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NCT02671461

Safety and Efficacy Study of a Protease Activated Receptor-4 Antagonist Being Tested to Reduce the Chances of Having Additional Strokes or "Mini Strokes"

Completed Phase 2 Results posted Last updated 14 December 2018
What this trial tests

Phase 2 trial testing BMS-986141 in Thrombosis in 16 participants. Completed in 31 March 2017.

Timeline
25 April 2016
Primary endpoint
31 March 2017
31 March 2017

Quick facts

Lead sponsorBristol-Myers Squibb
PhasePhase 2
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingquadruple
Primary purposetreatment
Enrollment16
Start date25 April 2016
Primary completion31 March 2017
Estimated completion31 March 2017
Sites33 locations across Japan, United States

Drugs / interventions tested

Conditions studied

Sponsor

Bristol-Myers Squibb — full company profile →

Who can join

18 and older, any sex, with Thrombosis. Patients with the condition only — healthy volunteers not accepted.

Adverse events — posted to ClinicalTrials.gov

Time frame: From first dose until 30 days following last dose (assessed up to March 2017, approximately 6 months). Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Placebo
Serious: 0/3 (0%)
Deaths: 0/3
BMS-986141 0.8 mg
Serious: 0/5 (0%)
Deaths: 0/5
BMS-986141 4.8 mg
Serious: 1/7 (14%)
Deaths: 0/7

Serious adverse events (1 terms)

ReactionSystemPlaceboBMS-986141 0.8 mgBMS-986141 4.8 mg
EncephalopathyNervous system disorders
Other adverse events (12 terms — click to expand)

ReactionSystemPlaceboBMS-986141 0.8 mgBMS-986141 4.8 mg
ConstipationGastrointestinal disorders
Muscle SpasmsMusculoskeletal and connective tissue disorders
Blood Potassium IncreasedInvestigations
Tinea PedisInfections and infestations
Vaginal DischargeReproductive system and breast disorders
Vulvovaginal PruritisReproductive system and breast disorders
SinusitisInfections and infestations
Viral Upper Respiratory Tract InfectionInfections and infestations
Micturation UrgencyRenal and urinary disorders
Oedema PeripheralGeneral disorders
HypokalaemiaMetabolism and nutrition disorders
CoughRespiratory, thoracic and mediastinal disorders

Most-reported serious reactions: Encephalopathy.

Data from ClinicalTrials.gov NCT02671461 adverse events section.

Sponsor's own description

The purpose of this study is to determine whether BMS-986141 is effective in reducing the recurrence of stroke in people who recently had a stroke, or a transient ischemic attack (known as a TIA or "mini stroke") and are receiving acetylsalicylic acid (also known as aspirin or ASA) to treat the stroke or TIA.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Protease-activated receptors (PARs): mechanisms of action and potential therapeutic modulators in PAR-driven inflammatory diseases.
    Heuberger DM, Schuepbach RA. · · 2019 · cited 274× · PMID 30976204 · DOI 10.1186/s12959-019-0194-8
  2. Platelets as Mediators of Neuroinflammation and Thrombosis.
    Rawish E, Nording H, Münte T, Langer HF. · · 2020 · cited 101× · PMID 33123127 · DOI 10.3389/fimmu.2020.548631
  3. Platelets as Modulators of Cerebral Ischemia/Reperfusion Injury.
    Stegner D, Klaus V, Nieswandt B. · · 2019 · cited 76× · PMID 31736950 · DOI 10.3389/fimmu.2019.02505
  4. Novel Antiplatelet Therapies for Atherothrombotic Diseases.
    Majithia A, Bhatt DL. · · 2019 · cited 53× · PMID 30760019 · DOI 10.1161/atvbaha.118.310955
  5. The domino effect triggered by the tethered ligand of the protease activated receptors.
    Han X, Nieman MT. · · 2020 · cited 34× · PMID 32853981 · DOI 10.1016/j.thromres.2020.08.004
  6. A function-blocking PAR4 antibody is markedly antithrombotic in the face of a hyperreactive PAR4 variant.
    French SL, Thalmann C, Bray PF, Macdonald LE, et al · · 2018 · cited 24× · PMID 29884748 · DOI 10.1182/bloodadvances.2017015552
  7. PAR4 (Protease-Activated Receptor 4): PARticularly Important 4 Antiplatelet Therapy.
    Han X, Nieman MT. · · 2018 · cited 24× · PMID 29367229 · DOI 10.1161/atvbaha.117.310550
  8. Using PAR4 Inhibition as an Anti-Thrombotic Approach: Why, How, and When?
    Li S, Tarlac V, Hamilton JR. · · 2019 · cited 19× · PMID 31717963 · DOI 10.3390/ijms20225629

Verify or expand the search:

Other trials of BMS-986141

Trials testing the same drug.

Other recruiting trials for Thrombosis

Currently open trials in the same condition.

Other Bristol-Myers Squibb trials

Trials by the same sponsor.

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Data sources for this page

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing