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NCT02157636

A Phase 1 Study Evaluating CPI-0610 in Patients With Previously Treated Multiple Myeloma

Completed Phase 1 Last updated 18 April 2024
What this trial tests

Phase 1 trial testing CPI-0610 in Multiple Myeloma in 30 participants. Completed in 8 November 2016.

Timeline
15 July 2014
Primary endpoint
8 November 2016
8 November 2016

Quick facts

Lead sponsorConstellation Pharmaceuticals
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationna
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment30
Start date15 July 2014
Primary completion8 November 2016
Estimated completion8 November 2016

Drugs / interventions tested

Conditions studied

Sponsor

Constellation Pharmaceuticals — full company profile →

Who can join

18 and older, any sex, with Multiple Myeloma. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

Open-label, sequential dose escalation and expansion study of CPI-0610 in patients with previously treated multiple myeloma. CPI-0610 is a small molecule inhibitor of bromodomain and extra-terminal (BET) proteins.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Targeting epigenetic regulators for cancer therapy: mechanisms and advances in clinical trials.
    Cheng Y, He C, Wang M, Ma X, et al · · 2019 · cited 760× · PMID 31871779 · DOI 10.1038/s41392-019-0095-0
  2. Tumor biomarkers for diagnosis, prognosis and targeted therapy.
    Zhou Y, Tao L, Qiu J, Xu J, et al · · 2024 · cited 379× · PMID 38763973 · DOI 10.1038/s41392-024-01823-2
  3. Therapeutic targeting of "undruggable" MYC.
    Llombart V, Mansour MR. · · 2022 · cited 349× · PMID 34942444 · DOI 10.1016/j.ebiom.2021.103756
  4. Epigenetics in cancer stem cells.
    Toh TB, Lim JJ, Chow EK. · · 2017 · cited 286× · PMID 28148257 · DOI 10.1186/s12943-017-0596-9
  5. Achieving clinical success with BET inhibitors as anti-cancer agents.
    Shorstova T, Foulkes WD, Witcher M. · · 2021 · cited 272× · PMID 33723398 · DOI 10.1038/s41416-021-01321-0
  6. Epigenetics and Cancer Stem Cells: Unleashing, Hijacking, and Restricting Cellular Plasticity.
    Wainwright EN, Scaffidi P. · · 2017 · cited 250× · PMID 28718414 · DOI 10.1016/j.trecan.2017.04.004
  7. Drug Discovery Targeting Bromodomain-Containing Protein 4.
    Liu Z, Wang P, Chen H, Wold EA, et al · · 2017 · cited 234× · PMID 28195723 · DOI 10.1021/acs.jmedchem.6b01761
  8. Bromodomain and extra-terminal motif inhibitors: a review of preclinical and clinical advances in cancer therapy.
    Alqahtani A, Choucair K, Ashraf M, Hammouda DM, et al · · 2019 · cited 198× · PMID 30906568 · DOI 10.4155/fsoa-2018-0115

Verify or expand the search:

Other trials of CPI-0610

Trials testing the same drug.

Other recruiting trials for Multiple Myeloma

Currently open trials in the same condition.

Other Constellation Pharmaceuticals trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02157636.

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