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NCT03004534

A Study to Evaluate Changes in Human Breast Cancer Tissue Following Short-Term Use of Darolutamide

Completed EARLY_PHASE1 Results posted Last updated 3 April 2020
What this trial tests

EARLY_PHASE1 trial testing darolutamide in Breast Cancer Female in 36 participants. Completed in 13 March 2019.

Timeline
5 September 2017
Primary endpoint
14 February 2019
13 March 2019

Quick facts

Lead sponsorTranslational Research in Oncology
PhaseEARLY_PHASE1
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment36
Start date5 September 2017
Primary completion14 February 2019
Estimated completion13 March 2019
Sites14 locations across Canada, United States, Germany

Drugs / interventions tested

Conditions studied

Sponsor

Translational Research in Oncology — full company profile →

Who can join

18 and older, female only, with Breast Cancer Female. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Identifying Molecular Alterations in Breast Cancer Tissue Tumor Samples Following Short-Term Preoperative Exposure to Darolutamide in Female Patients Wit Early Breast Cancer. Primary · 1 year, 6 months

Androgen Receptor (AR) was assessed on the collected samples.

Androgen Receptor - Up
GroupValue95% CI
Presurgical Molecular Assessment7
Androgen Receptor - Unchanged
GroupValue95% CI
Presurgical Molecular Assessment12
Androgen Receptor - Down
GroupValue95% CI
Presurgical Molecular Assessment15
Number of Participants With Treatment-related Adverse Events (TEAE) as Assessed by CTCAE v4.03 Secondary · 1 year, 6 months

The assessment of safety will be performed for all subjects who have taken at least one tablet of darolutamide (defined as the "safety population")

GroupValue95% CI
Presurgical Molecular Assessment26
Presurgical Molecular Assessment10

Adverse events — posted to ClinicalTrials.gov

Time frame: 1 year, 6 months.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Presurgical Molecular Assessment
Serious: 0/36 (0%)
Deaths: 0/36
Other adverse events (12 terms — click to expand)

ReactionSystemPresurgical Molecular Asse…
FatigueGeneral disorders
ConstipationGastrointestinal disorders
DiarrhoeaGastrointestinal disorders
NaseaGastrointestinal disorders
NasopharyngitisInfections and infestations
Upper Respiratory Tract InfectionInfections and infestations
Procedural PainInjury, poisoning and procedural complications
ALAT IncreaseInvestigations
ASAT IncreaseInvestigations
ArthralgiaMusculoskeletal and connective tissue disorders
DysuriaRenal and urinary disorders
Breast PainReproductive system and breast disorders

Data from ClinicalTrials.gov NCT03004534 adverse events section.

Sponsor's own description

The purpose of this study is to evaluate the effect of short-term treatment with darolutamide on breast cancer cells (i.e., how the treatment may change the genes or proteins in breast cancer cells) and to evaluate its safety and the way it is tolerated by subjects. The intent is to study these changes in order to have a better understanding of the potential use of darolutamide for women with EBC, know which patients are likely or unlikely to respond to this treatment, and determine how darolutamide may be combined with other anti-cancer drugs.

Publications & conference data

7 peer-reviewed publications reference this trial (live from Europe PMC):

  1. ARe we there yet? Understanding androgen receptor signaling in breast cancer.
    Michmerhuizen AR, Spratt DE, Pierce LJ, Speers CW. · · 2020 · cited 82× · PMID 33062889 · DOI 10.1038/s41523-020-00190-9
  2. The Divergent Function of Androgen Receptor in Breast Cancer; Analysis of Steroid Mediators and Tumor Intracrinology.
    Bleach R, McIlroy M. · · 2018 · cited 40× · PMID 30416486 · DOI 10.3389/fendo.2018.00594
  3. Androgen receptor in breast cancer: The "5W" questions.
    Ravaioli S, Maltoni R, Pasculli B, Parrella P, et al · · 2022 · cited 29× · PMID 36111296 · DOI 10.3389/fendo.2022.977331
  4. Revisiting Androgen Receptor Signaling in Breast Cancer.
    Dai C, Ellisen LW. · · 2023 · cited 26× · PMID 36972361 · DOI 10.1093/oncolo/oyad049
  5. Modulating the Activity of Androgen Receptor for Treating Breast Cancer.
    You CP, Tsoi H, Man EPS, Leung MH, et al · · 2022 · cited 18× · PMID 36499670 · DOI 10.3390/ijms232315342
  6. Treatments Targeting the Androgen Receptor and Its Splice Variants in Breast Cancer.
    Tien AH, Sadar MD. · · 2024 · cited 11× · PMID 38339092 · DOI 10.3390/ijms25031817
  7. Androgen and oestrogen receptor co-expression determines the efficacy of hormone receptor-mediated radiosensitisation in breast cancer.
    Michmerhuizen AR, Lerner LM, Ward C, Pesch AM, et al · · 2022 · cited 6× · PMID 35618789 · DOI 10.1038/s41416-022-01849-9

Verify or expand the search:

Other recruiting trials for Breast Cancer Female

Currently open trials in the same condition.

Other Translational Research in Oncology trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT03004534.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing