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NCT02350868

Dose-Seeking Study of MPT0E028 in Subjects With Advanced Solid Malignancies Without Standard Treatment

Completed Phase 1 Last updated 11 April 2019
What this trial tests

Phase 1 trial testing MPT0E028 in Advanced Solid Malignancies in 23 participants. Completed in 19 January 2019.

Timeline
24 April 2015
Primary endpoint
19 January 2019
19 January 2019

Quick facts

Lead sponsorTaipei Medical University
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment23
Start date24 April 2015
Primary completion19 January 2019
Estimated completion19 January 2019
Sites2 locations across Taiwan

Drugs / interventions tested

Conditions studied

Sponsor

Taipei Medical University

Who can join

20 and older, any sex, with Advanced Solid Malignancies. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

The Dose Escalation Phase will determine the MTD of MPT0E028 and evaluate its safety and tolerability, PK, PD, and preliminary clinical effects; the subsequent Dose Confirmation Phase will be a cohort expansion at or below the MTD (i.e., an RP2D) of MPT0E028.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. The roles of histone modifications in tumorigenesis and associated inhibitors in cancer therapy.
    Yang Y, Zhang M, Wang Y. · · 2022 · cited 96× · PMID 39036551 · DOI 10.1016/j.jncc.2022.09.002
  2. Immunoepigenetics Combination Therapies: An Overview of the Role of HDACs in Cancer Immunotherapy.
    Banik D, Moufarrij S, Villagra A. · · 2019 · cited 96× · PMID 31067680 · DOI 10.3390/ijms20092241
  3. Targeting the epigenome in in-stent restenosis: from mechanisms to therapy.
    Yang X, Yang Y, Guo J, Meng Y, et al · · 2021 · cited 47× · PMID 33664994 · DOI 10.1016/j.omtn.2021.01.024
  4. Pharmacological targeting of the cancer epigenome.
    Mabe NW, Perry JA, Malone CF, Stegmaier K. · · 2024 · cited 36× · PMID 38937652 · DOI 10.1038/s43018-024-00777-2
  5. Histones and heart failure in diabetes.
    Yerra VG, Advani A. · · 2018 · cited 25× · PMID 29934664 · DOI 10.1007/s00018-018-2857-1
  6. Combination treatment strategy for pancreatic cancer involving the novel HDAC inhibitor MPT0E028 with a MEK inhibitor beyond K-Ras status.
    Chao MW, Chang LH, Tu HJ, Chang CD, et al · · 2019 · cited 24× · PMID 31142371 · DOI 10.1186/s13148-019-0681-6
  7. Processes and therapeutic perspectives of acylation modifications of lysine and cysteine in tumors.
    Jiang J, Chen J, Huang S, Tian Y, et al · · 2026 · PMID 41630001 · DOI 10.1186/s12964-026-02707-4
  8. Next-Generation HDAC Inhibitors: Advancing Zinc-Binding Group Design for Enhanced Cancer Therapy.
    Hawash M. · · 2025 · PMID 41440016 · DOI 10.3390/cells14241997

Verify or expand the search:

Other recruiting trials for Advanced Solid Malignancies

Currently open trials in the same condition.

Other Taipei Medical University trials

Trials by the same sponsor.

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Data sources for this page

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