What drugs target RyR2?

1+ drugs target RyR2, including .

What drug classes act on RyR2?

Drug classes acting on RyR2 include Ryanodine receptor 2 inhibitor.

RyR2 — Drug Target

Name: Drug Landscape Pharmaceutical Database
Creator: Drug Landscape
Published: 2026-01-01
License: https://creativecommons.org/licenses/by/4.0/

1 drugs

All drugs that target RyR2 — marketed and clinical-stage. Includes 1 drug classes acting on this target.

Drug classes

Ryanodine receptor 2 inhibitor

Phase 2 pipeline (1)

GSK256066 · GlaxoSmithKline · Ryanodine receptor 2 inhibitor · Cardiovascular
GSK256066 is a selective and potent inhibitor of the cardiac ryanodine receptor 2.