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NCT00693472

Study of Preladenant for the Treatment of Neuroleptic Induced Akathisia (Study P05145)

Terminated Phase 2 Results posted Last updated 7 November 2018
What this trial tests

Phase 2 trial testing Preladenant in Akathisia, Drug-Induced in 46 participants. Terminated before completion.

Timeline
15 August 2007
Primary endpoint
12 December 2008
9 January 2009

Quick facts

Lead sponsorMerck Sharp & Dohme LLC
PhasePhase 2
StatusTerminated
Study typeINTERVENTIONAL
Allocationrandomized
Designparallel
Maskingdouble
Primary purposetreatment
Enrollment46
Start date15 August 2007
Primary completion12 December 2008
Estimated completion9 January 2009

Drugs / interventions tested

Conditions studied

Sponsor

Merck Sharp & Dohme LLC — full company profile →

Who can join

Adults 18 to 65, any sex, with Akathisia, Drug-Induced or Antipsychotic Agents. Patients with the condition only — healthy volunteers not accepted.

Results — posted to ClinicalTrials.gov

Per-arm endpoint measurements with 95% confidence intervals where reported. Source: trial results section.

Part 1: Number of Participants With Akathisia Primary · Up to 13 days

Incidence of akathisia is reported as the number of participants who experienced akathisia. Akathisia is defined as a score of 3 on the Barnes akathisia scale (BAS) for 3 consecutive intervals or an akathisia score (BAS) of ≥4 for any single day, or the use of a rescue medication within 13 days of initiating treatment with haloperidol and preladenant. The BAS is scored as follows: objective akathisia, subjective awareness of restlessness and subjective distress related to restlessness are rated on a 4-point scale from 0 - 3 and are summed yielding a total score ranging from 0 (no akathisia) to

GroupValue95% CI
Part 1: Preladenant0
Part 1: Placebo0
Part 2: Number of Participants Who Were Treatment Failures Primary · Up to 14 days

Incidence of treatment failure is reported as the number of participants who were treatment failures. A treatment failure is defined as the failure to achieve at least a 1 point reduction from baseline in BAS score at 24 to 26 hours following study treatment. The BAS is scored as follows: objective akathisia, subjective awareness of restlessness and subjective distress related to restlessness are rated on a 4-point scale from 0 - 3 and are summed yielding a total score ranging from 0 (no akathisia) to 9 (severe akathisia).

GroupValue95% CI
Part 2: Preladenant4
Part 2: Standard of Care1
Part 1: Mean Global Clinical Impression at Day 14 Secondary · Day 14 of Part 1

Global clinical impression (GCI) was administered to assess whether any deterioration is due to akathisia or uncontrolled psychoses. Score on a scale +2 to -2 (+2 represents much improvement, +1 some improvement, 0 no change, -1 some worsening, and -2 much worsening).

GroupValue95% CI
Part 1: Preladenant0.9231± 0.7596
Part 1: Placebo1.7778± 0.4410
Part 1: Mean Positive and Negative Symptom Scale for Schizophrenia (PANSS) Total Score at Day 14 Secondary · Day 14 of Part 1

The PANSS is a 30-item clinician-rated instrument for assessing the symptoms of schizophrenia. It consists of 3 subscales: positive subscale (7 items), negative subscale (7 items), and general psychopathology subscale (16 items). Positive symptoms refer to an excess or distortion of normal mental status (e.g., delusions). Negative symptoms represent a diminution or loss of normal functions (e.g., emotional withdrawal). For each item, symptom severity was rated on a 7-point scale, from 0=absent to 6=extreme. The PANSS total score for each participant was calculated as the sum of the rating ass

GroupValue95% CI
Part 1: Preladenant38.4615± 19.4834
Part 1: Placebo36.3333± 17.0587
Part 2: Mean GCI at Day 14 Secondary · Day 14 of Part 2

The GCI was administered to assess whether any deterioration is due to akathisia or uncontrolled psychoses. Score on a scale +2 to -2 (+2 represents much improvement, +1 some improvement, 0 no change, -1 some worsening, and -2 much worsening).

GroupValue95% CI
Part 2: Preladenant0.6667± 1.0328
Part 2: Standard of Care2.0000± 0.0000
Part 2: PANSS Total Score at Day 14 Secondary · Day 14 of Part 2

The PANSS is a 30-item clinician-rated instrument for assessing the symptoms of schizophrenia. It consists of 3 subscales: positive subscale (7 items), negative subscale (7 items), and general psychopathology subscale (16 items). Positive symptoms refer to an excess or distortion of normal mental status (e.g., delusions). Negative symptoms represent a diminution or loss of normal functions (e.g., emotional withdrawal). For each item, symptom severity was rated on a 7-point scale, from 0=absent to 6=extreme. The PANSS total score for each participant was calculated as the sum of the rating assi

GroupValue95% CI
Part 2: Preladenant43.5000± 28.5430
Part 2: Standard of Care27.75± 11.2361

Adverse events — posted to ClinicalTrials.gov

Time frame: Up to 22 days (including follow-up). Reporting threshold: 5%. Adverse-event reports describe events observed during the trial — not all are caused by the drug.

Part 1: Placebo
Serious: 0/13 (0%)
Deaths:
Part 1: Preladenant
Serious: 0/19 (0%)
Deaths:
Part 2: Standard of Care
Serious: 0/6 (0%)
Deaths:
Part 2: Preladenant
Serious: 0/8 (0%)
Deaths:
Other adverse events (49 terms — click to expand)

ReactionSystemPart 1: PlaceboPart 1: PreladenantPart 2: Standard of CarePart 2: Preladenant
DIZZINESSNervous system disorders
HEADACHENervous system disorders
TREMORNervous system disorders
EXTRAPYRAMIDAL DISORDERNervous system disorders
SOMNOLENCENervous system disorders
NEUTROPENIABlood and lymphatic system disorders
TACHYCARDIACardiac disorders
CONJUNCTIVAL HYPERAEMIAEye disorders
ABDOMINAL PAIN UPPERGastrointestinal disorders
CONSTIPATIONGastrointestinal disorders
SALIVARY HYPERSECRETIONGastrointestinal disorders
VOMITINGGastrointestinal disorders
FATIGUEGeneral disorders
MALAISEGeneral disorders
ABSCESS ORALInfections and infestations
RHINITISInfections and infestations
TINEA PEDISInfections and infestations
TONSILLITISInfections and infestations
UPPER RESPIRATORY TRACT INFECTIONInfections and infestations
SKIN LACERATIONInjury, poisoning and procedural complications
SOFT TISSUE INJURYInjury, poisoning and procedural complications
ALANINE AMINOTRANSFERASE INCREASEDInvestigations
ASPARTATE AMINOTRANSFERASE INCREASEDInvestigations
LIVER FUNCTION TEST ABNORMALInvestigations
NEUTROPHIL COUNT DECREASEDInvestigations
WEIGHT INCREASEDInvestigations
BACK PAINMusculoskeletal and connective tissue disorders
JOINT STIFFNESSMusculoskeletal and connective tissue disorders
MUSCLE SPASMSMusculoskeletal and connective tissue disorders
MUSCULOSKELETAL STIFFNESSMusculoskeletal and connective tissue disorders
MYALGIAMusculoskeletal and connective tissue disorders
NECK PAINMusculoskeletal and connective tissue disorders
PAIN IN JAWMusculoskeletal and connective tissue disorders
AKATHISIANervous system disorders
COGWHEEL RIGIDITYNervous system disorders
DISTURBANCE IN ATTENTIONNervous system disorders
DYSKINESIANervous system disorders
DYSTONIANervous system disorders
HEAD TITUBATIONNervous system disorders
HYPERTONIANervous system disorders

Data from ClinicalTrials.gov NCT00693472 adverse events section.

Sponsor's own description

This study is designed to evaluate the effectiveness of preladenant in the prevention (Part 1) or treatment (Part 2) of antipsychotic induced akathisia in participants with acute psychosis using the Barnes Akathisia Scale.

Publications & conference data

1 peer-reviewed publication reference this trial (live from Europe PMC):

  1. The Adenosinergic System as a Therapeutic Target in the Vasculature: New Ligands and Challenges.
    Sousa JB, Diniz C. · · 2017 · cited 17× · PMID 28481238 · DOI 10.3390/molecules22050752

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