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NCT01608087

Pharmacokinetics and Safety Study of BI 695502 in Healthy Subjects

Completed Phase 1 Results posted Last updated 8 November 2019
What this trial tests

Phase 1 trial testing BI 695502 in Healthy in 91 participants. Completed in 1 November 2012.

Timeline
1 May 2012
Primary endpoint
1 November 2012
1 November 2012

Quick facts

Lead sponsorBoehringer Ingelheim
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingsingle
Primary purposetreatment
Enrollment91
Start date1 May 2012
Primary completion1 November 2012
Estimated completion1 November 2012
Sites2 locations across New Zealand

Drugs / interventions tested

Conditions studied

Sponsor

Boehringer Ingelheim — full company profile →

Who can join

Adults 21 to 50, male only, with Healthy. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Area Under the Concentration-time Curve of the Analyte in Plasma Over the Time Interval From 0 Extrapolated to Infinity (AUC0-∞). Primary · Pharmacokinetic samples were collected predose, just before the end of the infusion, 2, 4, and 8 hours after the start of the infusion

Area under the concentration-time curve of the analyte in plasma over the time interval from 0 extrapolated to infinity (AUC0-∞) is presented as adjusted geometric mean (gMean) and geometric coefficient of variation (%) (gCV%). Adjustment were made for treatment effect and weight.

GroupValue95% CI
BI 695502 (T)7013.010± 19.52
United States (US)-Licensed Avastin® (R1)7261.119± 15.57
European Union (EU)-Approved Avastin® (R2)7649.491± 18.29
Area Under the Concentration-time Curve of the Analyte in Plasma Over the Time Interval From 0 to the Time of the Last Quantifiable Data Point (AUC0-tz) Secondary · Pharmacokinetic samples were collected predose, just before the end of the infusion, 2, 4, and 8 hours after the start of the infusion

Area under the concentration-time curve of the analyte in plasma over the time interval from 0 to the time of the last quantifiable data point is presented as adjusted geometric mean (gMean) and geometric coefficient of variation (%) (gCV%). Adjustment was made for treatment effect and weight.

GroupValue95% CI
BI 695502 (T)6570.047± 20.68
United States (US)-Licensed Avastin® (R1)6639.315± 18.46
European Union (EU)-Approved Avastin® (R2)7167.313± 19.72
Maximum Measured Concentration of the Analyte in Plasma (Cmax) Secondary · Pharmacokinetic samples were collected predose, just before the end of the infusion, 2, 4, and 8 hours after the start of the infusion.

Maximum measured concentration of the analyte in plasma (Cmax) is presented as adjusted geometric mean (gMean) and geometric coefficient of variation (%) (gCV%). Adjustment was made for treatment effect and weight.

GroupValue95% CI
BI 695502 (T)23.783± 16.11
United States (US)-Licensed Avastin® (R1)23.425± 25.15
European Union (EU)-Approved Avastin® (R2)25.505± 15.18

Adverse events — posted to ClinicalTrials.gov

Time frame: From first drug administration to end of trial; up to 99 days.. Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

BI 695502 (T)
Serious: 0/30 (0%)
Deaths: 0/30
United States (US)-Licensed Avastin® (R1)
Serious: 0/30 (0%)
Deaths: 0/30
European Union (EU)-Approved Avastin® (R2)
Serious: 0/31 (0%)
Deaths: 0/31
Other adverse events (18 terms — click to expand)

ReactionSystemBI 695502 (T)United States (US)-License…European Union (EU)-Approv…
Upper respiratory tract infectionInfections and infestations
HeadacheNervous system disorders
Respiratory tract infectionInfections and infestations
DizzinessNervous system disorders
Back painMusculoskeletal and connective tissue disorders
Thermal burnInjury, poisoning and procedural complications
LacerationInjury, poisoning and procedural complications
GastroenteritisInfections and infestations
RhinitisInfections and infestations
Orthostatic hypotensionVascular disorders
ToothacheGastrointestinal disorders
DiarrhoeaGastrointestinal disorders
Gastrooesophageal reflux diseaseGastrointestinal disorders
NauseaGastrointestinal disorders
Musculoskeletal painMusculoskeletal and connective tissue disorders
MyalgiaMusculoskeletal and connective tissue disorders
ContusionInjury, poisoning and procedural complications
Muscle strainInjury, poisoning and procedural complications

Data from ClinicalTrials.gov NCT01608087 adverse events section.

Sponsor's own description

This trial will investigate the pharmacokinetics and safety of BI 695502 and to establish pharmacokinetic biosimilarity of BI 695502 compared to bevacizumab.

Publications & conference data

3 peer-reviewed publications reference this trial (live from Europe PMC):

  1. Bevacizumab in Colorectal Cancer: Current Role in Treatment and the Potential of Biosimilars.
    Rosen LS, Jacobs IA, Burkes RL. · · 2017 · cited 114× · PMID 28801849 · DOI 10.1007/s11523-017-0518-1
  2. Reviewing the role of healthy volunteer studies in drug development.
    Karakunnel JJ, Bui N, Palaniappan L, Schmidt KT, et al · · 2018 · cited 33× · PMID 30509294 · DOI 10.1186/s12967-018-1710-5
  3. A randomized, single-blind, Phase I trial (INVICTAN-1) assessing the bioequivalence and safety of BI 695502, a bevacizumab biosimilar candidate, in healthy subjects.
    Hettema W, Wynne C, Lang B, Altendorfer M, et al · · 2017 · cited 19× · PMID 28651442 · DOI 10.1080/13543784.2017.1347635

Verify or expand the search:

Other trials of BI 695502

Trials testing the same drug.

Other recruiting trials for Healthy

Currently open trials in the same condition.

Other Boehringer Ingelheim trials

Trials by the same sponsor.

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Data sources for this page

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing