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NCT02044419

A Comparative Bioavailability Study of Lomitapide 20 mg Intact vs Sprinkled

Completed Phase 1 Results posted Last updated 13 February 2018
What this trial tests

Phase 1 trial testing lomitapide in Healthy in 32 participants. Completed in 23 December 2013.

Timeline
30 October 2013
Primary endpoint
23 December 2013
23 December 2013

Quick facts

Lead sponsorAegerion Pharmaceuticals, Inc.
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designcrossover
Maskingnone
Primary purposeother
Enrollment32
Start date30 October 2013
Primary completion23 December 2013
Estimated completion23 December 2013
Sites1 location across United Kingdom

Drugs / interventions tested

Conditions studied

Sponsor

Aegerion Pharmaceuticals, Inc. — full company profile →

Who can join

Adults 18 to 40, any sex, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

AUC0-t Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Area under the concentration-time curve from hour 0 to the last measurable concentration of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)38.3± 15.2
Lomitapide Sprinkled in Mashed Banana (Treatment B)40.2± 13.4
Intact Capsule of 20 mg Lomitapide (Treatment C)43.6± 17.7
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)70.4± 20.2
Lomitapide Sprinkled in Mashed Banana (Treatment B)72.9± 23.1
Intact Capsule of 20 mg Lomitapide (Treatment C)75.2± 22.8
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)443± 308
Lomitapide Sprinkled in Mashed Banana (Treatment B)450± 292
Intact Capsule of 20 mg Lomitapide (Treatment C)460± 325
Cmax Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Maximum observed concentration of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)0.986± 0.536
Lomitapide Sprinkled in Mashed Banana (Treatment B)1.03± 0.463
Intact Capsule of 20 mg Lomitapide (Treatment C)1.13± 0.591
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)2.52± 0.748
Lomitapide Sprinkled in Mashed Banana (Treatment B)2.65± 0.813
Intact Capsule of 20 mg Lomitapide (Treatment C)2.74± 0.796
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)30.2± 15.6
Lomitapide Sprinkled in Mashed Banana (Treatment B)31.0± 13.3
Intact Capsule of 20 mg Lomitapide (Treatment C)28.6± 13.7
Tmax Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Time to reach maximum plasma concentration of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)4.001.00 – 12.0
Lomitapide Sprinkled in Mashed Banana (Treatment B)5.001.00 – 12.0
Intact Capsule of 20 mg Lomitapide (Treatment C)5.002.00 – 24.0
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)5.002.00 – 8.00
Lomitapide Sprinkled in Mashed Banana (Treatment B)5.002.00 – 6.00
Intact Capsule of 20 mg Lomitapide (Treatment C)5.003.00 – 8.00
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)2.031.00 – 4.00
Lomitapide Sprinkled in Mashed Banana (Treatment B)3.001.00 – 5.00
Intact Capsule of 20 mg Lomitapide (Treatment C)3.001.00 – 4.00
t1/2 Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Terminal elimination half-life of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)52.4± 13.3
Lomitapide Sprinkled in Mashed Banana (Treatment B)47.7± 12.2
Intact Capsule of 20 mg Lomitapide (Treatment C)48.8± 10.7
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)38.7± 7.56
Lomitapide Sprinkled in Mashed Banana (Treatment B)37.0± 6.78
Intact Capsule of 20 mg Lomitapide (Treatment C)39.1± 6.32
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)46.0± 13.1
Lomitapide Sprinkled in Mashed Banana (Treatment B)45.7± 11.5
Intact Capsule of 20 mg Lomitapide (Treatment C)44.0± 11.6
AUC0-∞ Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Area under the plasma concentration vs time curve from zero to infinity of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)42.5± 17.7
Lomitapide Sprinkled in Mashed Banana (Treatment B)43.8± 15.3
Intact Capsule of 20 mg Lomitapide (Treatment C)47.7± 20.6
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)72.8± 20.8
Lomitapide Sprinkled in Mashed Banana (Treatment B)75.2± 23.7
Intact Capsule of 20 mg Lomitapide (Treatment C)77.8± 23.9
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)457± 317
Lomitapide Sprinkled in Mashed Banana (Treatment B)464± 300
Intact Capsule of 20 mg Lomitapide (Treatment C)474± 333
λz Primary · predose and 1, 2, 3, 4, 5, 6, 8, 10, 12, 18, 24, 48, 72, 96, 120, 144, and 168 hours post-dose

Elimination rate constant estimated from individual linear regression of the terminal part of the log concentration vs time curve of lomitapide and its metabolites (M1\& M3).

Lomitapide
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)0.0140± 0.00341
Lomitapide Sprinkled in Mashed Banana (Treatment B)0.0153± 0.00343
Intact Capsule of 20 mg Lomitapide (Treatment C)0.0149± 0.00320
M1
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)0.0185± 0.00344
Lomitapide Sprinkled in Mashed Banana (Treatment B)0.0195± 0.00457
Intact Capsule of 20 mg Lomitapide (Treatment C)0.0182± 0.00309
M3
GroupValue95% CI
Lomitapide Sprinkled in Applesauce (Treatment A)0.0161± 0.00408
Lomitapide Sprinkled in Mashed Banana (Treatment B)0.0162± 0.00428
Intact Capsule of 20 mg Lomitapide (Treatment C)0.0167± 0.00405

Adverse events — posted to ClinicalTrials.gov

Reporting threshold: 0%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Lomitapide Sprinkled in Applesauce (Treatment A)
Serious: 0/30 (0%)
Deaths: 0/30
Lomitapide Sprinkled in Mashed Banana (Treatment B)
Serious: 0/31 (0%)
Deaths: 0/31
Intact Capsule of 20 mg Lomitapide (Treatment C)
Serious: 0/31 (0%)
Deaths: 0/31
Other adverse events (16 terms — click to expand)

ReactionSystemLomitapide Sprinkled in Ap…Lomitapide Sprinkled in Ma…Intact Capsule of 20 mg Lo…
Abdominal PainGastrointestinal disorders
HeadacheNervous system disorders
PolyuriaRenal and urinary disorders
PresyncopeVascular disorders
ConstipationGastrointestinal disorders
VomitingGastrointestinal disorders
Dry mouthGastrointestinal disorders
GlossodyniaGastrointestinal disorders
Oral painGastrointestinal disorders
NasopharyngitisRespiratory, thoracic and mediastinal disorders
Conjunctival haemorrhageEye disorders
Eye swellingEye disorders
Catheter site painGeneral disorders
Herpes simplexInfections and infestations
EpistaxisVascular disorders
RashSkin and subcutaneous tissue disorders

Data from ClinicalTrials.gov NCT02044419 adverse events section.

Sponsor's own description

To compare the relative bioavailability of lomitapide when administered by sprinkling the contents of a 20 mg capsule of lomitapide in applesauce or in mashed banana to a single oral intact capsule dose of 20 mg lomitapide in healthy subjects.

Publications & conference data

No peer-reviewed publications indexed yet for this trial. Completed trials usually publish results within 12-18 months.

Verify or expand the search:

Other trials of lomitapide

Trials testing the same drug.

Other recruiting trials for Healthy

Currently open trials in the same condition.

Other Aegerion Pharmaceuticals, Inc. trials

Trials by the same sponsor.

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Data sources for this page

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing