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NCT02992483

Phase I Study of MIK665, a Mcl-1 Inhibitor, in Patients With Refractory or Relapsed Lymphoma or Multiple Myeloma

Completed Phase 1 Last updated 3 August 2021
What this trial tests

Phase 1 trial testing MIK665 in Multiple Myeloma (MM), Lymphoma, Large B-Cell, Diffuse (DLBCL), Lymphoma in 31 participants. Completed in 7 June 2019.

Timeline
12 July 2017
Primary endpoint
7 June 2019
7 June 2019

Quick facts

Lead sponsorNovartis Pharmaceuticals
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment31
Start date12 July 2017
Primary completion7 June 2019
Estimated completion7 June 2019
Sites8 locations across France, Italy, Japan, Germany, Australia, United States, Spain

Drugs / interventions tested

Conditions studied

Sponsor

Novartis Pharmaceuticals — full company profile →

Who can join

18 and older, any sex, with Multiple Myeloma (MM), Lymphoma, Large B-Cell, Diffuse (DLBCL), Lymphoma. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

The purpose of this first in human study is to assess safety, tolerability, PK and preliminary clinical activity and to estimate the MTD(s)/RDE(s) of MIK665 (also referred as S64315) as single agent administered intravenously (i.v.) in adult patients with refractory or relapsed lymphoma or multiple myeloma.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Targeting apoptosis in cancer therapy.
    Carneiro BA, El-Deiry WS. · · 2020 · cited 1823× · PMID 32203277 · DOI 10.1038/s41571-020-0341-y
  2. Small molecules in targeted cancer therapy: advances, challenges, and future perspectives.
    Zhong L, Li Y, Xiong L, Wang W, et al · · 2021 · cited 1003× · PMID 34054126 · DOI 10.1038/s41392-021-00572-w
  3. Targeting BCL-2 regulated apoptosis in cancer.
    Campbell KJ, Tait SWG. · · 2018 · cited 352× · PMID 29769323 · DOI 10.1098/rsob.180002
  4. Apoptosis: A Comprehensive Overview of Signaling Pathways, Morphological Changes, and Physiological Significance and Therapeutic Implications.
    Mustafa M, Ahmad R, Tantry IQ, Ahmad W, et al · · 2024 · cited 264× · PMID 39594587 · DOI 10.3390/cells13221838
  5. Mitochondria-associated programmed cell death as a therapeutic target for age-related disease.
    Nguyen TT, Wei S, Nguyen TH, Jo Y, et al · · 2023 · cited 221× · PMID 37612409 · DOI 10.1038/s12276-023-01046-5
  6. Targeting MCL-1 in cancer: current status and perspectives.
    Wang H, Guo M, Wei H, Chen Y. · · 2021 · cited 210× · PMID 33883020 · DOI 10.1186/s13045-021-01079-1
  7. Targeting MCL-1 in hematologic malignancies: Rationale and progress.
    Wei AH, Roberts AW, Spencer A, Rosenberg AS, et al · · 2020 · cited 157× · PMID 32204955 · DOI 10.1016/j.blre.2020.100672
  8. Recent advances in targeted therapies in acute myeloid leukemia.
    Bhansali RS, Pratz KW, Lai C. · · 2023 · cited 151× · PMID 36966300 · DOI 10.1186/s13045-023-01424-6

Verify or expand the search:

Other trials of MIK665

Trials testing the same drug.

Other recruiting trials for Multiple Myeloma (MM), Lymphoma, Large B-Cell, Diffuse (DLBCL), Lymphoma

Currently open trials in the same condition.

Other Novartis Pharmaceuticals trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02992483.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing