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NCT03023319

Bosutinib in Combination With Pemetrexed in Patients With Selected Metastatic Solid Tumors

Completed Phase 1 Last updated 14 June 2022
What this trial tests

Phase 1 trial testing Bosutinib in Carcinoma, Non-Small-Cell Lung in 6 participants. Completed in 10 May 2022.

Timeline
10 December 2019
Primary endpoint
10 May 2022
10 May 2022

Quick facts

Lead sponsorNagla Abdel Karim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment6
Start date10 December 2019
Primary completion10 May 2022
Estimated completion10 May 2022
Sites1 location across United States

Drugs / interventions tested

Conditions studied

Sponsor

Nagla Abdel Karim

Who can join

18 and older, any sex, with Carcinoma, Non-Small-Cell Lung or Mesothelioma. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

This study will determine the maximum-tolerated dose (MTD) for oral bosutinib when used in combination with pemetrexed. The MTD is the highest dose of bosutinib with pemetrexed that can be given without causing severe side effects. This study will also test the safety of this combination and see what effects (good or bad) it has on participants and their cancer.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. AXL receptor tyrosine kinase as a promising anti-cancer approach: functions, molecular mechanisms and clinical applications.
    Zhu C, Wei Y, Wei X. · · 2019 · cited 398× · PMID 31684958 · DOI 10.1186/s12943-019-1090-3
  2. Targeting Cancer Stem Cells in Triple-Negative Breast Cancer.
    Park SY, Park SY, Choi JH, Nam JS. · · 2019 · cited 135× · PMID 31324052 · DOI 10.3390/cancers11070965
  3. Src Family Kinases as Therapeutic Targets in Advanced Solid Tumors: What We Have Learned so Far.
    Martellucci S, Clementi L, Sabetta S, Mattei V, et al · · 2020 · cited 100× · PMID 32498343 · DOI 10.3390/cancers12061448
  4. Tyrosine Kinase Receptors in Oncology.
    Esteban-Villarrubia J, Soto-Castillo JJ, Pozas J, San Román-Gil M, et al · · 2020 · cited 72× · PMID 33198314 · DOI 10.3390/ijms21228529
  5. The Crosstalk between Src and Hippo/YAP Signaling Pathways in Non-Small Cell Lung Cancer (NSCLC).
    Hsu PC, Yang CT, Jablons DM, You L. · · 2020 · cited 64× · PMID 32466572 · DOI 10.3390/cancers12061361
  6. Emerging Treatments for Malignant Pleural Mesothelioma: Where Are We Heading?
    Cantini L, Hassan R, Sterman DH, Sterman DH, et al · · 2020 · cited 47× · PMID 32226777 · DOI 10.3389/fonc.2020.00343
  7. AXL signaling in cancer: from molecular insights to targeted therapies.
    Yadav M, Sharma A, Patne K, Tabasum S, et al · · 2025 · cited 42× · PMID 39924521 · DOI 10.1038/s41392-024-02121-7
  8. Role of the ABL tyrosine kinases in the epithelial-mesenchymal transition and the metastatic cascade.
    Luttman JH, Colemon A, Mayro B, Pendergast AM. · · 2021 · cited 26× · PMID 34022881 · DOI 10.1186/s12964-021-00739-6

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Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT03023319.

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