 1-3: Day 15 Cycle 3, Arms A, B, C, D, E: Day 15 Cycle 3, Arm F, G, I: Day 21 Cycle 3, Arm K: Day 21 Cycle 3. Each cycle is 21 days.

Cmin was defined as the minimum or "trough" concentration of quavonlimab observed after its administration and just prior to the administration of a subsequent dose. Cmin determined by blood samples collected pre-dose and at designated timepoints post-dose are presented. Per protocol, no analysis was planned for the cross over phase. Cmin of quavonlimab is presented. Blood sampling was taken for Cohorts 1-3: Predose and Postdose on Days 1, 8, 15 on Cycles 1, 2 and 3. Arms A, B, C, D, E: Days 1, 8, 15 on Cycles 1, 2, 3. Arms F, G and I: Predose and Postdose on Day 1 and 21 on Cycles 1, 2, 3. Ar

Cycle 1
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1.440.00 – 2.11
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W3.290.00 – 6.86
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W8.011.51 – 17.8
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1.050.00 – 1.80
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W0.000.00 – 0.00
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W0.000.00 – 3.44
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W15.66.35 – 35.9
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W3.200.00 – 5.26
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin0.000.00 – 1.65
Arm G: MK-1308 25 mg Q6W0.000.00 – 1.26
Arm I: MK-1308A Q6W (Co-form)0.000.00 – 2.02
Arm K: MK-1308A Q6W (Co-form)0.000.00 – 1.32
Cycle 2
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1.750.00 – 3.10
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W2.830.00 – 10.3
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W17.41.73 – 19.2
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1.170.00 – 2.73
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W25.210.1 – 55.1
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W3.401.35 – 6.32
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin0.000.00 – 8.23
Arm G: MK-1308 25 mg Q6W0.000.00 – 2.09
Arm I: MK-1308A Q6W (Co-form)0.000.00 – 1.68
Arm K: MK-1308A Q6W (Co-form)0.000.00 – 1.65
Cycle 3
GroupValue95% CI
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W1.911.91 – 1.91
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1.420.00 – 2.86
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W0.000.00 – 0.00
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W0.000.00 – 3.10
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W29.310.4 – 56.7
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W2.912.21 – 5.77
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin0.000.00 – 7.50
Arm G: MK-1308 25 mg Q6W0.000.00 – 7.20
Arm I: MK-1308A Q6W (Co-form)0.000.00 – 2.37
Arm K: MK-1308A Q6W (Co-form)0.000.00 – 1.05
Number of Participants With Pembrolizumab Anti-drug Antibodies (ADAs) Secondary · Cohorts 1-3: Predose and day 1 of cycles 2, 3, 5, 6, 7, 9 and every 4 cycles up to 35 cycles. Arms A-E: Predose and day 1 of cycles 1-5, 6, 8 and every 4 cycles up to 35 cycles. Arms F, I, K: Predose and day 1 of cycles 1, 2, 3, 4. Each cycle is 21 days.

Non-Treatment emergent (TE) ADA refers to presence of ADAs (as determined by assay) in the absence of treatment with pembrolizumab (i.e., at predose). Evaluable participants (used as the denominator for analysis) are the total number of negative, inconclusive, and positive participants (non-treatment emergent, treatment emergent and treatment boosted). Inconclusive participants are the number of participants with no positive ADA samples present and the drug concentration in the last sample above the drug tolerance level. ADA determined by blood samples collected pre-dose and at designated time

Evaluable
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W12
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W13
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W5
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W36
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W39
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W37
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W35
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W11
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin103
Arm I: MK-1308A Q6W (Co-form)23
Arm K: MK-1308A Q6W (Co-form)20
Negative
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W12
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W12
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W5
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W31
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W33
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W33
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W31
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W10
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin94
Arm I: MK-1308A Q6W (Co-form)20
Arm K: MK-1308A Q6W (Co-form)13
Non - TE Neutralizing Antibody (NAB) NEG (Negative)
GroupValue95% CI
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W1
Arm I: MK-1308A Q6W (Co-form)1
TE NAB NEG
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W4
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W4
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W3
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W4
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W1
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin3
Arm K: MK-1308A Q6W (Co-form)2
TE NAB Positive (POS)
GroupValue95% CI
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W1
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W1
Arm K: MK-1308A Q6W (Co-form)1
Inconclusive
GroupValue95% CI
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W2
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin5
Arm I: MK-1308A Q6W (Co-form)2
Arm K: MK-1308A Q6W (Co-form)4
Treatment Boosted (TB) NAB NEG
GroupValue95% CI
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin1
Arm K: MK-1308A Q6W (Co-form)0
Number of Participants With Quavonlimab Anti-drug Antibodies (ADAs) Secondary · Cohort 1-3: Predose and day 1 of cycles 2, 3, 5, 6, 7, 9 and every 4 cycles up to 35 cycles. Arms A-E: Predose and day 1 of cycle 1-5, 6, 8 and every 4 cycles up to 35 cycles. Arms F, G, I, K: Predose and day 1 of cycles 1, 2, 3, 4. Each cycle is 21 days.

Non-Treatment emergent (TE) ADA refers to presence of ADAs (as determined by assay) in the absence of treatment with quavonlimab (i.e., at predose). Evaluable participants (used as the denominator for analysis) are the total number of negative, inconclusive, and positive participants (non-treatment emergent, treatment emergent and treatment boosted (TB)). Inconclusive participants are the number of participants with no positive ADA samples present and the drug concentration in the last sample above the drug tolerance level. ADA determined by blood samples collected pre-dose and at designated t

Evaluable
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W14
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W15
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W8
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W36
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W39
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W37
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W35
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W11
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin102
Arm G: MK-1308 25 mg Q6W38
Arm I: MK-1308A Q6W (Co-form)23
Arm K: MK-1308A Q6W (Co-form)20
Negative
GroupValue95% CI
Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W3
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W7
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W4
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W12
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W6
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W6
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W8
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W4
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin35
Arm G: MK-1308 25 mg Q6W21
Arm I: MK-1308A Q6W (Co-form)8
Arm K: MK-1308A Q6W (Co-form)6
Inconclusive
GroupValue95% CI
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W1
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin2
Arm G: MK-1308 25 mg Q6W1
Arm K: MK-1308A Q6W (Co-form)1
TB NAB MISSING
GroupValue95% CI
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W1
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W1
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin3
Arm G: MK-1308 25 mg Q6W2
Arm K: MK-1308A Q6W (Co-form)2

Adverse events — posted to ClinicalTrials.gov

Time frame: Up to approximately 77 months. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Cohort 1: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W
Serious: 2/14 (14%)
Deaths: 13/14
Cohort 2: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W
Serious: 10/17 (59%)
Deaths: 18/18
Cohort 3: MK-1308 200 mg Q3W + Pembro. 200 mg Q3W
Serious: 4/8 (50%)
Deaths: 7/8
Arm A: MK-1308 25 mg Q3W + Pembro. 200 mg Q3W
Serious: 20/40 (50%)
Deaths: 33/40
Arm B: MK-1308 25 mg Q6W + Pembro. 200 mg Q3W
Serious: 14/40 (35%)
Deaths: 31/40
Arm C: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W
Serious: 23/40 (57%)
Deaths: 32/41
Arm D: MK-1308 75 mg Q6W + Pembro. 200 mg Q3W
Serious: 16/40 (40%)
Deaths: 35/40
Arm E: MK-1308 75 mg Q3W + Pembro. 200 mg Q3W
Serious: 10/14 (71%)
Deaths: 9/14
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin
Serious: 31/111 (28%)
Deaths: 86/111
Arm F: MK-1308 25 mg Q6W + Pembro. 400 mg Q6W Co-admin After Crossover
Serious: 4/21 (19%)
Deaths: 17/21
Arm G: MK-1308 25 mg Q6W
Serious: 9/40 (23%)
Deaths: 16/40
Arm I: MK-1308A Q6W (Co-form)
Serious: 15/29 (52%)
Deaths: 22/29
Arm K: MK-1308A Q6W (Co-form)
Serious: 4/20 (20%)
Deaths: 15/20

Serious adverse events (135 terms)

ReactionSystemCohort 1: MK-1308 25 mg Q3…Cohort 2: MK-1308 75 mg Q3…Cohort 3: MK-1308 200 mg Q…Arm A: MK-1308 25 mg Q3W +…Arm B: MK-1308 25 mg Q6W +…Arm C: MK-1308 75 mg Q6W +…Arm D: MK-1308 75 mg Q6W +…Arm E: MK-1308 75 mg Q3W +…Arm F: MK-1308 25 mg Q6W +…Arm F: MK-1308 25 mg Q6W +…Arm G: MK-1308 25 mg Q6WArm I: MK-1308A Q6W (Co-fo…Arm K: MK-1308A Q6W (Co-fo…
PneumoniaInfections and infestations
PneumonitisRespiratory, thoracic and mediastinal disorders
ColitisGastrointestinal disorders
AnaemiaBlood and lymphatic system disorders
DiarrhoeaGastrointestinal disorders
PyrexiaGeneral disorders
Adrenal insufficiencyEndocrine disorders
EncephalitisInfections and infestations
Septic shockInfections and infestations
Alanine aminotransferase increasedInvestigations
Aspartate aminotransferase increasedInvestigations
Back painMusculoskeletal and connective tissue disorders
Acute kidney injuryRenal and urinary disorders
Chronic obstructive pulmonary diseaseRespiratory, thoracic and mediastinal disorders
Pleural effusionRespiratory, thoracic and mediastinal disorders
PneumothoraxRespiratory, thoracic and mediastinal disorders
Pulmonary embolismRespiratory, thoracic and mediastinal disorders
Autoimmune haemolytic anaemiaBlood and lymphatic system disorders
Febrile neutropeniaBlood and lymphatic system disorders
Mesenteric lymphadenitisBlood and lymphatic system disorders
Acute myocardial infarctionCardiac disorders
Atrial fibrillationCardiac disorders
Atrioventricular block completeCardiac disorders
Cardiac arrestCardiac disorders
Cardiac failureCardiac disorders
Other adverse events (167 terms — click to expand)

ReactionSystemCohort 1: MK-1308 25 mg Q3…Cohort 2: MK-1308 75 mg Q3…Cohort 3: MK-1308 200 mg Q…Arm A: MK-1308 25 mg Q3W +…Arm B: MK-1308 25 mg Q6W +…Arm C: MK-1308 75 mg Q6W +…Arm D: MK-1308 75 mg Q6W +…Arm E: MK-1308 75 mg Q3W +…Arm F: MK-1308 25 mg Q6W +…Arm F: MK-1308 25 mg Q6W +…Arm G: MK-1308 25 mg Q6WArm I: MK-1308A Q6W (Co-fo…Arm K: MK-1308A Q6W (Co-fo…
PruritusSkin and subcutaneous tissue disorders
DiarrhoeaGastrointestinal disorders
FatigueGeneral disorders
NauseaGastrointestinal disorders
RashSkin and subcutaneous tissue disorders
Decreased appetiteMetabolism and nutrition disorders
ConstipationGastrointestinal disorders
ArthralgiaMusculoskeletal and connective tissue disorders
HeadacheNervous system disorders
Abdominal painGastrointestinal disorders
AstheniaGeneral disorders
AnaemiaBlood and lymphatic system disorders
Aspartate aminotransferase increasedInvestigations
Alanine aminotransferase increasedInvestigations
CoughRespiratory, thoracic and mediastinal disorders
HypothyroidismEndocrine disorders
Abdominal pain upperGastrointestinal disorders
Dry mouthGastrointestinal disorders
PyrexiaGeneral disorders
Back painMusculoskeletal and connective tissue disorders
Pain in extremityMusculoskeletal and connective tissue disorders
DyspnoeaRespiratory, thoracic and mediastinal disorders
Oedema peripheralGeneral disorders
InsomniaPsychiatric disorders
Rash maculo-papularSkin and subcutaneous tissue disorders
Skin lesionSkin and subcutaneous tissue disorders
HyperthyroidismEndocrine disorders
Urinary tract infectionInfections and infestations
Weight decreasedInvestigations
HyperglycaemiaMetabolism and nutrition disorders
DizzinessNervous system disorders
VomitingGastrointestinal disorders
Blood alkaline phosphatase increasedInvestigations
C-reactive protein increasedInvestigations
HypoalbuminaemiaMetabolism and nutrition disorders
PneumonitisRespiratory, thoracic and mediastinal disorders
VitiligoSkin and subcutaneous tissue disorders
Upper respiratory tract infectionInfections and infestations
HyperkalaemiaMetabolism and nutrition disorders
HypokalaemiaMetabolism and nutrition disorders

Most-reported serious reactions: Pneumonia, Pneumonitis, Colitis, Anaemia, Diarrhoea, Pyrexia, Adrenal insufficiency, Encephalitis.

Data from ClinicalTrials.gov NCT03179436 adverse events section.

Sponsor's own description

This study will assess the safety, tolerability, pharmacokinetics (PK), and preliminary efficacy of escalating doses of quavonlimab when used in combination with pembrolizumab in participants with advanced solid tumors.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Immunotherapeutic approaches for small-cell lung cancer.
    Iams WT, Porter J, Horn L. · · 2020 · cited 237× · PMID 32055013 · DOI 10.1038/s41571-019-0316-z
  2. Dual blockade immunotherapy targeting PD-1/PD-L1 and CTLA-4 in lung cancer.
    Cheng W, Kang K, Zhao A, Wu Y. · · 2024 · cited 110× · PMID 39068460 · DOI 10.1186/s13045-024-01581-2
  3. Management of early melanoma recurrence despite adjuvant anti-PD-1 antibody therapy<sup>☆</sup>.
    Owen CN, Shoushtari AN, Chauhan D, Palmieri DJ, et al · · 2020 · cited 86× · PMID 32387454 · DOI 10.1016/j.annonc.2020.04.471
  4. Immune evasion in cancer: mechanisms and cutting-edge therapeutic approaches.
    Tufail M, Jiang CH, Li N. · · 2025 · cited 82× · PMID 40739089 · DOI 10.1038/s41392-025-02280-1
  5. Immune Checkpoint Inhibitors in Cancer Therapy-How to Overcome Drug Resistance?
    Lao Y, Shen D, Zhang W, He R, et al · · 2022 · cited 53× · PMID 35892835 · DOI 10.3390/cancers14153575
  6. Microsatellite Instability in Colorectal Cancers: Carcinogenesis, Neo-Antigens, Immuno-Resistance and Emerging Therapies.
    Randrian V, Evrard C, Tougeron D. · · 2021 · cited 51× · PMID 34205397 · DOI 10.3390/cancers13123063
  7. Standard-Dose Pembrolizumab Plus Alternate-Dose Ipilimumab in Advanced Melanoma: KEYNOTE-029 Cohort 1C, a Phase 2 Randomized Study of Two Dosing Schedules.
    Long GV, Robert C, Butler MO, Couture F, et al · · 2021 · cited 32× · PMID 34210681 · DOI 10.1158/1078-0432.ccr-21-0793
  8. Biomarkers and factors in small cell lung cancer patients treated with immune checkpoint inhibitors: A meta-analysis.
    Li LL, Yu CF, Xie HT, Chen Z, et al · · 2023 · cited 11× · PMID 37161541 · DOI 10.1002/cam4.5800

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Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT03179436.

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