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NCT03123094

Single Rising Dose Trial of Spesolimab (BI 655130) for Healthy Japanese Male Subjects

Completed Phase 1 Results posted Last updated 6 March 2024
What this trial tests

Phase 1 trial testing Spesolimab in Healthy in 32 participants. Completed in 4 January 2018.

Timeline
16 May 2017
Primary endpoint
4 January 2018
4 January 2018

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingdouble
Primary purposetreatment
Enrollment32
Start date16 May 2017
Primary completion4 January 2018
Estimated completion4 January 2018
Sites1 location across South Korea

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 20 to 45, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Number of Subjects With Drug-related Adverse Events (AEs) Primary · From first drug administration until the end of trial examination, up to 151 days.

The primary endpoint is to assess safety and tolerability of spesolimab as the number \[N\] of subjects with drug-related AEs.

GroupValue95% CI
Spesolimab Low Dose Group (Intravenous)0
Spesolimab Medium Dose Group (Intravenous)0
Spesolimab High Dose Group (Intravenous)0
Spesolimab Low Dose Group (Subcutaneous)0
Placebo Matching to Spesolimab0
Area Under the Concentration-time Curve of Spesolimab in Plasma Over the Time Interval From 0 Extrapolated to Infinity (AUC0-∞) Secondary · Up to 3528 hours after administration of spesolimab.

AUC0-∞, Area under the concentration-time curve of spesolimab in plasma over the time interval from 0 extrapolated to infinity is presented. Pharmacokinetic samples were collected within 2 hours pre-dose and at 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 hours after dosing of dose groups with intravenous administration of spesolimab. Pharmacokinetic samples were collected within 2 hours pre-dose and at 0.5, 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 hours after dosing of dose grou

GroupValue95% CI
Spesolimab Low Dose Group (Intravenous)1890± 19.9
Spesolimab Medium Dose Group (Intravenous)3930± 18.4
Spesolimab High Dose Group (Intravenous)7060± 18.0
Spesolimab Low Dose Group (Subcutaneous)1390± 24.8
Maximum Measured Concentration of Spesolimab in Plasma (Cmax) Secondary · Up to 3528 hours after administration of spesolimab.

Cmax, maximum measured concentration of spesolimab in plasma is presented. Pharmacokinetic samples were collected within 2 hours pre-dose and at 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 hours after dosing of dose groups with intravenous administration of Up to 3528 hours after administration of spesolimab. Pharmacokinetic samples were collected within 2 hours pre-dose and at 0.5, 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 hours after dosing of dose groups with subcutaneous admin

GroupValue95% CI
Spesolimab Low Dose Group (Intravenous)99.7± 10.4
Spesolimab Medium Dose Group (Intravenous)193.0± 17.9
Spesolimab High Dose Group (Intravenous)400.0± 12.9
Spesolimab Low Dose Group (Subcutaneous)32.2± 21.8
Total Clearance of Spesolimab in Plasma After Intravenous Administration (CL) Secondary · Pharmacokinetic samples were collected within 2 hours (h) pre-dose and at 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 h after dosing of dose groups with intravenous administration of spesolimab.

CL, total clearance of spesolimab in plasma after intravenous administration is presented for intravenous dose groups.

GroupValue95% CI
Spesolimab Low Dose Group (Intravenous)0.159± 19.9
Spesolimab Medium Dose Group (Intravenous)0.153± 18.4
Spesolimab High Dose Group (Intravenous)0.170± 18.0
Volume of Distribution at Steady State After Intravenous Administration of Spesolimab (Vss) Secondary · Pharmacokinetic samples were collected within 2 hours (h) pre-dose and at 1.5, 2, 3, 4, 8, 12, 24, 48, 72, 96, 168, 336, 504, 672, 840, 1008, 1344, 1680, 2184, 2856 and 3528 h after dosing of dose groups with intravenous administration of spesolimab.

Vss, volume of distribution at steady state after intravenous administration of spesolimab is presented for intravenous dose groups.

GroupValue95% CI
Spesolimab Low Dose Group (Intravenous)6.19± 18.1
Spesolimab Medium Dose Group (Intravenous)6.97± 11.9
Spesolimab High Dose Group (Intravenous)6.60± 11.6

Adverse events — posted to ClinicalTrials.gov

Time frame: From first drug administration until the end of trial examination, up to 151 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Spesolimab Low Dose Group (Intravenous)
Serious: 0/6 (0%)
Deaths: 0/6
Spesolimab Medium Dose Group (Intravenous)
Serious: 0/6 (0%)
Deaths: 0/6
Spesolimab High Dose Group
Serious: 0/6 (0%)
Deaths: 0/6
Spesolimab Low Dose Group (Subcutaneous)
Serious: 0/6 (0%)
Deaths: 0/6
Placebo Matching to Spesolimab
Serious: 0/8 (0%)
Deaths: 0/8
Other adverse events (7 terms — click to expand)

ReactionSystemSpesolimab Low Dose Group …Spesolimab Medium Dose Gro…Spesolimab High Dose GroupSpesolimab Low Dose Group …Placebo Matching to Spesol…
VomitingGastrointestinal disorders
Chest discomfortGeneral disorders
GastroenteritisInfections and infestations
Upper respiratory tract infectionInfections and infestations
ContusionInjury, poisoning and procedural complications
Temporomandibular joint syndromeMusculoskeletal and connective tissue disorders
Rhinitis allergicRespiratory, thoracic and mediastinal disorders

Data from ClinicalTrials.gov NCT03123094 adverse events section.

Sponsor's own description

The primary objective of this trial is to investigate the safety and tolerability of spesolimab following administration of single rising intravenous doses and single subcutaneous dose in healthy Japanese male volunteers. Secondary objective is the exploration of the pharmacokinetics including dose proportionality of spesolimab in healthy Japanese male volunteers.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. Assessment of the Pharmacokinetics and Safety of Spesolimab, a Humanised Anti-interleukin-36 Receptor Monoclonal Antibody, in Healthy Non-Japanese and Japanese Subjects: Results from Phase I Clinical Studies.
    Joseph D, Thoma C, Haeufel T, Li X. · · 2022 · cited 9× · PMID 36451029 · DOI 10.1007/s40262-022-01176-5

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing