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NCT00955773: Cancer

A Study of the GSK MEK Inhibitor GSK1120212 and Everolimus in Cancer Subjects

Completed Phase 1 Last updated 9 November 2017
What this trial tests

Phase 1 trial testing GSK1120212 plus everolimus in Cancer in 64 participants. Completed in 8 November 2011.

Timeline
17 August 2009
Primary endpoint
8 November 2011
8 November 2011

Quick facts

Lead sponsorGlaxoSmithKline
PhasePhase 1
StatusCompleted
Study typeINTERVENTIONAL
Allocationnon randomized
Designsingle group
Maskingnone
Primary purposetreatment
Enrollment64
Start date17 August 2009
Primary completion8 November 2011
Estimated completion8 November 2011
Sites3 locations across France, United States

Drugs / interventions tested

Conditions studied

Sponsor

GlaxoSmithKline — full company profile →

Who can join

18 and older, any sex, with Cancer. Patients with the condition only — healthy volunteers not accepted.

Sponsor's own description

The purpose of this study is to determine the recommended dose and regimen for the orally administered MEK inhibitor GSK1120212 dosed in combination with everolimus in subjects with solid tumors. The escalation part of the study will determine the MTD. The combination will be further explored in the expansion part in subjects with metastatic pancreatic cancer. In addition, subjects with KRAS mutant non-small cell lung cancer will be enrolled.

Publications & conference data

8 peer-reviewed publications reference this trial (live from Europe PMC):

  1. A central role for RAF→MEK→ERK signaling in the genesis of pancreatic ductal adenocarcinoma.
    Collisson EA, Trejo CL, Silva JM, Gu S, et al · · 2012 · cited 252× · PMID 22628411 · DOI 10.1158/2159-8290.cd-11-0347
  2. Molecularly targeted therapies in non-small-cell lung cancer annual update 2014.
    Morgensztern D, Campo MJ, Dahlberg SE, Doebele RC, et al · · 2015 · cited 106× · PMID 25535693 · DOI 10.1097/jto.0000000000000405
  3. A phase IB trial of the oral MEK inhibitor trametinib (GSK1120212) in combination with everolimus in patients with advanced solid tumors.
    Tolcher AW, Bendell JC, Papadopoulos KP, Burris HA, et al · · 2015 · cited 106× · PMID 25344362 · DOI 10.1093/annonc/mdu482
  4. Combating pancreatic cancer with PI3K pathway inhibitors in the era of personalised medicine.
    Conway JR, Herrmann D, Evans TJ, Morton JP, et al · · 2019 · cited 75× · PMID 30396902 · DOI 10.1136/gutjnl-2018-316822
  5. Targeting RAS mutants in malignancies: successes, failures, and reasons for hope.
    Yang H, Zhou X, Fu D, Le C, et al · · 2023 · cited 19× · PMID 36316602 · DOI 10.1002/cac2.12377
  6. Surgical and molecular considerations in the treatment of pediatric thalamopeduncular tumors.
    Lee RP, Foster KA, Lillard JC, Klimo P, et al · · 2017 · cited 15× · PMID 28686121 · DOI 10.3171/2017.4.peds16668
  7. Concurrent inhibition of pBADS99 synergistically improves MEK inhibitor efficacy in KRAS<sup>G12D</sup>-mutant pancreatic ductal adenocarcinoma.
    Tan YQ, Sun B, Zhang X, Zhang S, et al · · 2024 · cited 6× · PMID 38409090 · DOI 10.1038/s41419-024-06551-7
  8. Targeting <i>KRAS</i> in pancreatic adenocarcinoma: Progress in demystifying the holy grail.
    Elhariri A, Alhaj A, Ahn D, Sonbol MB, et al · · 2023 · cited 5× · PMID 37700806 · DOI 10.5306/wjco.v14.i8.285

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Data sources for this page

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