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NCT02475135

Relative Bioavailability and Food Effect for Darunavir/Cobicistat/Emtricitabine/Tenofovir Alafenamide Fixed Dose Combination

Completed Phase 1 Last updated 17 October 2017
What this trial tests

Phase 1 trial testing Darunavir/Cobicistat/Emtricitabine/Tenofovir alafenamide FDC in Healthy in 72 participants. Completed in 14 August 2015.

Timeline
1 June 2015
Primary endpoint
14 August 2015
14 August 2015

Quick facts

Lead sponsorJanssen Sciences Ireland UC
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingnone
Primary purposetreatment
Enrollment72
Start date1 June 2015
Primary completion14 August 2015
Estimated completion14 August 2015
Sites1 location across Belgium

Drugs / interventions tested

Conditions studied

Sponsor

Janssen Sciences Ireland UC — full company profile →

Who can join

Adults 18 to 55, any sex, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

The purpose of this study is to evaluate the pharmacokinetics and relative bioavailability of Emtricitabine (FTC) and Tenofovir alafenamide (TAF) when administered as a fixed-dose combination (FDC) with darunavir (DRV) and cobicistat (COBI) (darunavir/cobicistat/emtricitabine/tenofovir alafenamide (D/C/F/TAF) relative to administration as an FDC with Elvitegravir (EVG) and COBI (Elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide), under fed conditions in healthy subjects (Panel 1); evaluate the single-dose pharmacokinetics and relative bioavailability of DRV, COBI, FTC and TAF when administered as an FDC (D/C/F/TAF) or as separate agents (D+C+FTC/TAF), under fed conditions in healthy subjects (Panel 2) and to evaluate the impact of food (fasting or high-fat breakfast) on the single-dose pharmacokinetics of DRV, COBI, FTC, and TAF when administered as an FDC (D/C/F/TAF) in healthy subjects (Panel 3).

Publications & conference data

3 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Darunavir-cobicistat-emtricitabine-tenofovir alafenamide: safety and efficacy of a protease inhibitor in the modern era.
    Squillace N, Bozzi G, Colella E, Gori A, et al · · 2018 · cited 11× · PMID 30464395 · DOI 10.2147/dddt.s147493
  2. Bioequivalence of the Once-Daily Single-Tablet Regimen of Darunavir, Cobicistat, Emtricitabine, and Tenofovir Alafenamide Compared to Combined Intake of the Separate Agents and the Effect of Food on Bioavailability.
    Crauwels HM, Baugh B, Van Landuyt E, Vanveggel S, et al · · 2019 · cited 5× · PMID 30412360 · DOI 10.1002/cpdd.628
  3. International Congress of Drug Therapy in HIV Infection 23-26 October 2016, Glasgow, UK.
    · 2016 · cited 3× · PMID 27780519 · DOI 10.7448/ias.19.8.21487

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Other recruiting trials for Healthy

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Data sources for this page

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing