Last reviewed · How we verify

NCT02731742

Dose Evaluation of MK-1966 in Combination With SD-101 in Participants With Advanced Malignancies (MK-1966-001)

Terminated Phase 1 Results posted Last updated 4 February 2019
What this trial tests

Phase 1 trial testing MK-1966 in Neoplasms, Advanced in 14 participants. Terminated before completion.

Timeline
22 June 2016
Primary endpoint
8 January 2018
8 January 2018

Quick facts

Lead sponsorMerck Sharp & Dohme LLC
PhasePhase 1
StatusTerminated
Study typeINTERVENTIONAL
Allocationnon randomized
Designparallel
Maskingnone
Primary purposetreatment
Enrollment14
Start date22 June 2016
Primary completion8 January 2018
Estimated completion8 January 2018

Drugs / interventions tested

Conditions studied

Sponsor

Merck Sharp & Dohme LLC — full company profile →

Who can join

18 and older, any sex, with Neoplasms, Advanced. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Percentage of Participants With a Dose Limiting Toxicity (DLT) Primary · From time of first dose of study drug to the end of Cycle 1. Each cycle was 21 days. (Up to 21 days)

The occurrence of any of the following toxicities during Cycle 1 (Days 1-21), if assessed by the Investigator to be possibly, probably or definitely related to MK-1966 or SD-101, was considered a DLT: 1. Grade (Gr) 4 non-hematologic toxicity; 2. Gr 4 hematologic toxicity lasting \>7 days, except thrombocytopenia: \*Gr 4 thrombocytopenia of any duration; \*Gr 3 thrombocytopenia if associated with bleeding; 3. Gr 3 non-hematologic toxicity lasting \>3 days despite optimal supportive care; 4. Any Gr 3 or Gr 4 non-hematologic laboratory abnormality, if: medical intervention is required OR abnorma

GroupValue95% CI
MK-1966 70 mg+SD-101 1 mg0.00.0 – 33.1
MK-1966 70 mg+SD-101 4 mg0.00.0 – 33.1
MK-1966 210 mg+SD-101 4 mg20.05.1 – 44.8
MK-1966 700 mg+SD-101 4 mg0.00.0 – 41.5
Number of Participants With Adverse Events (AEs) Primary · From first dose of study drug through 90 days after last dose of study drug (Up to approximately 22 weeks)

An AE was defined as any untoward medical occurrence in a participant administered study drug and which does not necessarily have to have a causal relationship with this treatment. An AE could therefore be any unfavorable and unintended sign (including an abnormal laboratory finding, for example), symptom, or disease temporally associated with the use of study drug or protocol-specified procedure, whether or not considered related to the study drug or protocol-specified procedure. Any worsening (i.e., any clinically significant adverse change in frequency and/or intensity) of a pre-existing co

GroupValue95% CI
MK-1966 70 mg+SD-101 1 mg3
MK-1966 70 mg+SD-101 4 mg3
MK-1966 210 mg+SD-101 4 mg6
MK-1966 700 mg+SD-101 4 mg2
Number of Participants Discontinuing Study Drug Due to AEs Primary · From first dose of study drug up to last dose of study drug (Up to approximately 9 weeks)

The number of participants who discontinued study drug due to an AE is presented.

GroupValue95% CI
MK-1966 70 mg+SD-101 1 mg0
MK-1966 70 mg+SD-101 4 mg0
MK-1966 210 mg+SD-101 4 mg1
MK-1966 700 mg+SD-101 4 mg0

Adverse events — posted to ClinicalTrials.gov

Time frame: From first dose of study drug through 90 days after last dose of study drug (Up to approximately 22 weeks). Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

MK-1966 70 mg+SD-101 1 mg
Serious: 1/3 (33%)
Deaths: 1/3
MK-1966 70 mg+SD-101 4 mg
Serious: 1/3 (33%)
Deaths: 2/3
MK-1966 210 mg+SD-101 4 mg
Serious: 3/6 (50%)
Deaths: 5/6
MK-1966 700 mg+SD-101 4 mg
Serious: 1/2 (50%)
Deaths: 0/2

Serious adverse events (6 terms)

ReactionSystemMK-1966 70 mg+SD-101 1 mgMK-1966 70 mg+SD-101 4 mgMK-1966 210 mg+SD-101 4 mgMK-1966 700 mg+SD-101 4 mg
PyrexiaGeneral disorders
Skin infectionInfections and infestations
Urinary tract infectionInfections and infestations
HyponatraemiaMetabolism and nutrition disorders
Pleural effusionRespiratory, thoracic and mediastinal disorders
HypotensionVascular disorders
Other adverse events (81 terms — click to expand)

ReactionSystemMK-1966 70 mg+SD-101 1 mgMK-1966 70 mg+SD-101 4 mgMK-1966 210 mg+SD-101 4 mgMK-1966 700 mg+SD-101 4 mg
NauseaGastrointestinal disorders
FatigueGeneral disorders
StomatitisGastrointestinal disorders
VomitingGastrointestinal disorders
ChillsGeneral disorders
Injection site reactionGeneral disorders
Mucosal inflammationGeneral disorders
PyrexiaGeneral disorders
Candida infectionInfections and infestations
Tumour painNeoplasms benign, malignant and unspecified (incl cysts and polyps)
DizzinessNervous system disorders
CoughRespiratory, thoracic and mediastinal disorders
Oropharyngeal painRespiratory, thoracic and mediastinal disorders
RashSkin and subcutaneous tissue disorders
AnaemiaBlood and lymphatic system disorders
Lymph node painBlood and lymphatic system disorders
LymphadenopathyBlood and lymphatic system disorders
PalpitationsCardiac disorders
PericarditisCardiac disorders
HypothyroidismEndocrine disorders
Vision blurredEye disorders
ConstipationGastrointestinal disorders
Epigastric discomfortGastrointestinal disorders
Food poisoningGastrointestinal disorders
Oral painGastrointestinal disorders
AstheniaGeneral disorders
Chest discomfortGeneral disorders
Chest painGeneral disorders
Influenza like illnessGeneral disorders
Injection site erythemaGeneral disorders
Injection site haemorrhageGeneral disorders
Injection site painGeneral disorders
MalaiseGeneral disorders
PainGeneral disorders
CellulitisInfections and infestations
PneumoniaInfections and infestations
Rash pustularInfections and infestations
Upper respiratory tract infectionInfections and infestations
ExcoriationInjury, poisoning and procedural complications
Aspartate aminotransferase increasedInvestigations

Most-reported serious reactions: Pyrexia, Skin infection, Urinary tract infection, Hyponatraemia, Pleural effusion, Hypotension.

Data from ClinicalTrials.gov NCT02731742 adverse events section.

Sponsor's own description

This was a non-randomized, open-label study of MK-1966 used in combination with SD-101 in the treatment of advanced malignancies. The study included an initial Dose Evaluation phase (Part A) to determine the maximum tolerated dose (MTD)/maximum administered dose (MAD) by evaluating Dose Limiting Toxicities (DLTs) of four dose combinations of MK-1966 and SD-101. Following determination of the MTD/MAD, approximately 20 participants each were to be enrolled in two expansion cohorts (Parts B or C) to confirm/refine the MTD/MAD. The study was terminated by the Sponsor before enrollment into Part A concluded and before enrollment into Parts B and C began.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Re-Emergence of Dendritic Cell Vaccines for Cancer Treatment.
    Saxena M, Bhardwaj N. · · 2018 · cited 231× · PMID 29458962 · DOI 10.1016/j.trecan.2017.12.007
  2. Trial Watch: Toll-like receptor agonists in cancer immunotherapy.
    Smith M, García-Martínez E, Pitter MR, Fucikova J, et al · · 2018 · cited 171× · PMID 30524908 · DOI 10.1080/2162402x.2018.1526250
  3. Recent Advances in Oligonucleotide Therapeutics in Oncology.
    Xiong H, Veedu RN, Diermeier SD. · · 2021 · cited 132× · PMID 33804856 · DOI 10.3390/ijms22073295
  4. Turbocharging vaccines: emerging adjuvants for dendritic cell based therapeutic cancer vaccines.
    Saxena M, Bhardwaj N. · · 2017 · cited 50× · PMID 28732279 · DOI 10.1016/j.coi.2017.06.003
  5. Plasmacytoid dendritic cells at the forefront of anti-cancer immunity: rewiring strategies for tumor microenvironment remodeling.
    Monti M, Ferrari G, Gazzurelli L, Bugatti M, et al · · 2024 · cited 22× · PMID 39020402 · DOI 10.1186/s13046-024-03121-9
  6. Next-generation immunotherapy for pancreatic ductal adenocarcinoma: navigating pathways of immune resistance.
    Heumann T, Azad N. · · 2021 · cited 17× · PMID 34591243 · DOI 10.1007/s10555-021-09981-3
  7. Enhancement of Antitumor Vaccination by Targeting Dendritic Cell-Related IL-10.
    Llopiz D, Ruiz M, Silva L, Sarobe P. · · 2018 · cited 15× · PMID 30233565 · DOI 10.3389/fimmu.2018.01923
  8. Targeting pattern recognition receptors for cancer therapy: Mechanisms and strategies.
    Ouyang D, Chen R, Xie H, Yang X, et al · · 2025 · cited 1× · PMID 41311391 · DOI 10.1016/j.apsb.2025.09.007

Verify or expand the search:

Other Merck Sharp & Dohme LLC trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02731742.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing