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NCT02039063

A Phase 1/2 Study of Repeated Intravenous E6011 Administration in Japanese Subjects With Crohn's Disease

Completed Phase 1, PHASE2 Results posted Last updated 30 January 2023
What this trial tests

Phase 1, PHASE2 trial testing E6011 2 mg/kg in Crohn's Disease in 28 participants. Completed in 27 November 2017.

Timeline
5 April 2014
Primary endpoint
6 January 2017
27 November 2017

Quick facts

Lead sponsorEA Pharma Co., Ltd.
PhasePhase 1, PHASE2
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designparallel
Primary purposetreatment
Enrollment28
Start date5 April 2014
Primary completion6 January 2017
Estimated completion27 November 2017
Sites17 locations across Japan

Drugs / interventions tested

Conditions studied

Sponsor

EA Pharma Co., Ltd. — full company profile →

Who can join

Adults 20 to 64, any sex, with Crohn's Disease. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Number of Participants With Treatment-emergent Adverse Events (TEAEs) and Serious Adverse Events (SAEs) Primary · Baseline up to Week 62 (70 days after last dose of study drug)

TEAEs was defined as adverse event (AEs) that emerged during the treatment, having been absent at pretreatment (Baseline) or re-emerged during treatment, having been present at pretreatment (Baseline) but stopped before treatment, or worsened in severity during treatment relative to the pretreatment state, when the AE was continuous. An AE was defined as any untoward medical occurrence in a participants or clinical study participant temporally associated with the use of study treatment, whether or not considered related to the study treatment. A SAE was defined as any untoward medical occurren

TEAE
GroupValue95% CI
Cohort 1: E6011 2 mg/kg6
Cohort 2: E6011 5 mg/kg6
Cohort 3: E6011 10 mg/kg7
Cohort 4: E6011 15 mg/kg3
SAE
GroupValue95% CI
Cohort 1: E6011 2 mg/kg1
Cohort 2: E6011 5 mg/kg1
Cohort 3: E6011 10 mg/kg5
Cohort 4: E6011 15 mg/kg0
Number of Participants With Clinically Significant Change in Laboratory Parameters Primary · Baseline up to Week 52

Clinical laboratory parameters included biochemistry, hematology, urinalysis and other screening test. Number of participants with clinically significant abnormalities in laboratory parameters which were deemed clinically significant by the investigator were reported.

GroupValue95% CI
Cohort 1: E6011 2 mg/kg0
Cohort 2: E6011 5 mg/kg0
Cohort 3: E6011 10 mg/kg0
Cohort 4: E6011 15 mg/kg0
Number of Participants With Clinically Significant Change in Vital Sign Measurements Primary · Baseline up to Week 52

Vital sign measurements included blood pressure (systolic and diastolic blood pressure) and pulse rate. Number of participants with clinically significant change in vital signs measurements which were deemed clinically significant by the investigator were reported.

GroupValue95% CI
Cohort 1: E6011 2 mg/kg0
Cohort 2: E6011 5 mg/kg0
Cohort 3: E6011 10 mg/kg0
Cohort 4: E6011 15 mg/kg0
Number of Participants With Treatment-emergent Clinically Significant Abnormal Electrocardiogram (ECG) Findings Primary · Baseline up to Week 52

Number of participants with treatment-emergent clinically significant abnormal ECG findings which were deemed clinically significant by the investigator were reported.

GroupValue95% CI
Cohort 1: E6011 2 mg/kg0
Cohort 2: E6011 5 mg/kg0
Cohort 3: E6011 10 mg/kg0
Cohort 4: E6011 15 mg/kg0
Number of Participants With Abnormal Chest X-ray Findings Primary · Baseline up to Week 52

Number of participants with abnormal chest X-ray findings were reported.

GroupValue95% CI
Cohort 1: E6011 2 mg/kg0
Cohort 2: E6011 5 mg/kg0
Cohort 3: E6011 10 mg/kg0
Cohort 4: E6011 15 mg/kg0
Number of Participants With Neurological Findings Primary · Baseline up to Week 52

Number of participants with neurological findings were reported.

GroupValue95% CI
Cohort 1: E6011 2 mg/kg0
Cohort 2: E6011 5 mg/kg0
Cohort 3: E6011 10 mg/kg0
Cohort 4: E6011 15 mg/kg0
Mean Trough Serum Concentration of E6011 at Week 12 and 52 Secondary · Week 12: Pre-dose; Week 52: Pre-dose
Week 12
GroupValue95% CI
Cohort 1: E6011 2 mg/kg3.40± 3.74
Cohort 2: E6011 5 mg/kg26.1± 10.4
Cohort 3: E6011 10 mg/kg96.8± 60.3
Cohort 4: E6011 15 mg/kg146± 91.9
Week 52
GroupValue95% CI
Cohort 1: E6011 2 mg/kg10.8± NA
Cohort 2: E6011 5 mg/kg17.3± 2.90
Cohort 3: E6011 10 mg/kg105± 9.69
Cohort 4: E6011 15 mg/kg93.9± 46.8
Number of Participants With Serum Anti-E6011 Antibody at Week 12 and 52 Secondary · At Week 12 and Week 52

Number of participants with serum anti-E6011 antibody were reported.

Week 12
GroupValue95% CI
Cohort 1: E6011 2 mg/kg4
Cohort 2: E6011 5 mg/kg3
Cohort 3: E6011 10 mg/kg2
Cohort 4: E6011 15 mg/kg1
Week 52
GroupValue95% CI
Cohort 1: E6011 2 mg/kg4
Cohort 2: E6011 5 mg/kg3
Cohort 3: E6011 10 mg/kg2
Cohort 4: E6011 15 mg/kg1

Adverse events — posted to ClinicalTrials.gov

Time frame: Baseline up to Week 62 (70 days after last dose of study drug). Reporting threshold: 0%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Cohort 1: E6011 2 mg/kg
Serious: 1/6 (17%)
Deaths: 0/6
Cohort 2: E6011 5 mg/kg
Serious: 1/8 (13%)
Deaths: 0/8
Cohort 3: E6011 10 mg/kg
Serious: 5/7 (71%)
Deaths: 0/7
Cohort 4: E6011 15 mg/kg
Serious: 0/7 (0%)
Deaths: 0/7

Serious adverse events (3 terms)

ReactionSystemCohort 1: E6011 2 mg/kgCohort 2: E6011 5 mg/kgCohort 3: E6011 10 mg/kgCohort 4: E6011 15 mg/kg
Crohn's diseaseGastrointestinal disorders
AnaemiaBlood and lymphatic system disorders
Miscarriage of partnerSocial circumstances
Other adverse events (41 terms — click to expand)

ReactionSystemCohort 1: E6011 2 mg/kgCohort 2: E6011 5 mg/kgCohort 3: E6011 10 mg/kgCohort 4: E6011 15 mg/kg
NasopharyngitisInfections and infestations
PyrexiaGeneral disorders
Device related infectionInfections and infestations
HeadacheNervous system disorders
Sudden hearing lossEar and labyrinth disorders
AsthenopiaEye disorders
Abdominal distensionGastrointestinal disorders
Abdominal pain upperGastrointestinal disorders
Aphthous ulcerGastrointestinal disorders
CheilitisGastrointestinal disorders
NauseaGastrointestinal disorders
StomatitisGastrointestinal disorders
VomitingGastrointestinal disorders
MalaiseGeneral disorders
CholelithiasisHepatobiliary disorders
Hepatic steatosisHepatobiliary disorders
Anal abscessInfections and infestations
Enterocolitis infectiousInfections and infestations
GingivitisInfections and infestations
InfluenzaInfections and infestations
ParonychiaInfections and infestations
PharyngitisInfections and infestations
TonsillitisInfections and infestations
Infusion related reactionInjury, poisoning and procedural complications
CD4 lymphocytes decreasedInvestigations
ArthralgiaMusculoskeletal and connective tissue disorders
ArthritisMusculoskeletal and connective tissue disorders
Back painMusculoskeletal and connective tissue disorders
BursitisMusculoskeletal and connective tissue disorders
Musculoskeletal painMusculoskeletal and connective tissue disorders
MyalgiaMusculoskeletal and connective tissue disorders
Neck painMusculoskeletal and connective tissue disorders
Upper respiratory tract inflammationRespiratory, thoracic and mediastinal disorders
Dry skinSkin and subcutaneous tissue disorders
EczemaSkin and subcutaneous tissue disorders
Erythema nodosumSkin and subcutaneous tissue disorders
Seborrhoeic dermatitisSkin and subcutaneous tissue disorders
UrticariaSkin and subcutaneous tissue disorders
Hot flushVascular disorders
HyperaemiaVascular disorders

Most-reported serious reactions: Crohn's disease, Anaemia, Miscarriage of partner.

Data from ClinicalTrials.gov NCT02039063 adverse events section.

Sponsor's own description

This study is a multicenter, open-label, uncontrolled, multiple ascending dose (MAD) study to evaluate mainly the safety and tolerability of 12-week repeated intravenous administration of E6011. A total of 24 subjects will enroll into four cohorts. Six subjects per cohort will receive repeated intravenous administration of E6011.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. Phase 1 study on the safety and efficacy of E6011, antifractalkine antibody, in patients with Crohn's disease.
    Matsuoka K, Naganuma M, Hibi T, Tsubouchi H, et al · · 2021 · cited 16× · PMID 33599356 · DOI 10.1111/jgh.15463

Verify or expand the search:

Other recruiting trials for Crohn's Disease

Currently open trials in the same condition.

Other EA Pharma Co., Ltd. trials

Trials by the same sponsor.

Verify against primary sources

Data sources for this page

Drug Landscape aggregates and links these public records for informational use only. Always verify against the primary source before clinical or regulatory decisions. Canonical URL: https://druglandscape.com/trial/NCT02039063.

Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing