Last reviewed · How we verify

NCT02841709

Efficacy and Safety of ACT-541468 in Elderly Subjects With Insomnia Disorder

Completed Phase 2 Results posted Last updated 24 April 2020
What this trial tests

Phase 2 trial testing ACT-541468 in Insomnia Disorder in 58 participants. Completed in 29 June 2017.

Timeline
28 November 2016
Primary endpoint
31 May 2017
29 June 2017

Quick facts

Lead sponsorIdorsia Pharmaceuticals Ltd.
PhasePhase 2
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingquadruple
Primary purposetreatment
Enrollment58
Start date28 November 2016
Primary completion31 May 2017
Estimated completion29 June 2017
Sites10 locations across United States, Germany

Drugs / interventions tested

Conditions studied

Sponsor

Idorsia Pharmaceuticals Ltd. — full company profile →

Who can join

65 and older, any sex, with Insomnia Disorder. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Change in Wake After Sleep Onset (WASO) From Baseline to Days 1 and 2 Primary · Baseline to Day 1 and Day 2 of each treatment period

WASO is the time in minutes spent awake after onset of persistent sleep until lights on as determined by polysomnography (PSG)

GroupValue95% CI
ACT-541468 5 mg-18.9± 4.44
ACT-541468 10 mg-32.0± 4.50
ACT-541468 25 mg-45.1± 4.47
ACT-541468 50 mg-61.4± 4.44
Placebo-13.6± 4.50
Change in Mean Latency to Persistent Sleep (LPS) From Baseline to Days 1 and 2 Secondary · Baseline to Day 1 and Day 2 of each treatment period

LPS is the duration of time in minutes from lights off to persistent sleep onset as determined by PSG

GroupValue95% CI
ACT-541468 5 mg-37.92± 48.76
ACT-541468 10 mg-44.61± 41.28
ACT-541468 25 mg-44.81± 41.56
ACT-541468 50 mg-44.88± 44.22
Placebo-33.88± 41.74

Adverse events — posted to ClinicalTrials.gov

Time frame: Start of screening until the end of the safety follow-up period.. Reporting threshold: 0%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Single-blind Placebo (Run-in Period)
Serious: 0/58 (0%)
Deaths: 0/58
Placebo
Serious: 0/54 (0%)
Deaths: 0/54
ACT-541468 5 mg
Serious: 0/56 (0%)
Deaths: 0/56
ACT-541468 10 mg
Serious: 0/54 (0%)
Deaths: 0/54
ACT-541468 25 mg
Serious: 0/55 (0%)
Deaths: 0/55
ACT-541468 50 mg
Serious: 0/56 (0%)
Deaths: 0/56
Other adverse events (58 terms — click to expand)

ReactionSystemSingle-blind Placebo (Run-…PlaceboACT-541468 5 mgACT-541468 10 mgACT-541468 25 mgACT-541468 50 mg
FatigueGeneral disorders
Gait disturbanceGeneral disorders
NasopharyngitisInfections and infestations
Back painMusculoskeletal and connective tissue disorders
DizzinessNervous system disorders
HeadacheNervous system disorders
Bundle branch block leftCardiac disorders
Supraventricular extrasystolesCardiac disorders
Ventricular extrasystolesCardiac disorders
Cerumen impactionEar and labyrinth disorders
PhotophobiaEye disorders
Abdominal discomfortGastrointestinal disorders
Abdominal pain upperGastrointestinal disorders
Defaecation urgencyGastrointestinal disorders
DiarrhoeaGastrointestinal disorders
Dry mouthGastrointestinal disorders
DyspepsiaGastrointestinal disorders
Frequent bowel movementsGastrointestinal disorders
Gastrooesophageal reflux diseaseGastrointestinal disorders
NauseaGastrointestinal disorders
VomitingGastrointestinal disorders
Feeling abnormalGeneral disorders
CystitisInfections and infestations
Upper respiratory tract infectionInfections and infestations
ContusionInjury, poisoning and procedural complications
FallInjury, poisoning and procedural complications
Alanine aminotransferase increasedInvestigations
Blood pressure increasedInvestigations
Blood pressure systolic increasedInvestigations
Blood thyroid stimulating hormone increasedInvestigations
Blood triglycerides increasedInvestigations
Gamma-glutamyltransferase increasedInvestigations
HypochloraemiaMetabolism and nutrition disorders
Muscle spasmsMusculoskeletal and connective tissue disorders
Pain in extremityMusculoskeletal and connective tissue disorders
Cerebellar ataxiaNervous system disorders
DysgeusiaNervous system disorders
HyporeflexiaNervous system disorders
MigraineNervous system disorders
SomnolenceNervous system disorders

Data from ClinicalTrials.gov NCT02841709 adverse events section.

Sponsor's own description

This study evaluates the dose response of ACT-541468 on the change of wake after sleep onset (WASO) assessed by polysomnography (PSG) on the first 2 days of each treatment period.

Publications & conference data

6 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Daridorexant, a new dual orexin receptor antagonist, in elderly subjects with insomnia disorder.
    Zammit G, Dauvilliers Y, Pain S, Sebök Kinter D, et al · · 2020 · cited 66× · PMID 32341187 · DOI 10.1212/wnl.0000000000009475
  2. Daridorexant: First Approval.
    Markham A. · · 2022 · cited 45× · PMID 35298826 · DOI 10.1007/s40265-022-01699-y
  3. Advances in Molecular Pathology of Obstructive Sleep Apnea.
    Zhang M, Lu Y, Sheng L, Han X, et al · · 2022 · cited 11× · PMID 36500515 · DOI 10.3390/molecules27238422
  4. Different doses of dual orexin receptor antagonists in primary insomnia: a Bayesian network analysis.
    Xue T, Wu X, Li J, Chen S, et al · · 2023 · cited 10× · PMID 37261282 · DOI 10.3389/fphar.2023.1175372
  5. Daridorexant, a Recently Approved Dual Orexin Receptor Antagonists (DORA) in Treatment of Insomnia.
    Sarathi Chakraborty D, Choudhury S, Lahiry S. · · 2023 · cited 8× · PMID 37425970 · DOI 10.1055/s-0043-1770805
  6. Daridorexant for the treatment of insomnia disorder: A systematic review and meta-analysis of randomized controlled trials.
    Jiang F, Li H, Chen Y, Lu H, et al · · 2023 · cited 6× · PMID 36800596 · DOI 10.1097/md.0000000000032754

Verify or expand the search:

Other trials of ACT-541468

Trials testing the same drug.

Other recruiting trials for Insomnia Disorder

Currently open trials in the same condition.

Other Idorsia Pharmaceuticals Ltd. trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02841709.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing